santa cruz biotechnology, inc.
SCBT Logo

Willkommen!        Produkt(e) im Warenkorb.     Bestellen
 

Neurotransmitters and Drugs

  • 1-(α,α,α-Trifluoro-m-tolyl)piperazine
    Serotonin receptor agonist which has preference for 5-HT1B serotonin receptors.
    Katalog #CAS NummerSummenformelMenge
    sc-25386915532-75-9C11H13F3N25 g
  • 1-Deoxyforskolin from Coleus forskohlii
    Katalog #CAS NummerSummenformelMenge
    sc-22978672963-77-0C22H34O61 mg
  • 1-Methyl-4-(2'-methylphenyl)-1,2,3,6-tetrahydropyridine hydrochloride
    Dopaminergic neurotoxin displaying higher toxicity than MPTP in mice.
    Katalog #CAS NummerSummenformelMenge
    sc-251522102417-86-7C13H18ClN10 mg
  • 1-Methylhistamine dihydrochloride
    Histaming metabolite obtained from histamine N-methyltransferase.
    Katalog #CAS NummerSummenformelMenge
    sc-2588206481-48-7C6H11N3 ·2HCl25 mg
  • 1-Methylnicotinamide chloride
    Niacin metabolite excreted via the urinary system.
    Katalog #CAS NummerSummenformelMenge
    sc-2375831005-24-9C7H9N2OCl1 g
  • 1-Phenyl-1,3,8-triazaspiro[4.5]decan-4-one
    Katalog #CAS NummerSummenformelMenge
    sc-2539461021-25-6C13H17N3O5 g
  • (1,2,5,6-Tetrahydropyridin-4-yl)methylphosphinic acid hydrate
    A hybrid of isoguvacine and 3-APMPA designed to retain affinity for GABAC receptors but not to interact with GABAA or GABAB receptors.
    Katalog #CAS NummerSummenformelMenge
    sc-251571182485-36-5 (anhydrous)C6H12NO2P ·H2O10 mg
  • 1,3-Dimethyl-8-phenylxanthine
    Selective A1 adenosine receptor antagonist.
    Katalog #CAS NummerSummenformelMenge
    sc-253981961-45-5C13H12N4O2100 mg
  • 1,4-Dihydro-2,6-dimethyl-4-(3-nitrophenyl)-3,5-pyridinedicarboxylic Acid 3-Methyl Ester
    Derivative of 1,4-dihydropyridine used in the therapy and prevention of atherosclerotic degradation of arterial walls.
    Katalog #CAS NummerSummenformelMenge
    sc-21352974936-72-4C16H16N2O6100 mg
  • (1R,9S)-(−)-β-Hydrastine
    Katalog #CAS NummerSummenformelMenge
    sc-352027118-08-1C21H21NO6250 mg
  • 2-((3-Trifluoromethyl)phenyl)histamine dimaleate
    Found to be the most potent and selective H1 histamine receptor agonist of a panel of compounds in functional in vitro studies on histamine H2, H3, and other neurotransmitter receptors. It showed better potency at the guinea pig H1 histamine receptor than at the human H1 histamine receptor (pKi : 5.9). The selectivity of 2-((3-Trifluoromethyl)phenyl)histamine dimaleate was found to be 2138 (H1:H2), > 64 (H1:H3), 1000 (H1:M3), 105 (H1: a1), 708 (H1:β1), and 71 (H1:5HT2A). This substance does not cross the blood-brain barrier.
    Katalog #CAS NummerSummenformelMenge
    sc-251656162049-83-4C20H20F3N3O85 mg
  • 2-(Methylthio)adenosine 5'-diphosphate trisodium salt hydrate
    A P2 purinoceptor agonist, which induces platelet aggregation and shape change and inhibits cyclic AMP accumulation in platelets exposed to prostaglandin E1. Compared with ADP, 2-methylthio-ADP was 3 to 5 times as active as an aggregating agent and 150 to 200 times as active as an inhibitor of cyclic AMP accumulation. Purinergic signaling may be an important factor in TSP-1-mediated cell-matrix and cell-cell interactions such as those occurring during development and repair.
    Katalog #CAS NummerSummenformelMenge
    sc-251675475193-31-8 (anhydrous)C11H14N5Na3O10P2S•xH2O5 mg
  • 2-(Methylthio)adenosine 5'-triphosphate tetrasodium salt hydrate
    2-Methylthioadenosine triphosphate is a potent P2Y purinoceptor agonist
    Katalog #CAS NummerSummenformelMenge
    sc-287618n.n.C11H14N5Na4O13P3S•xH2O5 mg
  • (±)-2-Amino-6,7-dihydroxy-1,2,3,4-tetrahydronaphthalene hydrobromide
    A dopamine receptor agonist.
    Katalog #CAS NummerSummenformelMenge
    sc-25169313575-86-5C10H13NO2•HBr10 mg/25 mg
  • 2-Chloro-N6-cyclopentyladenosine hemihydrate
    Highly selective A1 adenosine receptor agonist.
    Katalog #CAS NummerSummenformelMenge
    sc-25173237739-05-2 (anhydrous)C15H20ClN5O4•0.5 ·H2O10 mg
  • 2-Chloroadenosine triphosphate tetrasodium hydrate
    P2Y purinoceptor agonist.
    Katalog #CAS NummerSummenformelMenge
    sc-288070n.n.C10H11ClN5Na4O13P3•xH2O5 mg
  • 2-Ethylidene-1,5-dimethyl-3,3-diphenylpyrrolidine perchlorate
    Metabolite of methadone. A useful marker in GC-MS analyses.
    Katalog #CAS NummerSummenformelMenge
    sc-25174766729-78-0C20H23N•HClO410 mg
  • 2-Methylserotonin maleate salt
    5-HT3 serotonin receptor agonist.
    Katalog #CAS NummerSummenformelMenge
    sc-25178778263-91-9C11H14N2O•C4H4O450 mg
  • 3-(1H-Imidazol-4-yl)propyl di(p-fluorophenyl)methyl ether hydrochloride
    H3 histamine receptor antagonist.
    Katalog #CAS NummerSummenformelMenge
    sc-298704n.n.C19H18F2N2O•HCl10 mg
  • 3-(N-Acetylamino)-5-(N-decyl-N-methylamino)benzyl alcohol
    Designed PKC activator, demonstrating an increase in the surface expression of BCA 225, a tumor-associated antigen, and various other cellular antigens in T47D cells.
    Katalog #CAS NummerSummenformelMenge
    sc-251920103955-90-4C20H34N2O21 mg
  • 3-Amino-1-propanesulfonic acid sodium salt
    GABAA receptor agonist.
    Katalog #CAS NummerSummenformelMenge
    sc-25193781028-90-2C3H8NO3SNa1 g
  • 3-Hydroxy-4-methoxyphenethylamine hydrochloride
    A dopamine metabolite.
    Katalog #CAS NummerSummenformelMenge
    sc-256512645-33-0C9H13NO2•HCl25 mg/100 mg
  • 3-Methoxytyramine hydrochloride
    This is a major metabolite of dopamine; a product of catechol O-methyltransferase.
    Katalog #CAS NummerSummenformelMenge
    sc-2545001477-68-5CH3OC6H3-4-(OH)CH2CH2NH2··HCl100 mg
  • 3-Propylxanthine
    Weak competitor antagonist at both A1 and A2 adenosine receptors.
    Katalog #CAS NummerSummenformelMenge
    sc-25203541078-02-8C8H10N4O225 mg/250 mg
  • 3,4-Dihydroxy-DL-phenylalanine
    Immediate precursor of dopamine. Product of tyrosine hydroxylase.
    Katalog #CAS NummerSummenformelMenge
    sc-25658463-84-3C9H11NO41 g/5 g
  • 3,5,5,-Trimethyloxazolidine-2,4-dione
    Katalog #CAS NummerSummenformelMenge
    sc-232150127-48-0C6H9NO31 g
  • [3S-(3α,4aβ,8aβ)]-N-(tert-Butyl)decahydro-3-isoquinolinecarboxamide
    Fragment present in various HIV-1 protease inhibitors currently in clinical trials for AIDS treatment.
    Katalog #CAS NummerSummenformelMenge
    sc-209788136465-81-1C14H26N2O1 g
  • 3α,21-Dihydroxy-5α-pregnan-20-one
    Positive allosteric modulator of GABAA receptors.
    Katalog #CAS NummerSummenformelMenge
    sc-252069567-02-2C21H34O35 mg
  • 4-Aminomethylbenzenesulfonamide hydrochloride
    Katalog #CAS NummerSummenformelMenge
    sc-226489138-37-4C7H10N2O2S ·HCl25 g
  • 4-Deoxypyridoxine hydrochloride
    Vitamin B6 antagonist.
    Katalog #CAS NummerSummenformelMenge
    sc-238830148-51-6C8H11NO2•HCl500 mg
  • 4-Diphenylacetoxy-N-(2-chloroethyl)piperidine hydrochloride
    An irreversible muscarinic acetylcholine receptor antagonist with essentially equivalent affinity for M1, M3, M4, and M5 receptors and a much lower affinity for M2 receptors.
    Katalog #CAS NummerSummenformelMenge
    sc-252148130817-71-9C21H24ClNO2•HCl25 mg/100 mg
  • (±)4-Hydroxydebrisoquin
    A major metabolite of debrisoquin. It is a very useful indicator for cytochrome P-450 polymorphism.
    Katalog #CAS NummerSummenformelMenge
    sc-20072959333-79-8C10H13N3O10 mg/50 mg
  • 4-Phenylbenzaldoxime
    Katalog #CAS NummerSummenformelMenge
    sc-23295840143-27-9C13H11NO1 g
  • 5-Carboxamidotryptamine maleate salt hemiethanolate
    An agonist at 5-HT1A, 5-HT1B, 5-HT1D, 5-HT5 and 5-HT7 serotonin receptors.
    Katalog #CAS NummerSummenformelMenge
    sc-25225874885-72-6C11H13N3O ·0.5 ·C2H6O ·C4H4O45 mg
  • 5-Hydroxyindole-3-acetic acid
    A major serotonin metabolite.
    Katalog #CAS NummerSummenformelMenge
    sc-25692154-16-0C10H9NO3100 mg/500 mg
  • 5-Hydroxyindole-3-acetic acid (dicyclohexylammonium) salt
    Major serotonin metabolite.
    Katalog #CAS NummerSummenformelMenge
    sc-25692266866-39-5C22H32N2O3100 mg
  • 5-Methylurapidil
    Selective α1A-adrenoceptor antagonist that exhibits antihypertensive properties.
    Katalog #CAS NummerSummenformelMenge
    sc-25485534661-85-3C21H31N5O310 mg/50 mg
  • 5α-Pregnane-3,11,20-trione
    Katalog #CAS NummerSummenformelMenge
    sc-2270312089-06-7C21H30O350 mg
  • 6-Acetyl-7-deacetylforskolin
    Antihypertensive also exhibiting positive ionotropic and adenyl cyclase activating properties.
    Katalog #CAS NummerSummenformelMenge
    sc-26276664657-21-2C22H34O71 mg
  • 6-Nitroquipazine maleate salt
    A potent and selective serotonin transport blocker.
    Katalog #CAS NummerSummenformelMenge
    sc-25230177372-73-7C17H18N4O6100 mg
  • 7-Benzyloxytryptamine
    Katalog #CAS NummerSummenformelMenge
    sc-23911731677-75-5C17H18N2O100 mg
  • 7-Deacetyl-1-deoxyforskolin from Coleus forskohlii
    Katalog #CAS NummerSummenformelMenge
    sc-233676121606-18-6C20H32O51 mg
  • (±)-7-Hydroxy-2-(di-n-propylamino)tetralin hydrobromide
    A selective D3 dopamine receptor agonist; has a much weaker affinity for other dopamine receptor subtypes.
    Katalog #CAS NummerSummenformelMenge
    sc-252308159795-63-8C16H25NO•HBr25 mg
  • 8-Bromoadenosine 5'-triphosphate sodium salt
    P2X purinoceptor agonist with similar reactivity to ATP.
    Katalog #CAS NummerSummenformelMenge
    sc-25231281035-56-5C10H15BrN5O13P3•Na5 mg
  • 9-Deoxyforskolin from Coleus forskohlii
    Katalog #CAS NummerSummenformelMenge
    sc-23372684048-28-2C22H34O61 mg
  • 12β-Hydroxydigitoxin
    This compound is a cardiac glycoside which serves as a substrate for Pgp. It upregulates Pgp expression and down regulates SXR (Steroid Xenobiotic Receptor).
    Katalog #CAS NummerSummenformelMenge
    sc-21360420830-75-5C41H64O141 g/5 g
  • α-Hydroxy-triazolam
    Metabolite of triazolam.
    Katalog #CAS NummerSummenformelMenge
    sc-222434n.n.C17H12Cl2N4O1 mg
  • α-Methylserotonin maleate salt
    A salt of α-Methylserotonin maleate and a serotonin receptor agonist.
    Katalog #CAS NummerSummenformelMenge
    sc-25492997469-12-0C11H14N2O ·C4H4O410 mg/50 mg
  • α5IA
    A selective inverse agonist for a5 subtype of GABAA receptor with a higher intrincing efficacy to the a5 subtype than other drugs.
    Katalog #CAS NummerSummenformelMenge
    sc-252345215874-86-5C17H14N8O25 mg
  • A-315456
    A selective α1D-adrenoceptor antagonist.
    Katalog #CAS NummerSummenformelMenge
    sc-300143n.n.C18H23N3O2S5 mg
  • A-317491 sodium salt hydrate
    A non-nucleotide P2X3 and P2X2/3 receptor antagonist, which inhibits calcium flux mediated by the receptors. This compound can also bind to 86 other receptors, enzymes, and ion channels.
    Katalog #CAS NummerSummenformelMenge
    sc-300144n.n.C33H27NO8•xNa+•yH2O5 mg
  • A-331440 dihydrochloride
    A non-imidazole H3 histamine receptor antagonist. Presynaptic histamine H3 receptors regulate the release of histamine and other neurotransmitters, and histamine H3receptor antagonists enhance neurotransmitter release. A-331440 is a histamine H(3) receptor antagonist, which binds strongly and selectively to both human and rat histamine H3 receptors (K(i)=25 nM). Mice on a high-fat diet (45 kcal % lard) prior to 28-day oral b.i.d. dosing for measurement of obesity-related parameters. A-331440 administered at 0.5 mg/kg had no significant effect on weight, whereas 5 mg/kg decreased weight comparably to dexfenfluramine (10 mg/kg). A-331440 administered at 15 mg/kg reduced weight to a level comparable to mice on the low-fat diet. The two higher doses reduced body fat and the highest dose also normalized an insulin tolerance test. Both data shows that the histamine H3 receptor antagonist, A-331440, has potential as an antiobesity agent.
    Katalog #CAS NummerSummenformelMenge
    sc-252330392338-13-5 (non-salt)C22H27N3O•2HCl5 mg
  • Acamprosate Calcium
    It is of interest for the treatment of alcoholism and other neurochemical disorders.
    Katalog #CAS NummerSummenformelMenge
    sc-21073377337-73-6C10H20CaN2O8S2100 mg
  • Acetyl Coenzyme A Trilithium Salt Trihydrate
    Acetyl coenzyme A is an essential cofactor and carrier of acyl groups in enzymatic acetyl transfer reactions. Also the precursor for lipid biosynthesis and the neurotransmitter acetylcholine.
    Katalog #CAS NummerSummenformelMenge
    sc-29179472-89-9C23H35Li3N7O17P3S ·3H2O1 mg/5 mg
  • Acetyl-β-methylcholine chloride
    Metabolically stable analog of acetylcholine; muscarinic agonist. Its ability to constrict airway smooth muscle is used to assess bronchial reactivity in the laboratory and clinically.
    Katalog #CAS NummerSummenformelMenge
    sc-25706362-51-1C8H18ClNO25 g/25 g
  • Acetylcholine bromide
    This is an endogenous neurotransmitter at cholinergic synapses, which amplifies action potential of the sarcolemma thereby inducing muscle contractions.
    Katalog #CAS NummerSummenformelMenge
    sc-25235066-23-9C7H16BrNO2100 g
  • Acetylcholine perchlorate
    Katalog #CAS NummerSummenformelMenge
    sc-233810927-86-6C7H16NO2•O4Cl5 g
  • Acetylthiocholine chloride
    An acetylcholinesterase substrate and nicotinic acetylcholine receptor agonist.
    Katalog #CAS NummerSummenformelMenge
    sc-2570666050-81-3C7H16ClNOS1 g
  • Adenosine amine congener hydrate
    Potent aqueous-soluble A1 adenosine receptor agonist.
    Katalog #CAS NummerSummenformelMenge
    sc-25493896760-69-9 (anhydrous)C28H32N8O6•xH2O5 mg
  • Adiphenine hydrochloride
    Katalog #CAS NummerSummenformelMenge
    sc-23382150-42-0C20H25NO2•HCl10 g
  • Alaproclate hydrochloride
    Strong and selective serotonin uptake inhibitor.
    Katalog #CAS NummerSummenformelMenge
    sc-25707560719-83-7C13H18ClNO2•HCl25 mg
  • Altanserin hydrochloride hydrate
    This is a specific 5HT2/serotonergic antagonist.
    Katalog #CAS NummerSummenformelMenge
    sc-25236576330-71-7 (non-salt)C22H22FN3O2S•HCl•xH2O10 mg
  • ALX-1393
    Inhibitor of the glycine transporter GlyT-2.
    Katalog #CAS NummerSummenformelMenge
    sc-300191n.n.C23H22NO4F500 µg
  • Amcinonide
    Katalog #CAS NummerSummenformelMenge
    sc-22724551022-69-6C28H35FO71 g
  • Amodiaquin dihydrochloride dihydrate
    Katalog #CAS NummerSummenformelMenge
    sc-2338706398-98-7C20H22ClN3O•2HCl•2H2O5 g
  • Antazoline phosphate salt
    An imidazoline agonist that is more potent than efaroxan in inducing insulin release from β cells; H1 histamine receptor antagonist.
    Katalog #CAS NummerSummenformelMenge
    sc-239251154-68-7C17H22N3O4P1 g
  • Ara-G hydrate
    An inducer of apoptosis inhibitor of DNA synthesis antimetabolite and antineoplastic. Ara-G is converted by cellular kinases to the active 5'-triphosphate, Ara-GTP. Incorporation of Ara-GTP into DNA leads to inhibition of DNA synthesis and apoptosis. The cellular accumulation of Ara-GTP is indicative of the clinical response to treatment with nelarabine, the prodrug. The differential accumulation and consequent selective cytotoxicity of Ara-G in T cells has been postulated to be due to the higher accumulation and slower elimination of ara-GTP in these cells. Nelarabine was developed because of poor water solubility of Ara-G, but Ara-G is DMSO-soluble. Nelarabine is approved in the United States for the treatment of T-cell acute lymphoblastic leukemia (T-ALL) and T-cell lymphoblastic lymphoma (T-LBL).
    Katalog #CAS NummerSummenformelMenge
    sc-21454838819-10-2 (anhydrous)C10H13N5O5 ·xH2O5 mg/25 mg
  • Arecaidine hydrochloride
    Katalog #CAS NummerSummenformelMenge
    sc-2338896018-28-6C7H11NO2 ·HCl100 mg
  • Arecaidine propargyl ester hydrobromide
    A potent muscarinic acetylcholine receptor agonist exhibiting slight selectivity for M2 receptors; inactive at nicotinic receptors.
    Katalog #CAS NummerSummenformelMenge
    sc-257091116511-28-5C10H13NO2•HBr25 mg
  • Atropine
    Competitive nonselective antagonist at central and peripheral muscarinic acetylcholine receptors.
    Katalog #CAS NummerSummenformelMenge
    sc-25239251-55-8C17H23NO35 g
  • AZ11645373
    A selective and potent human P2X7 purinoceptor antagonist.
    Katalog #CAS NummerSummenformelMenge
    sc-252394227088-94-0C24H21N3O5S5 mg
  • β, γ-Methyleneadenosine 5'-triphosphate disodium salt
    Selective P2X purinoceptor agonist which is more potent than ATP and less potent than α, β-methylene-L-adenosine 5'-triphosphate.
    Katalog #CAS NummerSummenformelMenge
    sc-2530427414-56-4C11H16N5O12P3 ·2Na5 mg/10 mg
  • B-HT 933 dihydrochloride
    A selective α2-adrenoceptor agonist.
    Katalog #CAS NummerSummenformelMenge
    sc-25495136067-72-8C9H15N3O•2HCl5 mg
  • Bamethane hemisulfate salt
    Katalog #CAS NummerSummenformelMenge
    sc-2339085716-20-1HOC6H4CH(OH)CH2NH(CH2)3CH3•1/2H2SO45 g
  • Benazoline oxalate salt
    I2 imidazoline receptor agonist; has high affinity and selectivity for I2 imidazoline receptors over α-adrenoceptors.
    Katalog #CAS NummerSummenformelMenge
    sc-2571191021868-82-5C13H12N2•C2H2O45 mg
  • Bendroflumethiazide
    Katalog #CAS NummerSummenformelMenge
    sc-23392873-48-3C15H14F3N3O4S21 g
  • Benfotiamine
    Lipid-soluble thiamine derivative used as a treatment for diabetic neuropathy. More effective at increasing thiamin levels in blood and tissues than water-soluble salts like the previous vitamin B1.
    Katalog #CAS NummerSummenformelMenge
    sc-20463922457-89-2C19H23N4O6PS250 mg/1 g
  • Benoxathian hydrochloride
    Selective α1-adrenoceptor antagonist.
    Katalog #CAS NummerSummenformelMenge
    sc-25495492642-97-2C19H23NO4S•HCl10 mg
  • Benzbromarone
    Katalog #CAS NummerSummenformelMenge
    sc-2339343562-84-3C17H12Br2O31 g
  • Bephenium hydroxynaphthoate
    Katalog #CAS NummerSummenformelMenge
    sc-2340123818-50-6C17H22NO•C11H7O310 g
  • Bicyclol
    A anti-hepatitis drug, used in China for chronic hepatitis B and presumably C. The drug appears to protect against liver injury in animals. Recently was reported that bicyclol induces the expression of hepatic HSP27 and HSP70, and consequently inhibits the transcription factor NF-?B-mediated apoptosis and necrosis in liver tissue. It appears that bicyclol induces hepatic HSP27 and HSP70 expression through the activation transcription of HSPs genes.
    Katalog #CAS NummerSummenformelMenge
    sc-252435118159-48-1C19H18O95 mg
  • Bilobalide
    Bilobalide is a terpenoid extracted from ginkgo biloba with neuroprotective, antibacterial, and inhibitory effects.
    Katalog #CAS NummerSummenformelMenge
    sc-20106133570-04-6C15H18O810 mg/50 mg
  • BRL 35135A
    BRL 35135A is an agonist for the β3-adrenoceptor.
    Katalog #CAS NummerSummenformelMenge
    sc-300301n.n.C20H25BrClNO425 mg
  • BRL 37344 sodium salt hydrate
    A selective β3-adrenoceptor agonist. Studies support the hypothesis that there are peripheral β3 adrenergic receptors that can reduce food intake and that central β2 or β3 adrenergic receptors mediate the peripheral effects of the β3 agonist.
    Katalog #CAS NummerSummenformelMenge
    sc-252513127299-93-8 (anhydrous)C19H21ClNNaO4•xH2O5 mg
  • BU224 hydrochloride
    BU224 hydrochloride is an antagonist for the I2 Imidazoline receptor.
    Katalog #CAS NummerSummenformelMenge
    sc-300306187173-05-3C12H11N3•HCl5 mg
  • Bufexamac
    Katalog #CAS NummerSummenformelMenge
    sc-2275372438-72-4C12H17NO310 g
  • Buflomedil hydrochloride
    Katalog #CAS NummerSummenformelMenge
    sc-23422535543-24-9C17H25NO4•HCl1 g
  • Bupivacaine hydrochloride
    Na+ channel blocker, local anesthetic.
    Katalog #CAS NummerSummenformelMenge
    sc-25252418010-40-7C18H28N2O··HCl1 g/5 g
  • Butacaine
    Katalog #CAS NummerSummenformelMenge
    sc-234227149-16-6C18H30N2O21 g
  • (±)-Butaclamol hydrochloride
    Katalog #CAS NummerSummenformelMenge
    sc-23422836504-94-6C25H31NO•HCl25 mg
  • (-)-Butaclamol hydrochloride
    Dopamine receptor antagonist; less active enantiomer.
    Katalog #CAS NummerSummenformelMenge
    sc-25252655528-08-0C25H31NO•HCl25 mg
  • (+)-Butaclamol hydrochloride
    A dopamine D2 receptor antagonist. This compound is 2 to 4 times more active than its enantiomer at inhibiting the D2 receptor.
    Katalog #CAS NummerSummenformelMenge
    sc-25252555528-07-9C25H31NO•HCl5 mg
  • Butethamate citrate salt
    Katalog #CAS NummerSummenformelMenge
    sc-22754013900-12-4C16H25NO2 ·C6H8O75 g
  • Butoxamine hydrochloride
    Katalog #CAS NummerSummenformelMenge
    sc-2342335696-15-1C15H25NO3 ·HCl50 mg
  • Camylofine dihydrochloride
    Katalog #CAS NummerSummenformelMenge
    sc-23427554-30-8C19H32N2O2•2HCl1 g
  • Carbamyl-β-methylcholine chloride
    Katalog #CAS NummerSummenformelMenge
    sc-234279590-63-6C7H17N2O2Cl5 g
  • Carprofen
    A non-steroidal anti-inflammatory drug whose mechanism of action is dependent upon inhibiting the production of cox-2 and other sources of prostaglandins
    Katalog #CAS NummerSummenformelMenge
    sc-20562153716-49-7C15H12ClNO21 g/5 g
  • CAY10415
    Potent antidiabetic drug that, when adminstered as a food admixture at 100 mg/kg for four days, effectively lowers blood glucose levels in obese, hyperglycemic, hyperinsulinemic, and insulin-resistant KKAy mice. Also shown to enhance the rate of insulin-stimulated lipogenesis in 3T3-L1 adipocytes in a dose-dependent manner.
    Katalog #CAS NummerSummenformelMenge
    sc-205236146062-49-9C19H18N2O4S1 mg/10 mg
  • Cefadroxil
    Katalog #CAS NummerSummenformelMenge
    sc-23429150370-12-2C16H17N3O5S1 g
  • Cerivastatin Lactone
    Synthesized statin used to lower cholesterol and prevent cardiovascular disease.
    Katalog #CAS NummerSummenformelMenge
    sc-204679145599-86-6C26H32FNO45 mg/10 mg
  • CGP 35348 hydrate
    A GABAB-receptor antagonist.
    Katalog #CAS NummerSummenformelMenge
    sc-252561123690-79-9 (non-salt)C8H20NO4P•xH2O5 mg
  • CGS-21680 hydrochloride hydrate
    An adenosine receptor agonist that possesses selectivity for A2 verses A1 receptors.
    Katalog #CAS NummerSummenformelMenge
    sc-252562124182-57-6 (anhydrous)C23H29N7O6•HCl•xH2O5 mg/10 mg
  • Chloro-APB hydrobromide
    Full D1 dopamine receptor agonist.
    Katalog #CAS NummerSummenformelMenge
    sc-25257380751-65-1C19H20ClNO2•HBr5 mg/25 mg
  • Chlorocitalopram
    This compound is an internal standard of Citalopram, as well as an uptake inhibitor of serotonin (5-HT).
    Katalog #CAS NummerSummenformelMenge
    sc-20742364169-57-9C20H21ClN2O1 mg
  • Chlorocitalopram, Hydrobromide
    An internal standard of Citalopram which is also an uptake inhibitor of serotonin (5-HT).
    Katalog #CAS NummerSummenformelMenge
    sc-20742464169-58-0C20H22BrClN2O1 mg
  • Chloroethylclonidine dihydrochloride
    An rreversible α1B-adrenoceptor alkylating agent.
    Katalog #CAS NummerSummenformelMenge
    sc-25258798086-36-3C13H17Cl3N4•2HCl10 mg/25 mg
  • Chloropyramine hydrochloride
    Katalog #CAS NummerSummenformelMenge
    sc-2343456170-42-9C16H20ClN3•HCl1 g
  • Chlorzoxazone
    Muscle relaxant (skeletal).
    Katalog #CAS NummerSummenformelMenge
    sc-21107895-25-0C7H4ClNO210 mg
  • Choline bitartrate
    Acyl group acceptor
    Katalog #CAS NummerSummenformelMenge
    sc-25259987-67-2C9H19NO7100 g
  • CI 1020
    Highly selective, orally active, non-peptide endothelin-A receptor (ETA) antagonist (IC50 values are 0.3 and 480 nM for ETA and ETB receptors respectively). Antihypertensive; blocks ET-1-induced pressor responses following oral administration.
    Katalog #CAS NummerSummenformelMenge
    sc-204687162256-50-0C28H26O910 mg/50 mg
  • Cinchonine hemisulfate salt
    Katalog #CAS NummerSummenformelMenge
    sc-2343605949-16-6C19H22N2O•1/2H2SO4100 g
  • Ciproxifan hydrochloride
    Ciproxifan belongs to a novel chemical series of histamine H3-receptor antagonists. In vitro, it behaved as a competitive antagonist at the H3 autoreceptor controlling 3H histamine release from synaptosomes and displayed similar Ki values (0.5-1.9 nM) at the H3 receptor controlling the electrically-induced contraction of guinea pig ileum or at the brain H3 receptor labeled with 125I-iodoproxyfan. This appears to be an orally bioavailable, extremely selective and potent H3-receptor antagonist whose vigilance- and attention-promoting effects are promising for therapeutic applications in aging disorders.
    Katalog #CAS NummerSummenformelMenge
    sc-2572451049741-81-2C16H18N2O2•HCl5 mg
  • Ciproxifan maleate
    Strong, selective H3 histamine receptor antagonist.
    Katalog #CAS NummerSummenformelMenge
    sc-252608184025-19-2C16H18N2O2•C4H4O45 mg
  • cis-Entacapone
    An antiparkinsonian (Z)-Isomer of Entacapone polymorphic form B.
    Katalog #CAS NummerSummenformelMenge
    sc-214739145195-63-7C14H15N3O52.5 mg
  • Cisapride monohydrate
    5-HT4 serotonin receptor agonist
    Katalog #CAS NummerSummenformelMenge
    sc-252619260779-88-2C23H29N3O4ClF•H2O10 mg
  • Clenbuterol Hydrochloride
    β2-adrenoreceptor agonist with ability to potentiate hyopxemia due to increased shunt fraction in horses anesthetized via IV. Has also been shown to enhance memory in sham-lesioned male Sprague Dawley rats.
    Katalog #CAS NummerSummenformelMenge
    sc-20563521898-19-1C12H18Cl2N2O ·HCl25 mg/100 mg
  • Clioquinol
    A metal chelating ligand and a member of the hydroxyquinoline family, which inhibits certain enzymes related to DNA replication.
    Katalog #CAS NummerSummenformelMenge
    sc-201066130-26-7C9H5ClINO1 g/5 g
  • Clofazimine
    Katalog #CAS NummerSummenformelMenge
    sc-2344022030-63-9C27H22Cl2N45 g
  • Clofibric acid
    A compound that reduces cholesterol levels in blood through diminishing the activity of NADPH.
    Katalog #CAS NummerSummenformelMenge
    sc-203000882-09-7C10H11ClO310 g/50 g
  • Clofoctol
    Katalog #CAS NummerSummenformelMenge
    sc-23440337693-01-9C21H26Cl2O1 g
  • Cloperastine hydrochloride
    Katalog #CAS NummerSummenformelMenge
    sc-23440514984-68-0C20H24ClNO•HCl10 g
  • Clozapine N-oxide
    Major metabolite of Clozapine (sc-200402). Observed to to decrease 5-HT2 serotonin receptor density in vitro.
    Katalog #CAS NummerSummenformelMenge
    sc-20111134233-69-7C18H19ClN4O5 mg/25 mg
  • Condelphine
    A nicotinic acetylcholine receptor antagonist.
    Katalog #CAS NummerSummenformelMenge
    sc-2526257633-69-4C25H39NO620 mg
  • Cyclazosin hydrochloride
    α1B-adrenoceptor antagonist.
    Katalog #CAS NummerSummenformelMenge
    sc-239599146929-33-1C23H27N5O4•HCl5 mg
  • Cysteamine S-phosphate sodium salt
    Katalog #CAS NummerSummenformelMenge
    sc-2344993724-89-8C2H7NO3PSNa50 mg
  • D-Tryptophan
    An unnatural isomer of tryptophan.
    Katalog #CAS NummerSummenformelMenge
    sc-255066153-94-6C11H12N2O25 g/25 g
  • DEABL
    Anticonvulsant; positive modulator of GABAA receptor
    Katalog #CAS NummerSummenformelMenge
    sc-252664175698-05-2C8H15NO50 mg
  • Deacetylforskolin
    Katalog #CAS NummerSummenformelMenge
    sc-23451664657-20-1C20H32O61 mg
  • Debrisoquin sulfate (Ro 5-3307)
    This is an antihypertensive. It is metabolized to 4-hydroxydebrisoquin by debrisoquin 4-hydroxylase. Useful indicator for cytochrome P-450 polymorphism.
    Katalog #CAS NummerSummenformelMenge
    sc-200725581-88-4C20H28N6O4S50 mg/500 mg
  • Delsoline
    Nicotinic receptor antagonist, ganglion blocker; exhibits weak affinity at brain α-bungarotoxin-sensitive nicotinic acetylcholine receptors.
    Katalog #CAS NummerSummenformelMenge
    sc-252666509-18-2C25H41NO720 mg
  • Desoximetasone
    Katalog #CAS NummerSummenformelMenge
    sc-234529382-67-2C22H29FO41 g
  • Despropionylfentanyl
    Katalog #CAS NummerSummenformelMenge
    sc-22153721409-26-7C19H24N21 mg/10 mg
  • Desvenlafaxine hydrochloride
    A dual SERT/NET reuptake inhibitor and a major active metabolite of venlafaxine. A brain penetrant.
    Katalog #CAS NummerSummenformelMenge
    sc-255071300827-87-6C16H25NO2•HCl10 mg
  • Diacerein
    An interleukin-1 inhibitor used for treating osteoarthritis.
    Katalog #CAS NummerSummenformelMenge
    sc-20471713739-02-1C19H12O850 mg/250 mg
  • Diaveridine
    A coccidiostat and antiprotozoal drug.
    Katalog #CAS NummerSummenformelMenge
    sc-2056465355-16-8C13H16N4O21 g/10 g
  • Diethylstilbestrol dipropionate
    Katalog #CAS NummerSummenformelMenge
    sc-227859130-80-3C24H28O41 g
  • Diflorasone diacetate
    Katalog #CAS NummerSummenformelMenge
    sc-22786133564-31-7C26H32F2O7100 mg
  • Dihydroergotamine (+)-tartrate salt
    Vasoconstrictor and vascular serotonin receptor agonist. Also exhibits alpha-adrenergic and dopamine D2 receptor partial agonist activity.
    Katalog #CAS NummerSummenformelMenge
    sc-2630915989-77-5(C33H37N5O5)2•C4H6O650 mg
  • Dihydrotachysterol
    Katalog #CAS NummerSummenformelMenge
    sc-23469567-96-9C28H46O50 mg
  • Dimenhydrinate
    Katalog #CAS NummerSummenformelMenge
    sc-234708523-87-5C17H21NO•C7H7ClN4O210 g
  • Diminazene Aceturate
    An anti-protozoal drug and anti-trypanosomal.
    Katalog #CAS NummerSummenformelMenge
    sc-205651908-54-3C14H15N7•2C4H7NO31 g/5 g
  • Diperodon hydrochloride
    Katalog #CAS NummerSummenformelMenge
    sc-234775537-12-2C22H27N3O4•HCl5 g
  • Dipyrone
    A non-steroidal anti-inflammatory drug that, when coadministered with morphine, potentiates its antinociceptive action and delays the development of tolerance. Dipyrone is a selective inhibitor of cyclooxygenase-3 (COX-3), with lower activity against COX-1 and no activity against COX-2. This also blocks PGE2-induced hyperalgesia in several models.
    Katalog #CAS NummerSummenformelMenge
    sc-25275568-89-3C13H16N3O4SNa25 g
  • Diquine
    A nicotinic cholinoreceptor antagonist at the neuromuscular junction which is a curare-like ganglioblocker.
    Katalog #CAS NummerSummenformelMenge
    sc-2551193563-63-1C34H50Cl2N22 mg
  • Dithiobiuret
    Paralytic agent.
    Katalog #CAS NummerSummenformelMenge
    sc-252760541-53-7C2H5N3S2100 mg
  • DL-threo-β-(3,4-Dihydroxyphenyl)serine
    An amino acid precursor of noradrenaline (NA); elevates the concentration of NA in the brain.
    Katalog #CAS NummerSummenformelMenge
    sc-2527643916-18-5C9H11NO51 g
  • Dothiepin hydrochloride
    Dothiepin hydrochloride is a tricyclic antidepressant.
    Katalog #CAS NummerSummenformelMenge
    sc-300503897-15-4C19H21NS ·HCl5 mg
  • Doxazosin Mesylate
    An alpha-blocker drug. It reduces progression of benign prostatic hyperplasia.
    Katalog #CAS NummerSummenformelMenge
    sc-20565677883-43-3C24H29N5O8S50 mg/250 mg
  • Drofenine hydrochloride
    Katalog #CAS NummerSummenformelMenge
    sc-234845548-66-3C20H31NO2•HCl10 g
  • (±)-Dropropizine
    Katalog #CAS NummerSummenformelMenge
    sc-23484617692-31-8C13H20N2O25 g
  • DS1
    Potently (low nM) enhances GABA-evoked currents mediated by α4β3δ receptors. It has little effect on GABA responses mediated by α4β3 2 receptors. At similar concentrations, DS1 directly activates this receptor and is the most potent known agonist of α4β3δ receptors. This compound has an opportunity to be become an agonist golden stardard for δ-GABAA receptors.
    Katalog #CAS NummerSummenformelMenge
    sc-252769372497-52-4C18H10Br2ClN3OS5 mg
  • Dyclonine, Hydrochloride
    Used as a local anesthetic.
    Katalog #CAS NummerSummenformelMenge
    sc-211385536-43-6C18H28ClNO225 g
  • Eletriptan Free Base
    Used in the treatment of migraine headaches.
    Katalog #CAS NummerSummenformelMenge
    sc-204736143322-58-1C22H26N2O2S1 mg/5 mg
  • (-)-Epinephrine
    A predominent neurotransmitter. Found to be effective beta2-agonist bronchodilator.
    Katalog #CAS NummerSummenformelMenge
    sc-20567451-43-4C9H13NO31 g/5 g
  • (±)-Epinephrine
    Katalog #CAS NummerSummenformelMenge
    sc-252779329-65-7C9H13NO35 g/25 g
  • (±)-Epinephrine hydrochloride
    Adrenergic receptor agonist.
    Katalog #CAS NummerSummenformelMenge
    sc-252780329-63-5C9H13NO3 ·HCl5 g
  • Etbicythionat
    A potent non-competitive GABA antagonist in mammals. Causes epileptiform seizures.
    Katalog #CAS NummerSummenformelMenge
    sc-252786224790-71-0C6H11O3PS100 µg
  • Ethylhydrocupreine
    Katalog #CAS NummerSummenformelMenge
    sc-235094522-60-1C21H28N2O25 g
  • Ethylhydrocupreine hydrochloride
    Sensitive and specific reagent for the identification of Streptococcus pneumoniae.
    Katalog #CAS NummerSummenformelMenge
    sc-2551663413-58-9n.n.100 mg/1 g
  • Famprofazone
    Katalog #CAS NummerSummenformelMenge
    sc-23512222881-35-2C24H31N3O10 g
  • FAUC 213
    A highly selective D4 dopamine receptor full antagonist.
    Katalog #CAS NummerSummenformelMenge
    sc-252820337972-47-1C18H19ClN45 mg
  • Fenoprofen calcium salt hydrate
    Katalog #CAS NummerSummenformelMenge
    sc-23998953746-45-5C30H26O6Ca. ·xH2O5 g
  • Fenoterol hydrobromide
    A β2-adrenoceptor agonist. Bronchodilator.
    Katalog #CAS NummerSummenformelMenge
    sc-2528221944-12-3C17H21NO4•HBr1 g
  • Fiduxosin hydrochloride
    Has been shown to be an α1-Adrenoceptor antagonist.
    Katalog #CAS NummerSummenformelMenge
    sc-300692208992-74-9C30H29N5O4S•HCl5 mg
  • Fipexide HCl
    Fipexide has been shown to be a nootropic agent and possible mild dopamine agonist.
    Katalog #CAS NummerSummenformelMenge
    sc-20106534161-23-4C20H21ClN2O4 ·HCl1 g
  • Fipexide hydrochloride
    Katalog #CAS NummerSummenformelMenge
    sc-23513634161-24-5C20H21ClN2O4•HCl5 g
  • Flucybene
    A potent non-competitive GABA antagonist in mammals, molluscs and insects; convulsant.
    Katalog #CAS NummerSummenformelMenge
    sc-2528253289-22-3C11H8F6N21 mg
  • Fluorocurarine chloride
    A short-acting selective sympathetic ganglioblocker with weak antagonist activity on the nicotinic receptor at the neuromuscular junction. Hypotensive.
    Katalog #CAS NummerSummenformelMenge
    sc-25282922273-09-2C20H23ClN2O20 mg
  • Fluspirilene
    Dopamine receptor antagonist; calcium channel blocker; antipsychotic.
    Katalog #CAS NummerSummenformelMenge
    sc-2528321841-19-6C29H31F2N3O10 mg
  • FSCPX
    Irreversible A1 adenosine receptor antagonist.
    Katalog #CAS NummerSummenformelMenge
    sc-252841156547-56-7C23H27FN4O6S25 mg
  • gamma-oryzanol
    Katalog #CAS NummerSummenformelMenge
    sc-29500611042-64-1C40H58O425 g/250 g
  • Gefitinib
    An epidermal growth factor receptor (EGFR)-tyrosine kinase inhibitor that has been shown to increase phosphorylation of c-Jun NH2 -terminal kinase (JNK) and p38 mitogen-activated protein kinase (MAPK) in HaCaT cells.
    Katalog #CAS NummerSummenformelMenge
    sc-202166184475-35-2C22H24ClFN4O3100 mg/250 mg
  • Glycine hydrochloride
    Spinal cord inhibitory neurotransmitter. Also allosterically regulates NMDA receptors.
    Katalog #CAS NummerSummenformelMenge
    sc-2633466000-43-7C2H5NO2 ·HCl100 g/500 g
  • Guaifenesin
    An expectorant reported to have muscle relaxant and sedative activity, where it is often used as anesthetic during animal surgery.
    Katalog #CAS NummerSummenformelMenge
    sc-20571093-14-1C10H14O425 g/100 g
  • Guvacine hydrochloride
    Inhibits GABA uptake.
    Katalog #CAS NummerSummenformelMenge
    sc-2633476027-91-4C6H9NO2•HCl25 mg
  • Hemicholinium-3
    A potent and selective choline uptake blocker.
    Katalog #CAS NummerSummenformelMenge
    sc-252873312-45-8C24H34Br2N2O4100 mg
  • Hesperetin
    A dietary flavanone with a chemopreventive effect.
    Katalog #CAS NummerSummenformelMenge
    sc-25287869097-99-0C16H14O61 g
  • Hexamethonium chloride
    A preferential nicotinic receptor blocker at the level of autonomic ganglia. Has been shown to cross the blood-brain barrier only in high doses.
    Katalog #CAS NummerSummenformelMenge
    sc-26338360-25-3(CH3)3N(Cl)(CH2)6N(Cl)(CH3)35 g
  • Hexestrol dipropionate
    Katalog #CAS NummerSummenformelMenge
    sc-2501114825-53-0C24H30O45 g
  • Hydrastinine hydrochloride
    Katalog #CAS NummerSummenformelMenge
    sc-2501244884-68-8C11H13NO3•HCl100 mg
  • Hydrocortisone 17-valerate
    Katalog #CAS NummerSummenformelMenge
    sc-23533257524-89-7C26H38O6500 mg
  • Hydrocortisone 21-hemisuccinate
    Katalog #CAS NummerSummenformelMenge
    sc-2283192203-97-6C25H34O81 g
  • Hydroxocobalamin hydrochloride
    Katalog #CAS NummerSummenformelMenge
    sc-23533658288-50-9C62H89CoN13O15P•HCl100 mg
  • Hydroxyzine pamoate salt
    Katalog #CAS NummerSummenformelMenge
    sc-22832710246-75-0C44H43ClN2O810 g
  • I-AB-MECA
    A reference standard used for radioiodinated I-AB-MECA. This is a widely used, high affinity radioligand for the A3 adenosine receptor.
    Katalog #CAS NummerSummenformelMenge
    sc-250141152918-27-9C18H20IN7O41 mg
  • Imidazole-4-acetic acid sodium salt
    Competitive antagonist at GABAC receptors.
    Katalog #CAS NummerSummenformelMenge
    sc-25290056368-58-2C5H5N2NaO2500 mg/1 g
  • Imipramine N-oxide
    The tertiary amine-oxidized metabolite of Imipramine. A useful standard for investigating FMO-mediated oxidation activity with Imipramine as a substrate.
    Katalog #CAS NummerSummenformelMenge
    sc-2009736829-98-7C19H24N2O5 mg/25 mg
  • Indapamide
    An antihypertensive agent that reduces intracellular calcium levels. Maintains magnesium ion but reduces phosphate ions involved in arterial rigidity and many other functions.
    Katalog #CAS NummerSummenformelMenge
    sc-20477726807-65-8C6H16ClN3O3S250 mg/1 g
  • Indoramin hydrochloride
    α1-adrenoceptor antagonist.
    Katalog #CAS NummerSummenformelMenge
    sc-25290638821-52-2C22H26ClN3O10 mg
  • Ipratropium bromide monohydrate
    N-isopropyl quaternary salt of atropine. A nonselective muscarinic acetylcholine receptor antagonist; bronchodilator.
    Katalog #CAS NummerSummenformelMenge
    sc-25291166985-17-9C20H31BrNO3250 mg
  • Isoetharine mesylate salt
    β-Adrenergic receptor agonist, bronchodilator.
    Katalog #CAS NummerSummenformelMenge
    sc-2529187279-75-6C13H21NO3 ·CH4O3S1 g
  • (-)-Isoproterenol (+)-bitartrate salt
    β-Adrenoceptor agonist. increases cytosolic cAMP.
    Katalog #CAS NummerSummenformelMenge
    sc-25292654750-10-6C11H17NO3 ·C4H6O6100 mg/500 mg
  • Isosilybin
    Useful in the treatment of liver disease.
    Katalog #CAS NummerSummenformelMenge
    sc-21519972581-71-6C25H22O101 mg
  • JNJ7777120
    A potent, selective non-imidazole H4 histamine receptor antagonist.
    Katalog #CAS NummerSummenformelMenge
    sc-252930459168-41-3C14H16N3OCl5 mg
  • Kisspeptin-234 trifluoroacetate salt
    Katalog #CAS NummerSummenformelMenge
    sc-300857n.n.C63H76N17O14•xC2HF3O21 mg
  • L-741,626
    A selective antagonist of the dopamine D2 receptor.
    Katalog #CAS NummerSummenformelMenge
    sc-25293681226-60-0C20H21ClN2O10 mg
  • L-Allylglycine
    A Glutamic acid decarboxylase inhibitor.
    Katalog #CAS NummerSummenformelMenge
    sc-25523616338-48-0C5H9NO2500 mg
  • L-Cysteinesulfinic acid monohydrate
    A putative excitatory amino acid neurotransmitter.
    Katalog #CAS NummerSummenformelMenge
    sc-215212207121-48-0C3H7NO4S•H2O100 mg/250 mg
  • L-Glutamic acid monosodium salt hydrate
    An excitatory amino acid neurotransmitter which is an agonist at kainate, quisqualate and NMDA receptors.
    Katalog #CAS NummerSummenformelMenge
    sc-215218142-47-2 (anhydrous)C5H8NNaO4•xH2O100 g/500 g
  • L-Histidine monohydrochloride monohydrate
    Histamine precursor via histidine decarboxylase.
    Katalog #CAS NummerSummenformelMenge
    sc-2634425934-29-2C6H9N3O2•HCl•H2O5 g/25 g
  • L-Tyrosine disodium salt hydrate
    This is an amino acid precursor of dopamine and other catecholamines.
    Katalog #CAS NummerSummenformelMenge
    sc-25294069847-45-6C9H9NNa2O3•xH2O25 g/100 g
  • Labetalol hydrochloride
    Competitive β-adrenoceptor antagonist.
    Katalog #CAS NummerSummenformelMenge
    sc-25294232780-64-6C19H24N2O3 ·HCl5 g
  • Lapatinib Ditosylate
    A selective and effective inhibitor of ErbB-2 and EGFR dual tyrosine kinases. Research studies have reported that the compound can inhibit breast cancer cell proliferation.
    Katalog #CAS NummerSummenformelMenge
    sc-202205388082-78-8C29H26ClFN4O4S ·2C7H8O3S10 mg/25 mg
  • Lofepramine hydrochloride
    An antidepressant and a serotonin and norepinephrine re-uptake inhibitor (SNRI).
    Katalog #CAS NummerSummenformelMenge
    sc-25525626786-32-3C26H28Cl2N2O5 mg
  • Lupinine
    An alkaloid isolate from Anabisis aphylla. Able to reduce the effect of ethanol anesthesia.
    Katalog #CAS NummerSummenformelMenge
    sc-205737486-70-4C10H19NO25 mg/100 mg
  • LY-165,163
    Selective 5-HT1A and 5-HT1D serotonin receptor antagonists.
    Katalog #CAS NummerSummenformelMenge
    sc-2529771814-64-8C19H22F3N325 mg
  • m-Tyramine hydrochloride
    Katalog #CAS NummerSummenformelMenge
    sc-2552573458-98-8C8H11NO··HCl100 mg
  • MADAM dihydrochloride
    High affinity ligand for the serotonin transporter SERT
    Katalog #CAS NummerSummenformelMenge
    sc-252980411208-45-2C16H22Cl2N2S5 mg
  • Magnesium L-aspartate salt
    Katalog #CAS NummerSummenformelMenge
    sc-29526318962-61-3n.n.25 g
  • Mebeverine hydrochloride
    Katalog #CAS NummerSummenformelMenge
    sc-2355792753-45-9C25H35NO5•HCl10 g
  • Mebhydroline 1,5-naphthalenedisulfonate salt
    Antagonist to H1 Histamine receptors.
    Katalog #CAS NummerSummenformelMenge
    sc-2634596153-33-9C19H20N2 ·1/2C10H8O6S21 g
  • Melphalan
    Cytotoxic drug used to treat multiple myeloma. Phenylamine derivative of mechorethamine.
    Katalog #CAS NummerSummenformelMenge
    sc-204799148-82-3C13H18Cl2N2O2100 mg/250 mg
  • Mepirizole
    Katalog #CAS NummerSummenformelMenge
    sc-23558918694-40-1C11H14N4O210 g
  • Metaproterenol hemisulfate salt
    This compound is a β2-adrenoceptor agonist.
    Katalog #CAS NummerSummenformelMenge
    sc-2577015874-97-5C22H36N2O10S1 g
  • Metaraminol (+)-bitartrate salt
    An α-adrenoceptor agonist.
    Katalog #CAS NummerSummenformelMenge
    sc-25300433402-03-8C9H13NO2•C4H6O61 g
  • Methazolamide
    Katalog #CAS NummerSummenformelMenge
    sc-235615554-57-4C5H8N4O3S21 g
  • Methiothepin mesylate salt
    Methiothepin mesylate salt is a 5-HT1, 5-HT6, 5-HT7 serotonin receptor antagonist that blocks serotonin auto receptors.
    Katalog #CAS NummerSummenformelMenge
    sc-25300574611-28-2C20H24N2S2•CH3SO3H100 mg
  • Methoctramine hydrate
    This is a selective M2 muscarinic receptor antagonist at nM concentrations. At mM concentrations, methoctramine directly inhibits the high affinity GTPase activity of G proteins. The increase in calcium and arachidonic acid release were attenuated by the M2 receptor antagonist methoctramine, this is not only by the M3 receptor antagonist p-fluoro-hexahydro siladifenidol.
    Katalog #CAS NummerSummenformelMenge
    sc-257709104807-46-7 (anhydrous)C36H62N4O2•4HCl•xH2O10 mg/25 mg
  • Methoxamine hydrochloride
    Agonist to alpha-1-adrenoceptors.
    Katalog #CAS NummerSummenformelMenge
    sc-26346861-16-5C11H17NO3•HCl500 mg
  • Methyl 6-Methoxy-2-naphthylacetate
    A potential prodrug.
    Katalog #CAS NummerSummenformelMenge
    sc-21187123981-48-8C14H14O325 mg
  • Methyllycaconitine citrate hydrate
    A potent and specific nicotinic receptor antagonist that binds to neuronal α-bungarotoxin sites.
    Katalog #CAS NummerSummenformelMenge
    sc-25304321019-30-7 (non-salt)C43H58N2O175 mg
  • Metoclopramide hydrochloride
    This is a D2 antagonist and a 5-HT3 antagonist. Antipsychotic. Anti-emetic.
    Katalog #CAS NummerSummenformelMenge
    sc-2530467232-21-5C14H22ClN3O2•HCl10 g/25 g
  • Metrazoline
    A potent and selective imidazoline binding site ligand.
    Katalog #CAS NummerSummenformelMenge
    sc-253047221225-04-3C14H16N2O45 mg
  • Minaprine dihydrochloride
    Antidepressant
    Katalog #CAS NummerSummenformelMenge
    sc-25304925905-77-5C17H22N4O•2HCl1 g
  • MK-912 hydrate
    A selective α2-adrenoceptor antagonist.
    Katalog #CAS NummerSummenformelMenge
    sc-253050119942-70-0 (anhydrous)C20H25N3O2•HCl•xH2O5 mg
  • Moguisteine
    An anti-tussive with similar properties to codeine.
    Katalog #CAS NummerSummenformelMenge
    sc-204810119637-67-1C16H21NO5S100 mg/250 mg
  • Montelukast Sodium
    A potent, selective CysLT1 receptor antagonist (IC50 < 5nM), competitive with respect to LTD4, with no appreciable affect on the CysLT2 receptor.
    Katalog #CAS NummerSummenformelMenge
    sc-202231151767-02-1C35H35ClNO3S•Na10 mg/25 mg
  • Mosapride citrate dihydrate
    Antagonist to both 5-HT4 and 5-HT3 receptors.
    Katalog #CAS NummerSummenformelMenge
    sc-263722636582-62-2C21H25ClFN3O3 ·C6H8O7 ·2H2O10 mg
  • Moxisylyte hydrochloride
    α1-adrenoceptor antagonist; peripheral vasodilator.
    Katalog #CAS NummerSummenformelMenge
    sc-255308964-52-3C16H25NO3•HCl1 g/5 g
  • MPP+ iodide
    MPP+ iodide is an active metabolite of dopaminergic neurotoxin MPTP.
    Katalog #CAS NummerSummenformelMenge
    sc-25530936913-39-0C12H12IN100 mg
  • MRS 1191
    A selective A3 adenosine receptor antagonist. Selective for both human and rat.
    Katalog #CAS NummerSummenformelMenge
    sc-253056185222-90-6C31H27NO42 mg
  • MRS 1523
    A selective A3 adenosine receptor antagonist in the rat.
    Katalog #CAS NummerSummenformelMenge
    sc-253057212329-37-8C23H29NO3S5 mg
  • MRS 2179 ammonium salt hydrate
    Competitive to P2Y1 puinoreceptor antagonist.
    Katalog #CAS NummerSummenformelMenge
    sc-253058101204-49-3 (non-salt)C11H17N5O9P2•xNH3•yH2O5 mg
  • MRS 2395
    An antagonist for the P2Y12 purinoceptor, which causes platelet aggregation in rats via ADP induction.
    Katalog #CAS NummerSummenformelMenge
    sc-253059491611-55-3C20H30ClN5O45 mg
  • MSX-3 hydrate
    A selective A2A adenosine receptor antagonist prodrug.
    Katalog #CAS NummerSummenformelMenge
    sc-255310261717-23-1 (anhydrous)C21H21N4O7PNa2•xH2O5 mg
  • (+)-Muscarine chloride
    Active enantiomer; prototype muscarinic acetylcholine receptor agonist.
    Katalog #CAS NummerSummenformelMenge
    sc-2530602303-35-7C9H20ClNO25 mg
  • (±)-Muscarine chloride hydrate
    A muscarinic acetylcholine receptor agonist which was originally isolated from Amanita muscaria.
    Katalog #CAS NummerSummenformelMenge
    sc-2553112936-25-6 (anhydrous)C9H20ClNO2•xH2O5 mg
  • (+)-Muscarine iodide
    Katalog #CAS NummerSummenformelMenge
    sc-36276924570-49-8C9H20INO210 mg
  • N -Methyl-5-hydroxy trypt amine oxalate salt
    A serotonin receptor ligand.
    Katalog #CAS NummerSummenformelMenge
    sc-2530611975-81-1C13H16N2O5500 mg
  • N-Acetyl-N-acetoxy-4-chlorobenzenesulfonamide
    A pro-drug of the potent vasorelaxant nitroxyl, H-N=O, which it slowly releases in neutral solution. HNO eventually dimerizes and dehydrates to N2O, without producing NO.
    Katalog #CAS NummerSummenformelMenge
    sc-203441142867-52-5C10H10CINO5S10 mg/50 mg
  • N-Desmethylclozapine
    A major metabolite of clozapine (sc-200402), found to act as a potent antagonist of the 5-HT1C serotonin receptor, and a moderate agonist of M(1) mAChR.
    Katalog #CAS NummerSummenformelMenge
    sc-2011136104-71-8C17H17ClN45 mg/25 mg
  • N-Methyl dopamine hydrochloride
    Used as an internal standard for catecholamine analyses. Dopamine receptor agonist, α-adrenoceptor agonist.
    Katalog #CAS NummerSummenformelMenge
    sc-35843062-32-8C9H13NO2•HCl25 mg/50 mg
  • N-Methylhistaprodifen dioxalate salt
    More potent than a histamine by a factor of 3.5 on guinea pig ileum and more potent than histamine by a factor of 4.3 on guinea pig arterial H1-receptor-mediated vasoconstriction. The most potent H1-receptor agonist on the guinea pig ileum out of 17 agonists tested. Does not stimulate H2 and H3 histamine receptors and has potential use in the study of H1-receptor-mediated physiological and pathophysiological functions.
    Katalog #CAS NummerSummenformelMenge
    sc-255360270079-48-6C21H25N3•2 ·C2H2O45 mg
  • (-)-N-Methylphysostigmine
    Katalog #CAS NummerSummenformelMenge
    sc-236078103877-07-2C16H23N3O25 mg
  • N-Methylspiperone hydrochloride
    A D2 dopamine receptor antagonist.
    Katalog #CAS NummerSummenformelMenge
    sc-25312187539-19-3C24H28FN3O2•HCl5 mg
  • N,N-Dipropyl-5-carboxamidotryptamine maleate salt
    A selective and potent 5-HT1A serotonin receptor agonist.
    Katalog #CAS NummerSummenformelMenge
    sc-25315174885-25-9C17H25N3O ·C4H4O45 mg
  • Nα-Methylhistamine dihydrochloride
    Production of N-alpha-methyl-histamine, which is a histamine 3 receptor (H3R) agonist, is promoted in Helicobacter pylori infected human gastric mucosa. NAMH acts directly on H2Rs in animals to stimulate acid secretion and to be a H2R agonist. NAMH dose dependently stimulated cAMP productions in CHO-H2R cells. This production was inhibited by famotidine but not by thioperamide. Control CHO cells were unresponsive to either histamine or NAMH. In addition, the effect of NAMH, in terms of cAMP production in CHO-H2R cells, was more potent than that of histamine-that is, with a lower EC50 concentration and higher maximal cAMP production. Both NAMH and histamine, but not R-alpha-methyl-histamine, effectively inhibited [(3)H] tiotidine binding to CHO-H2R cells. These results confirm that NAMH, which is produced in the gastric mucosa by H pylori, is a potent H2R agonist as well as a H3R agonist.
    Katalog #CAS NummerSummenformelMenge
    sc-25317416503-22-3C6H11N3•2HCl10 mg
  • N6-(2-Phenylethyl)adenosine
    Selective A1 adenosine receptor agonist.
    Katalog #CAS NummerSummenformelMenge
    sc-25316820125-39-7C18H21N5O410 mg
  • (-)-N6-(2-Phenylisopropyl)adenosine
    A1 adenosine receptor agonist. Its affinity for adenosine receptor is approximately 100x that of the (+)-isomer.
    Katalog #CAS NummerSummenformelMenge
    sc-25316938594-96-6C19H23N5O425 mg
  • N6-2-(4-Aminophenyl)ethyladenosine
    A potent, non-selective A3 adenosine receptor agonist.
    Katalog #CAS NummerSummenformelMenge
    sc-25317089705-21-5C18H22N6O425 mg
  • N6-Cyclohexyladenosine
    Selective A1 adenosine receptor agonist.
    Katalog #CAS NummerSummenformelMenge
    sc-25538536396-99-3C16H23N5O450 mg
  • N8-Acetylspermidine dihydrochloride
    Katalog #CAS NummerSummenformelMenge
    sc-23615134450-15-2C9H21N3O•2HCl100 mg
  • Nadolol
    A polar and hydrophilic, non-selective β blocker, which displays activity against β-1 and β-2 receptors. It is known that Nadolol inhibits the release of catecholamines from the adrenal glands.
    Katalog #CAS NummerSummenformelMenge
    sc-25317542200-33-9C17H27NO41 g
  • Nafronyl oxalate salt
    Exhibits properties of a vasodilator.
    Katalog #CAS NummerSummenformelMenge
    sc-2531763200-06-4C24H33NO3•C2H2O45 g
  • Naftopidil hydrochloride hydrate
    Antihypertensive and antagonist to α1-adrenoceptor.
    Katalog #CAS NummerSummenformelMenge
    sc-26394157149-07-2 (non-salt)C24H28N2O3•xHCl•yH2O25 mg
  • NCS-356 sodium salt hydrate
    γ-Hydroxybutyrate (GHB) receptor agonist.
    Katalog #CAS NummerSummenformelMenge
    sc-253182430440-66-7C10H8ClO3Na•xH2O50 mg
  • Nefiracetam
    A nootropic drug of the racetam family. Used to treat Alzheimer’s disease and other diseases related to learning and memory deficits.
    Katalog #CAS NummerSummenformelMenge
    sc-20576677191-36-7C14H18N2O2100 mg/250 mg
  • Nifekalant Hydrochloride
    A class III antiarrhythmic drug that has shown to be effective against ventricular tachyarrhythmias by inhibiting HERG channels in a voltage-dependent and frequency-dependent manner.
    Katalog #CAS NummerSummenformelMenge
    sc-204819130656-51-8C19H27N5O5 ·HCl10 mg/25 mg
  • Nifenazone
    Katalog #CAS NummerSummenformelMenge
    sc-2361752139-47-1C17H16N4O25 g
  • (±)-Norepinephrine (+)-bitartrate salt
    An adrenergic neurotransmitter.
    Katalog #CAS NummerSummenformelMenge
    sc-2553963414-63-9C8H11NO3•C4H6O61 g
  • (+)-Norfenfluramine hydrochloride
    (+)-Norfenfluramine is the major hepatic metabolite of (+)-fenfluramine and is primarily responsible for the anorexic effect, as well as side effects; (+)-norfenfluramine causes vasoconstriction and a blood pressure increase in rats with normal blood; more potent than fenfluramine at inducing dopamine release; acts primarily on the cytoplasmic pool of serotonin.
    Katalog #CAS NummerSummenformelMenge
    sc-25320037936-89-3C10H12F3N ·HCl10 mg
  • Norfentanyl
    Major urinary metabolite of a narcotic analgesic fentanyl.
    Katalog #CAS NummerSummenformelMenge
    sc-2220771609-66-1C14H20N2O1 mg/10 mg
  • Nylidrin hydrochloride
    Katalog #CAS NummerSummenformelMenge
    sc-358467849-55-8C19H25NO2•HCl200 mg/5 g
  • Octoclothepin maleate salt
    5-HT2 serotonin receptor antagonist; D2 dopamine receptor antagonist.
    Katalog #CAS NummerSummenformelMenge
    sc-2532154789-68-8C23H25ClN2O4S25 mg
  • Opiorphin
    A natural analgesic that is secreted into human saliva. Opiorphin demonstrates dual-inhibitory potency on the enkephalin-inactivating ectopeptidases human NEP (hNEP) and human AP-N (hAP-N). As an analgesic, Opiorphin is 6 times stronger than the opiate morphine. Opiorphin is closely related to the rat sialorphin peptide, which is an inhibitor of pain perception and acts by potentiating endogenous micro- and ∂-opioid receptor-dependent enkephalinergic pathways. In rat studies, Opiorphin suppressed pain sensation for both chemical-induced inflammation and acute physical pain. In both cases, the administered dose of 1 mg/kg provided the same painkilling power as 3-6 mg/kg of morphine.
    Katalog #CAS NummerSummenformelMenge
    sc-253217864084-88-8C29H48N12O81 mg
  • Org 24598 lithium salt
    This is a selective, potent inhibitor of glial GlyT (GlyT1, glycine transporter type 1). In rats (P12-P16) and kynurenic acid, 6-cyano-7-nitroquinoxaline-2,3-dione (CNQX) and bicuculline, ORG 24598 at a concentration of 10 µM induced a mean inward current of -10/-50 pA at -60 mV and increased significantly the decay time constants of miniature (mIPSCs), spontaneous (sIPSCs) and electrically evoked glycinergic (eIPSCs) inhibitory postsynaptic currents. Replacing extracellular sodium with N-methyl-d-glucamine or superfusing the slice with micromolar concentrations of glycine also increased the decay time constant of glycinergic IPSCs. Glycine (1-5 µM and d-serine (10 µM) increased the amplitude of eEPSCs whereas l-serine had no effect. Org 24598 increased significantly the amplitude of NMDA receptor-mediated eEPSCs without affecting the amplitude of non-NMDA receptor-mediated eEPSCs. This brings conclusion that blocking glial glycine transporter by Org 24598 increased the level of glycine in spinal cord slices, which in turn prolonged the duration of glycinergic synaptic current and potentiated the NMDA-mediated synaptic response.
    Katalog #CAS NummerSummenformelMenge
    sc-253218722456-08-8C19H19F3LiNO35 mg
  • p-Aminoclonidine hydrochloride
    This product is an α2-adrenoceptor agonist.
    Katalog #CAS NummerSummenformelMenge
    sc-30150873218-79-8C9H10Cl2N4•xHCl1 mg
  • p-Fluorohexahydro-sila-difenidol hydrochloride
    High affinity M3 muscarinic acetylcholine receptor antagonist.
    Katalog #CAS NummerSummenformelMenge
    sc-257953116679-83-5C20H32FNOSi ·HCl10 mg
  • p-MPPI monohydrochloride
    A selective 5-HT1A serotonin receptor antagonist that crosses the blood-brain barrier.
    Katalog #CAS NummerSummenformelMenge
    sc-253226220643-77-6C25H27IN4O2 ·HCl250 mg
  • p-MPPI trihydrochloride
    Katalog #CAS NummerSummenformelMenge
    sc-358823155204-23-2 (free base)C25H27IN4O210 mg
  • P1,P4-Di(adenosine-5') tetraphosphate ammonium salt
    A derivative of Diadenosine polyphosphate, which is stored in secretory granules of thrombocytes, chromaffin, and neuronal cells. Has been shown to function as a pancreatic cell secondary messenger, phospholipase D stimulator, change intracellular calcium levels, nitric oxide release inductor, 5’-nucleotidase activator and adenosine kinase activity inhibitor in vitro.
    Katalog #CAS NummerSummenformelMenge
    sc-253229102783-36-8C20H31N11O19P410 mg
  • P7C3
    Katalog #CAS NummerSummenformelMenge
    sc-362776301353-96-8C21H18Br2N2O10 mg/50 mg
  • Pasiniazid
    Katalog #CAS NummerSummenformelMenge
    sc-2506522066-89-9C13H14N4O410 g
  • PD 116,948
    PD 116,948, a xanthine derivative, is a very potent and selective adenosine A1 receptor antagonist.
    Katalog #CAS NummerSummenformelMenge
    sc-200115102146-07-6C16H24N4O220 mg/100 mg
  • (+/-)-PD 128,907 hydrochloride
    Selective D3 dopamine receptor agonist.
    Katalog #CAS NummerSummenformelMenge
    sc-257969112960-16-4C14H19NO3•HCl5 mg
  • Pheniramine maleate salt
    A H1 histamine receptor antagonist.
    Katalog #CAS NummerSummenformelMenge
    sc-253258132-20-7C16H20N2•C4H4O45 g
  • Phenyltoloxamine citrate salt
    Katalog #CAS NummerSummenformelMenge
    sc-2289401176-08-5C17H21NO•C6H8O750 g
  • Picrotoxinin
    GABAA receptor antagonist that binds to the GABA receptor-linked Cl- channel. Active component of picrotoxin
    Katalog #CAS NummerSummenformelMenge
    sc-25327717617-45-7C15H16O6250 mg
  • Pimethixene maleate salt
    Katalog #CAS NummerSummenformelMenge
    sc-22894913187-06-9C19H19NS•C4H4O4250 mg
  • Pipamperone dihydrochloride
    Antipsychotic; D2 dopamine receptor antagonist; 5-HT2 serotonin receptor antagonist.
    Katalog #CAS NummerSummenformelMenge
    sc-2532782448-68-2C21H30N3O2F•2HCl100 mg
  • Piperidine-4-sulfonic acid
    GABAAreceptor agonist.
    Katalog #CAS NummerSummenformelMenge
    sc-25327972450-62-5C5H11NO3S25 mg
  • Pirenperone
    5-HT2 serotonin receptor antagonist.
    Katalog #CAS NummerSummenformelMenge
    sc-25328075444-65-4C23H24FN3O225 mg
  • (±)-PPHT hydrochloride
    Potent D2 dopamine receptor agonist. A series of new dopamine (DA) receptor agonists, of the 2-aminotetralin group, i.e. N-0434, N-0437 and N-0734 were investigated both in vivo and in vitro pharmacological test systems. In vivo, the reversal of the gamma-butyrolactone-induced an increase in rat central DOPA biosynthesis, the rate was taken as a measure of presynaptic activity. The homovanillic acid (HVA) decrease, after intraperitoneal and after oral administration of the drugs was also taken as a measure of presynaptic activity. Postsynaptic activity was measured in two behavioural models, i.e. stereotypy induction and reserpine reversal. The effects of (±)-PPHT (N-0434) these drugs on noradrenaline and dopamine turnover (alpha-MpT method) were studied in addition. The results indicate that all three compounds N-0434 ((±)-PPHT), N-0437 and N-0734 are potent and selective DA agonists that lack significant alpha 2 activity.
    Katalog #CAS NummerSummenformelMenge
    sc-25331371787-90-1C21H28ClNO10 mg
  • Pramoxine hydrochloride
    Skin or mucous membrane topical anesthetic.
    Katalog #CAS NummerSummenformelMenge
    sc-264141637-58-1C17H28ClNO310 g
  • Pranoprofen
    A non-steroidal antiinflammatory drug. It inhibits platelet aggregation.
    Katalog #CAS NummerSummenformelMenge
    sc-20581452549-17-4C15H13NO3100 mg/250 mg
  • Primaquine phosphate
    Antimalarial drug with genotoxicity (Ames test) and cardiotoxicity (inhibitor of cardiac Na+ current).
    Katalog #CAS NummerSummenformelMenge
    sc-20581763-45-6C15H21N3O.2H3PO45 g/10 g
  • Propantheline bromide
    Inhibits action of acetylcholine at post-ganglionic synapses; muscarinic acetylcholine receptor antagonist; antispasmodic; reduces gastric acid secretion.
    Katalog #CAS NummerSummenformelMenge
    sc-25332050-34-0C23H30NO3Br5 g
  • Proparacaine hydrochloride
    Topical ophthalmic anesthetic
    Katalog #CAS NummerSummenformelMenge
    sc-2641465875-06-9C16H27ClN2O31 g
  • Protriptyline hydrochloride
    A norepinephrine uptake blocker.
    Katalog #CAS NummerSummenformelMenge
    sc-2507991225-55-4C19H21N•HCl100 mg
  • Proxymetacaine Hydrochloride
    A local anesthetic that is used to numb the surface of a body part.
    Katalog #CAS NummerSummenformelMenge
    sc-2058205875-06-9C16H27ClN2O3100 mg/250 mg
  • PSB 1115 potassium salt hydrate
    A highly selective, water-soluble, human A2B adenosine receptor antagonist.
    Katalog #CAS NummerSummenformelMenge
    sc-253323409344-71-4 (anhydrous)C14H13KN4O5S•xH2O10 mg
  • Pyridoxal phosphate-6-azo(benzene-2,4-disulfonic acid) tetrasodium salt hydrate
    A selective P2 purinoceptor antagonist which blocks responses at both pre- and post-junctional sites.
    Katalog #CAS NummerSummenformelMenge
    sc-253332192575-19-2 (anhydrous)C14H10N3Na4O12PS2•xH2O10 mg/50 mg
  • (±)-Quinpirole dihydrochloride
    D2-like dopamine receptor agonist which has some activity at D3 sites.
    Katalog #CAS NummerSummenformelMenge
    sc-25333873625-62-4C13H21N3•2HCl50 mg
  • (-)-Quinpirole hydrochloride
    The putative D2 dopamine receptor agonist quinpirole is the most widely used D2 agonist in in vivo and in vitro studies. Active enantiomer of (±)-quinpirole. Quinpirole is a dopamine agonist with high affinity for the D2 and D3 dopamine receptor subtypes. Specific [3H]quinpirole binding in rat brain was saturable, and dependent on temperature, membrane concentration, sodium concentration and guanine nucleotides. Saturation analysis revealed high affinity binding characteristics (Kd = 2.3 +/- 0.3 nM) which were confirmed by association-dissociation kinetics. The regional distribution of [3H]quinpirole binding sites roughly paralleled the distribution of [3H]spiperone binding sites, with greatest densities present in the striatum, nucleus accumbens and olfactory tubercles. A variety of drugs, most notably monoamine oxidase inhibitors (MAOls), inhibit the binding of [3H]quinpirole, but not [3H]spiperone or [3H](-)N-n-Propylnorapomorphine, in rat striatal membranes by a mechanism that does not appear to involve the enzymatic activity of MAO. Clinically antidepressant MAOIs exhibited selectivity between sites labeled by [3H]quinpirole and [3H]spiperone as did a number of structurally related propargylamines and N-acylethylenediamine derivatives and other drugs such as debrisoquin and phenylbiguanide. The MAOIs clorgyline and Ro 41-1049 were the most potent. MAOIs interact with a novel binding site,may be associated with D2-like dopamine receptors, that is labeled by [3H]quinpirole or that modulates [3H]quinpirole binding.
    Katalog #CAS NummerSummenformelMenge
    sc-25333985798-08-9C13H21N3•HCl10 mg/25 mg
  • (+/-)-Quinuclidinyl benzilate
    Nonselective antagonist to muscarinic ACh receptors.
    Katalog #CAS NummerSummenformelMenge
    sc-2641946581-06-2C21H23NO35 mg/10 mg
  • Quirestine
    Potent short-acting ganglioblocker. Nicotinic acetylcholine receptor antagonist.
    Katalog #CAS NummerSummenformelMenge
    sc-25334041663-80-3C12H24IN2 mg
  • R-(-)-Apomorphine hydrochloride hemihydrate
    A nonselective dopamine agonist that causes nausea and emesis.
    Katalog #CAS NummerSummenformelMenge
    sc-25334141372-20-7C17H17NO2 ·HCl ·1/2H2O100 mg/250 mg
  • R-(-)-Desmethyldeprenyl hydrochloride
    Neuroprotectant and an anti-apoptotic.
    Katalog #CAS NummerSummenformelMenge
    sc-258056115586-38-4C12H15N•HCl5 mg
  • R(-)-2,10,11-Trihydroxy-N-propyl-noraporphine hydrobromide hydrate
    A potent, selective D2 dopamine receptor agonist.
    Katalog #CAS NummerSummenformelMenge
    sc-25335079640-85-0 (anhydrous)C19H21NO3•HBr•xH2O10 mg/25 mg
  • R(-)-2,10,11-Trihydroxyaporphine hydrobromide
    Dopamine receptor agonist.
    Katalog #CAS NummerSummenformelMenge
    sc-25335177630-01-4C17H17NO3•HBr50 mg
  • R(-)-Denopamine
    Katalog #CAS NummerSummenformelMenge
    sc-36070371771-90-9C18H23NO45 mg
  • R(-)-Propylnorapomorphine hydrochloride
    Very potent and selective D2 dopamine receptor agonist.
    Katalog #CAS NummerSummenformelMenge
    sc-25335418426-20-5C19H21NO2•HCl10 mg/25 mg
  • R(+)-3-(3-Hydroxyphenyl)-N-propylpiperidine hydrochloride
    A D2 dopamine receptor agonist. Also functions as 1 receptor antagonist with essentially no affinity for the phencylidine site on the NMDA receptor.
    Katalog #CAS NummerSummenformelMenge
    sc-25335589874-80-6C14H21NO•HCl25 mg
  • R(+)-7-Hydroxy-DPAT hydrobromide
    Active enantiomer of (±)-7-hydroxy-DPAT; selective D3 dopamine receptor agonist.
    Katalog #CAS NummerSummenformelMenge
    sc-25335682730-72-1C16H26BrNO5 mg
  • R(+)-SKF-81297 hydrobromide
    A selective D1 dopamine receptor agonist.
    Katalog #CAS NummerSummenformelMenge
    sc-253357253446-15-0C16H16ClNO2•HBr5 mg
  • R(+)-UH-301 hydrochloride
    A potent and selective 5-HT1A serotonin receptor agonist.
    Katalog #CAS NummerSummenformelMenge
    sc-253358127126-18-5C16H25ClFNO1 mg
  • (R)-(+)-8-Hydroxy-DPAT hydrobromide
    (R)-(+)-8-Hydroxy-DPAT is a full 5-HT1A serotonin receptor agonist; active enantiomer of (±)-8-hydroxy-DPAT.
    Katalog #CAS NummerSummenformelMenge
    sc-25340478095-19-9C16H25NO•HBr5 mg/25 mg
  • (R)-(+)-SKF-38393 hydrochloride
    Active enantiomer of (±)-SKF-38393; D1 dopamine receptor agonist.
    Katalog #CAS NummerSummenformelMenge
    sc-25341281702-42-3C16H17NO2··HCl5 mg
  • (R)-SKF-82957 hydrobromide
    A selective D1 dopamine receptor agonist.
    Katalog #CAS NummerSummenformelMenge
    sc-255520288262-87-3C17H18ClNO2•HBr5 mg
  • Reboxetine mesylate hydrate
    A selective noradrenaline uptake inhibitor.
    Katalog #CAS NummerSummenformelMenge
    sc-25342698769-84-7 (anhydrous)C20H29NO7S5 mg
  • RF9 trifluoroacetate salt
    A neuropeptide FF receptor antagonist.
    Katalog #CAS NummerSummenformelMenge
    sc-253428876310-60-0 (non-salt)C26H38N6O3•xC2HF3O21 mg
  • Ro 27-3225 trifluoroacetate salt
    This is a selective melanocortin MC4 receptor agonist. EC50 = 1 nM.
    Katalog #CAS NummerSummenformelMenge
    sc-311523n.n.C39H52N12O6•xC2HF3O21 mg
  • Ro 4-1284
    A reversible VMAT2 inhibitor.
    Katalog #CAS NummerSummenformelMenge
    sc-255523303-75-3C21H33NO35 mg
  • Ro4368554
    A 5-HT6 receptor antagonist. Acts selectively at 5-HT6 receptors where it binds with a greater than 100-fold selectivity over other monoamine receptor subtypes.
    Katalog #CAS NummerSummenformelMenge
    sc-253435478082-99-4C19H21N3O2S5 mg
  • S-(-)-SKF-38393 hydrochloride
    Less active enantiomer of (±)-SKF-38393; D1 dopamine receptor agonist.
    Katalog #CAS NummerSummenformelMenge
    sc-25344081702-43-4C16H17NO2•HCl100 mg
  • S-(+)-Chlorpheniramine maleate salt
    Active isomer; H1 histamine receptor antagonist.
    Katalog #CAS NummerSummenformelMenge
    sc-2534412438-32-6C20H23ClN2O41 g
  • S-(+)-O-Desmethylraclopride hydrobromide
    Precursor to radiolabeled S-(+)-raclopride.
    Katalog #CAS NummerSummenformelMenge
    sc-258091113310-88-6C14H18Cl2N2O3•HBr5 mg
  • S-(4-Nitrobenzyl)-6-thioinosine (NBTI, NBMPR)
    An inhibitor of equilibrative nucleoside trasport proteins. Blocks the uptake and transport of adenosine.
    Katalog #CAS NummerSummenformelMenge
    sc-20011738048-32-7C17H17N5O6S50 mg
  • S(-)-Baclofen hydrochloride
    The less active enantiomer of baclofen, which happens to be the same enantiomer as S(+)-baclofen free base.
    Katalog #CAS NummerSummenformelMenge
    sc-26424663701-56-4C10H12ClNO2•HCl25 mg/100 mg
  • S(-)-Cyanopindolol hemifumarate salt
    A 5-HT1A/1B serotonin receptor antagonist; β3-adrenoceptor antagonist.
    Katalog #CAS NummerSummenformelMenge
    sc-253460874882-72-1C32H42N6O4··C4H4O41 mg
  • S(-)-Raclopride (+)-tartrate salt
    A selective D2 dopamine receptor antagonist.
    Katalog #CAS NummerSummenformelMenge
    sc-25346198185-20-7C15H20Cl2N2O3··C4H6O625 mg
  • S(-)-UH-301 hydrochloride
    A potent, selective 5-HT1A serotonin receptor antagonist and D2/D3 dopamine receptor agonist.
    Katalog #CAS NummerSummenformelMenge
    sc-253462127126-22-1C16H24FNO•HCl1 mg/5 mg
  • S(+)-Propylnorapomorphine hydrochloride
    Limbic-selective dopamine antagonist.
    Katalog #CAS NummerSummenformelMenge
    sc-25346379703-31-4C19H21NO2•HCl5 mg
  • (S)-(-)-3-(3-Hydroxyphenyl)-N-propylpiperidine hydrochloride
    A dopamine autoreceptor agonist and a postsynaptic dopamine receptor antagonist.
    Katalog #CAS NummerSummenformelMenge
    sc-25347788768-67-6C14H22ClNO25 mg/100 mg
  • (S)-(+)-Apomorphine hydrochloride hydrate
    Dopamine receptor antagonist. Is inactive as an agonist.
    Katalog #CAS NummerSummenformelMenge
    sc-25350541035-30-7 (anhydrous)C17H17NO2•HCl•xH2O5 mg
  • (S)-Mephenytoin
    A hydantoin used in the (S)-Mephenytoin 4’-hydroxylation assay for studying CYP2C19 polymorphism.
    Katalog #CAS NummerSummenformelMenge
    sc-20097570989-04-7C12H14N2O25 mg/25 mg
  • (S)-Nafadotride tartrate
    D3 Dopamine receptor antagonist.
    Katalog #CAS NummerSummenformelMenge
    sc-253523173429-65-7C26H33O8N31 mg
  • SB 242084 hydrochloride
    An antagonist of the 5-HT2C receptor (pKi= 9.0), with at least 100-fold more selectivity over other 5-HT, dopamine or adrenergic receptors; used extensively in animal research to evaluate, for example, 5-HT2C receptor agonists and neurotransmitter receptor interactions in mice.
    Katalog #CAS NummerSummenformelMenge
    sc-3518481049747-87-6C21H19ClN4O2•2HCl1 mg/5 mg
  • SB 242084 dihydrochloride hydrate
    Crosses the blood-brain barrier; selective 5-HT2c serotonin receptor antagonist.
    Katalog #CAS NummerSummenformelMenge
    sc-253538181632-25-7 (non-salt)C21H19ClN4O2•2HCl•xH2O5 mg
  • SB-215505
    Selective 5-HT2B serotonin receptor antagonist; 100-fold higher affinity at 2B compared to 2C.
    Katalog #CAS NummerSummenformelMenge
    sc-253540162100-15-4C19H16N3OCl5 mg
  • SB-224289 hydrochloride
    Selective 5-HT1B serotonin receptor antagonist
    Katalog #CAS NummerSummenformelMenge
    sc-253541180084-26-8C32H32N4O3•HCl5 mg
  • SB-269970 hydrochloride
    A selective 5-HT7 serotonin receptor antagonist.
    Katalog #CAS NummerSummenformelMenge
    sc-255605261901-57-9C18H28N2O3S•HCl5 mg
  • (-)-Scopolamine hydrochloride
    Competitive nonselective muscarinic acetylcholine antagonist. Scopolamine-induced amnesia in laboratory animals is a commonly-used model of memory deficit.
    Katalog #CAS NummerSummenformelMenge
    sc-25354455-16-3C17H21NO4•HCl1 g
  • (-)-Scopolamine methyl bromide
    A competitive muscarinic acetylcholine receptor antagonist.
    Katalog #CAS NummerSummenformelMenge
    sc-253545155-41-9C18H24NO4•Br1 g
  • (-)Scopolamine methyl nitrate
    Competitive antagonist to muscarinic receptors for use in the treatment of motion sickness.
    Katalog #CAS NummerSummenformelMenge
    sc-2643016106-46-3C17H21NO4•CH3NO31 g
  • Serotonin creatinine sulfate complex
    A neurotransmitter.
    Katalog #CAS NummerSummenformelMenge
    sc-215845971-74-4C14H19N5O2•H2O4S•H2O250 mg/500 mg
  • SKF 86002
    A bicyclic imidazole that specifically inhibits p38 MAP kinase, and is also described as a cytokine-suppressant and an anti-inflammatory compound.
    Katalog #CAS NummerSummenformelMenge
    sc-20326572873-74-6C16H12FN3S5 mg
  • (+/-)-SKF-38393 hydrochloride
    Agonist to D1 Dopamine receptors.
    Katalog #CAS NummerSummenformelMenge
    sc-26430662717-42-4C16H17NO2•HCl100 mg/500 mg
  • SKF-86466 hydrochloride
    Selective and potent α2 adrenoceptor antagonist.
    Katalog #CAS NummerSummenformelMenge
    sc-25356686129-54-6C11H15Cl2N10 mg
  • SKF-89976A
    GABA transporter type 1 inhibitor that crosses the blood brain barrier.
    Katalog #CAS NummerSummenformelMenge
    sc-25356785375-15-1C22H25NO2•HCl10 mg
  • SKF-95282 dimaleate salt
    Antagonist to H2 His receptor
    Katalog #CAS NummerSummenformelMenge
    sc-255616104076-39-3C22H27N3OS•2C4H4O410 mg
  • Sulfadimethoxine sodium salt
    Katalog #CAS NummerSummenformelMenge
    sc-2293441037-50-9C12H13N4O4SNa10 g
  • Suloctidil
    Katalog #CAS NummerSummenformelMenge
    sc-23695754767-75-8C20H35NOS5 g
  • T62
    Allosteric enhancer of A1 adenosine receptor.
    Katalog #CAS NummerSummenformelMenge
    sc-25361840312-34-3C15H14ClNOS5 mg
  • Temechine hydrobromide
    A neuronal nicotinic acetylcholine receptor antagonist and a potent ganglioblocker.
    Katalog #CAS NummerSummenformelMenge
    sc-25562930015-57-7C11H21N•HBr2 mg
  • Tempoxime hydrochloride
    A neuronal nicotinic AChR antagonist and potent ganglioblocker.
    Katalog #CAS NummerSummenformelMenge
    sc-30186663467-53-8C9H18N2O•HCl2 mg
  • tert-Butyl bicyclo[2.2.2]phosphorothionate
    GABAA receptor antagonist, chloride channel blocker and an extremely potent convulsant.
    Katalog #CAS NummerSummenformelMenge
    sc-25363370636-86-1C8H15O3PS2 mg
  • Tiapride hydrochloride
    D2 and D3 dopamine receptor antagonist; antipsychotic.
    Katalog #CAS NummerSummenformelMenge
    sc-25369751012-32-9C15H24N2O4S ·HCl5 g
  • TMPH hydrochloride
    A potent inhibitor of neuronal nicotinic receptors. Evaluation of nicotinic acetylcholine receptor subunits expressed in Xenopus laevis oocytes indicated that TMPH can produce a potent and long-lasting inhibition of neuronal nAChR formed by the pairwise combination of the most abundant neuronal alpha (i.e., alpha3 and alpha4) and beta subunits (beta2 and beta4), with relatively little effect, because of rapid reversibility of inhibition, on muscle-type (alpha1beta1gammadelta) or alpha7 receptors. However, the inhibition of neuronal beta subunit-containing receptors was also decreased if any of the nonessential subunits alpha5, alpha6, or beta3 were coexpressed. This decrease in inhibition is shown to be associated with a single amino acid present in the second transmembrane domain of these subunits. TMPH ability to relate the diverse central nervous system effects to specific nAChR subtypes makes it a helpful tool for studying the functional roles of nAChR.
    Katalog #CAS NummerSummenformelMenge
    sc-253705849461-91-2C16H32ClNO25 mg
  • Tobramycin Sulfate
    Used in the treatment of respiratory infection and cystic fibrosis.
    Katalog #CAS NummerSummenformelMenge
    sc-20586579645-27-5C18H37N5O9 ··· ·xH2SO4100 mg/500 mg
  • Todralazine hydrochloride
    Antihypertensive
    Katalog #CAS NummerSummenformelMenge
    sc-2537073778-76-5C11H12N4O2•HCl1 g
  • Toloxatone
    A reversible monoamine oxidase A inhibitor (MAOI) and antidepressant. Belongs to the aryloxazolidinones, a relatively new class of reversible monoamine oxidase A inhibitors (MAOI). Studies show that derivatives such as 3-aryloxazolidin-2-one (oxazolidinones), which are regularly used to treat gram positive infections, represent a new class of reversible as well as irreversible inhibitors for MAO-A and MAO-B enzymes that are able to inhibit protein synthesis and also used for neurodegenerative-type pathologies.
    Katalog #CAS NummerSummenformelMenge
    sc-25566529218-27-7C11H13NO310 mg
  • Trifluperidol hydrochloride
    Katalog #CAS NummerSummenformelMenge
    sc-2537572062-77-3C22H23F4NO2•HCl25 mg
  • Tropine 2-(phenylthio)butanoate oxalate salt
    Strong analgesic. Results in an increased release of acetylcholine at central muscarinic synapses.
    Katalog #CAS NummerSummenformelMenge
    sc-253806155059-55-5C20H27NO6S50 mg
  • U-99194 maleate
    A putative D3 antagonist with a 30-fold preference for the dopamine D3 compared to D2 receptor.
    Katalog #CAS NummerSummenformelMenge
    sc-253817234757-41-6C17H27NO2•C4H4O425 mg
  • Valacyclovir hydrochloride hydrate
    A potent inhibitor of viral DNA polymerase which serves as a prodrug of acyclovir that is useful in viral, AIDS, and immune system regulation research.
    Katalog #CAS NummerSummenformelMenge
    sc-216047124832-27-5 (anhydrous)C13H20N6O4•HCl•xH2O50 mg/250 mg
  • VU0029767
    VU0029767 is a selective, novel M1 positive allosteric modulator. M1 is a member of the muscarinic acetylcholine family of GPCRs (mAChRs) and is a therapeutic target for cognitive deficits in schizophrenia and Alzheimer's disease. VU0029767 increases both potency and efficacy of acetylcholine (ACh) at M1. VU0029767 also potentiates a mutant M1 receptor, as well as the effects of allosteric agonist TBPB. VU0029767 weakly increases ACh potency at M1 in phospholipase C and phospholipase D assays. This compound was discovered in conjuction with VU0090157 (different chemotype), another M1 modulator, which differs in its activities at the mutant form of M1, potentiation of TBPB, and phospholipase assays. The two modulators differentially regulate G protein signaling following M1 activation. Thus, VU0029767 and VU0090157 are valuable compounds when used together to tease out ligand-directed trafficking.
    Katalog #CAS NummerSummenformelMenge
    sc-253833326001-01-8C21H21N3O325 mg
  • VU255035 hydrate
    VU0255035 is the first highly selective antagonist at the orthosteric site of the M1 receptor (75-fold selective for M1 relative to other muscarininc subtypes and devoid of activity at other GPCRs, ion channels, transporters and kinases). There are no highly selective M1 muscarinic receptor antagonists. The existing non-selective drugs do not permit direct evaluation of the role of M1 receptors in CNS fucntions and do not premit therapeutic targeting of M1 receptors in various disease states in which M1 receptors are implicated (epilepsy, Parkinson's disease, attention and cognitive disorders, dystonia, etc).
    Katalog #CAS NummerSummenformelMenge
    sc-2583341135243-19-4 (anhydrous)C18H20N6O3S2•xH2O5 mg
  • WAY-100635 maleate salt
    Selective 5-HT1A Ser receptor antagonist.
    Katalog #CAS NummerSummenformelMenge
    sc-264493634908-75-1C25H34N4O2•C4H4O45 mg/50 mg
  • Xanthine amine congener
    Xanthine amine congener is a potent, nonselective adenosine receptor antagonist (A1 and A2B > A2A).
    Katalog #CAS NummerSummenformelMenge
    sc-25571796865-92-8C21H28N6O425 mg
  • Xli 093 hydrate
    Katalog #CAS NummerSummenformelMenge
    sc-264494646066-59-3 (anhydrous)C33H26N6O6•xH2O5 mg
  • Xylazine
    α2-adrenoceptor agonist, sedative, muscle relaxant.
    Katalog #CAS NummerSummenformelMenge
    sc-2538387361-61-7C12H16N2S1 g
  • Xylometazoline hydrochloride
    α-adrenoceptor agonist; imidazoline binding site ligand.
    Katalog #CAS NummerSummenformelMenge
    sc-2557191218-35-5C16H24N2 ·HCl5 g