| | Neurotransmitters and Drugs
- 1-(α,α,α-Trifluoro-m-tolyl)piperazine
Serotonin receptor agonist which has preference for 5-HT1B serotonin receptors.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-253869 | 15532-75-9 | C11H13F3N2 | 5 g |
- 1-Deoxyforskolin from Coleus forskohlii
| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-229786 | 72963-77-0 | C22H34O6 | 1 mg |
- 1-Methyl-4-(2'-methylphenyl)-1,2,3,6-tetrahydropyridine hydrochloride
Dopaminergic neurotoxin displaying higher toxicity than MPTP in mice. | Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-251522 | 102417-86-7 | C13H18ClN | 10 mg |
- 1-Methylhistamine dihydrochloride
Histaming metabolite obtained from histamine N-methyltransferase.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-258820 | 6481-48-7 | C6H11N3 ·2HCl | 25 mg |
- 1-Methylnicotinamide chloride
Niacin metabolite excreted via the urinary system.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-237583 | 1005-24-9 | C7H9N2OCl | 1 g |
- 1-Phenyl-1,3,8-triazaspiro[4.5]decan-4-one
| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-253946 | 1021-25-6 | C13H17N3O | 5 g |
- (1,2,5,6-Tetrahydropyridin-4-yl)methylphosphinic acid hydrate
A hybrid of isoguvacine and 3-APMPA designed to retain affinity for GABAC receptors but not to interact with GABAA or GABAB receptors.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-251571 | 182485-36-5 (anhydrous) | C6H12NO2P ·H2O | 10 mg |
- 1,3-Dimethyl-8-phenylxanthine
Selective A1 adenosine receptor antagonist.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-253981 | 961-45-5 | C13H12N4O2 | 100 mg |
- 1,4-Dihydro-2,6-dimethyl-4-(3-nitrophenyl)-3,5-pyridinedicarboxylic Acid 3-Methyl Ester
Derivative of 1,4-dihydropyridine used in the therapy and prevention of atherosclerotic degradation of arterial walls.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-213529 | 74936-72-4 | C16H16N2O6 | 100 mg |
- (1R,9S)-(−)-β-Hydrastine
| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-352027 | 118-08-1 | C21H21NO6 | 250 mg |
- 2-((3-Trifluoromethyl)phenyl)histamine dimaleate
Found to be the most potent and selective H1 histamine receptor agonist of a panel of compounds in functional in vitro studies on histamine H2, H3, and other neurotransmitter receptors. It showed better potency at the guinea pig H1 histamine receptor than at the human H1 histamine receptor (pKi : 5.9). The selectivity of 2-((3-Trifluoromethyl)phenyl)histamine dimaleate was found to be 2138 (H1:H2), > 64 (H1:H3), 1000 (H1:M3), 105 (H1: a1), 708 (H1:β1), and 71 (H1:5HT2A). This substance does not cross the blood-brain barrier.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-251656 | 162049-83-4 | C20H20F3N3O8 | 5 mg |
- 2-(Methylthio)adenosine 5'-diphosphate trisodium salt hydrate
A P2 purinoceptor agonist, which induces platelet aggregation and shape change and inhibits cyclic AMP accumulation in platelets exposed to prostaglandin E1. Compared with ADP, 2-methylthio-ADP was 3 to 5 times as active as an aggregating agent and 150 to 200 times as active as an inhibitor of cyclic AMP accumulation. Purinergic signaling may be an important factor in TSP-1-mediated cell-matrix and cell-cell interactions such as those occurring during development and repair.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-251675 | 475193-31-8 (anhydrous) | C11H14N5Na3O10P2S•xH2O | 5 mg |
- 2-(Methylthio)adenosine 5'-triphosphate tetrasodium salt hydrate
2-Methylthioadenosine triphosphate is a potent P2Y purinoceptor agonist| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-287618 | n.n. | C11H14N5Na4O13P3S•xH2O | 5 mg |
- (±)-2-Amino-6,7-dihydroxy-1,2,3,4-tetrahydronaphthalene hydrobromide
A dopamine receptor agonist.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-251693 | 13575-86-5 | C10H13NO2•HBr | 10 mg/25 mg |
- 2-Chloro-N6-cyclopentyladenosine hemihydrate
Highly selective A1 adenosine receptor agonist.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-251732 | 37739-05-2 (anhydrous) | C15H20ClN5O4•0.5 ·H2O | 10 mg |
- 2-Chloroadenosine triphosphate tetrasodium hydrate
P2Y purinoceptor agonist.
| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-288070 | n.n. | C10H11ClN5Na4O13P3•xH2O | 5 mg |
- 2-Ethylidene-1,5-dimethyl-3,3-diphenylpyrrolidine perchlorate
Metabolite of methadone. A useful marker in GC-MS analyses. | Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-251747 | 66729-78-0 | C20H23N•HClO4 | 10 mg |
- 2-Methylserotonin maleate salt
5-HT3 serotonin receptor agonist.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-251787 | 78263-91-9 | C11H14N2O•C4H4O4 | 50 mg |
- 3-(1H-Imidazol-4-yl)propyl di(p-fluorophenyl)methyl ether hydrochloride
H3 histamine receptor antagonist.
| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-298704 | n.n. | C19H18F2N2O•HCl | 10 mg |
- 3-(N-Acetylamino)-5-(N-decyl-N-methylamino)benzyl alcohol
Designed PKC activator, demonstrating an increase in the surface expression of BCA 225, a tumor-associated antigen, and various other cellular antigens in T47D cells. | Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-251920 | 103955-90-4 | C20H34N2O2 | 1 mg |
- 3-Amino-1-propanesulfonic acid sodium salt
GABAA receptor agonist.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-251937 | 81028-90-2 | C3H8NO3SNa | 1 g |
- 3-Hydroxy-4-methoxyphenethylamine hydrochloride
A dopamine metabolite.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-256512 | 645-33-0 | C9H13NO2•HCl | 25 mg/100 mg |
- 3-Methoxytyramine hydrochloride
This is a major metabolite of dopamine; a product of catechol O-methyltransferase.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-254500 | 1477-68-5 | CH3OC6H3-4-(OH)CH2CH2NH2··HCl | 100 mg |
- 3-Propylxanthine
Weak competitor antagonist at both A1 and A2 adenosine receptors.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-252035 | 41078-02-8 | C8H10N4O2 | 25 mg/250 mg |
- 3,4-Dihydroxy-DL-phenylalanine
Immediate precursor of dopamine. Product of tyrosine hydroxylase.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-256584 | 63-84-3 | C9H11NO4 | 1 g/5 g |
- 3,5,5,-Trimethyloxazolidine-2,4-dione
| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-232150 | 127-48-0 | C6H9NO3 | 1 g |
- [3S-(3α,4aβ,8aβ)]-N-(tert-Butyl)decahydro-3-isoquinolinecarboxamide
Fragment present in various HIV-1 protease inhibitors currently in clinical trials for AIDS treatment. | Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-209788 | 136465-81-1 | C14H26N2O | 1 g |
- 3α,21-Dihydroxy-5α-pregnan-20-one
Positive allosteric modulator of GABAA receptors.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-252069 | 567-02-2 | C21H34O3 | 5 mg |
- 4-Aminomethylbenzenesulfonamide hydrochloride
| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-226489 | 138-37-4 | C7H10N2O2S ·HCl | 25 g |
- 4-Deoxypyridoxine hydrochloride
Vitamin B6 antagonist.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-238830 | 148-51-6 | C8H11NO2•HCl | 500 mg |
- 4-Diphenylacetoxy-N-(2-chloroethyl)piperidine hydrochloride
An irreversible muscarinic acetylcholine receptor antagonist with essentially equivalent affinity for M1, M3, M4, and M5 receptors and a much lower affinity for M2 receptors.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-252148 | 130817-71-9 | C21H24ClNO2•HCl | 25 mg/100 mg |
- (±)4-Hydroxydebrisoquin
A major metabolite of debrisoquin. It is a very useful indicator for cytochrome P-450 polymorphism.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-200729 | 59333-79-8 | C10H13N3O | 10 mg/50 mg |
- 4-Phenylbenzaldoxime
| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-232958 | 40143-27-9 | C13H11NO | 1 g |
- 5-Carboxamidotryptamine maleate salt hemiethanolate
An agonist at 5-HT1A, 5-HT1B, 5-HT1D, 5-HT5 and 5-HT7 serotonin receptors.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-252258 | 74885-72-6 | C11H13N3O ·0.5 ·C2H6O ·C4H4O4 | 5 mg |
- 5-Hydroxyindole-3-acetic acid
A major serotonin metabolite.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-256921 | 54-16-0 | C10H9NO3 | 100 mg/500 mg |
- 5-Hydroxyindole-3-acetic acid (dicyclohexylammonium) salt
Major serotonin metabolite.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-256922 | 66866-39-5 | C22H32N2O3 | 100 mg |
- 5-Methylurapidil
Selective α1A-adrenoceptor antagonist that exhibits antihypertensive properties.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-254855 | 34661-85-3 | C21H31N5O3 | 10 mg/50 mg |
- 5α-Pregnane-3,11,20-trione
| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-227031 | 2089-06-7 | C21H30O3 | 50 mg |
- 6-Acetyl-7-deacetylforskolin
Antihypertensive also exhibiting positive ionotropic and adenyl cyclase activating properties. | Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-262766 | 64657-21-2 | C22H34O7 | 1 mg |
- 6-Nitroquipazine maleate salt
A potent and selective serotonin transport blocker.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-252301 | 77372-73-7 | C17H18N4O6 | 100 mg |
- 7-Benzyloxytryptamine
| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-239117 | 31677-75-5 | C17H18N2O | 100 mg |
- 7-Deacetyl-1-deoxyforskolin from Coleus forskohlii
| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-233676 | 121606-18-6 | C20H32O5 | 1 mg |
- (±)-7-Hydroxy-2-(di-n-propylamino)tetralin hydrobromide
A selective D3 dopamine receptor agonist; has a much weaker affinity for other dopamine receptor subtypes.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-252308 | 159795-63-8 | C16H25NO•HBr | 25 mg |
- 8-Bromoadenosine 5'-triphosphate sodium salt
P2X purinoceptor agonist with similar reactivity to ATP.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-252312 | 81035-56-5 | C10H15BrN5O13P3•Na | 5 mg |
- 9-Deoxyforskolin from Coleus forskohlii
| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-233726 | 84048-28-2 | C22H34O6 | 1 mg |
- 12β-Hydroxydigitoxin
This compound is a cardiac glycoside which serves as a substrate for Pgp. It upregulates Pgp expression and down regulates SXR (Steroid Xenobiotic Receptor).| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-213604 | 20830-75-5 | C41H64O14 | 1 g/5 g |
- α-Hydroxy-triazolam
Metabolite of triazolam.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-222434 | n.n. | C17H12Cl2N4O | 1 mg |
- α-Methylserotonin maleate salt
A salt of α-Methylserotonin maleate and a serotonin receptor agonist.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-254929 | 97469-12-0 | C11H14N2O ·C4H4O4 | 10 mg/50 mg |
- α5IA
A selective inverse agonist for a5 subtype of GABAA receptor with a higher intrincing efficacy to the a5 subtype than other drugs.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-252345 | 215874-86-5 | C17H14N8O2 | 5 mg |
- A-315456
A selective α1D-adrenoceptor antagonist.
| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-300143 | n.n. | C18H23N3O2S | 5 mg |
- A-317491 sodium salt hydrate
A non-nucleotide P2X3 and P2X2/3 receptor antagonist, which inhibits calcium flux mediated by the receptors. This compound can also bind to 86 other receptors, enzymes, and ion channels.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-300144 | n.n. | C33H27NO8•xNa+•yH2O | 5 mg |
- A-331440 dihydrochloride
A non-imidazole H3 histamine receptor antagonist. Presynaptic histamine H3 receptors regulate the release of histamine and other neurotransmitters, and histamine H3receptor antagonists enhance neurotransmitter release. A-331440 is a histamine H(3) receptor antagonist, which binds strongly and selectively to both human and rat histamine H3 receptors (K(i)=25 nM). Mice on a high-fat diet (45 kcal % lard) prior to 28-day oral b.i.d. dosing for measurement of obesity-related parameters. A-331440 administered at 0.5 mg/kg had no significant effect on weight, whereas 5 mg/kg decreased weight comparably to dexfenfluramine (10 mg/kg). A-331440 administered at 15 mg/kg reduced weight to a level comparable to mice on the low-fat diet. The two higher doses reduced body fat and the highest dose also normalized an insulin tolerance test. Both data shows that the histamine H3 receptor antagonist, A-331440, has potential as an antiobesity agent.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-252330 | 392338-13-5 (non-salt) | C22H27N3O•2HCl | 5 mg |
- Acamprosate Calcium
It is of interest for the treatment of alcoholism and other neurochemical disorders.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-210733 | 77337-73-6 | C10H20CaN2O8S2 | 100 mg |
- Acetyl Coenzyme A Trilithium Salt Trihydrate
Acetyl coenzyme A is an essential cofactor and carrier of acyl groups in enzymatic acetyl transfer reactions. Also the precursor for lipid biosynthesis and the neurotransmitter acetylcholine.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-291794 | 72-89-9 | C23H35Li3N7O17P3S ·3H2O | 1 mg/5 mg |
- Acetyl-β-methylcholine chloride
Metabolically stable analog of acetylcholine; muscarinic agonist. Its ability to constrict airway smooth muscle is used to assess bronchial reactivity in the laboratory and clinically.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-257063 | 62-51-1 | C8H18ClNO2 | 5 g/25 g |
- Acetylcholine bromide
This is an endogenous neurotransmitter at cholinergic synapses, which amplifies action potential of the sarcolemma thereby inducing muscle contractions.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-252350 | 66-23-9 | C7H16BrNO2 | 100 g |
- Acetylcholine perchlorate
| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-233810 | 927-86-6 | C7H16NO2•O4Cl | 5 g |
- Acetylthiocholine chloride
An acetylcholinesterase substrate and nicotinic acetylcholine receptor agonist.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-257066 | 6050-81-3 | C7H16ClNOS | 1 g |
- Adenosine amine congener hydrate
Potent aqueous-soluble A1 adenosine receptor agonist.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-254938 | 96760-69-9 (anhydrous) | C28H32N8O6•xH2O | 5 mg |
- Adiphenine hydrochloride
| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-233821 | 50-42-0 | C20H25NO2•HCl | 10 g |
- Alaproclate hydrochloride
Strong and selective serotonin uptake inhibitor.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-257075 | 60719-83-7 | C13H18ClNO2•HCl | 25 mg |
- Altanserin hydrochloride hydrate
This is a specific 5HT2/serotonergic antagonist.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-252365 | 76330-71-7 (non-salt) | C22H22FN3O2S•HCl•xH2O | 10 mg |
- ALX-1393
Inhibitor of the glycine transporter GlyT-2.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-300191 | n.n. | C23H22NO4F | 500 µg |
- Amcinonide
| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-227245 | 51022-69-6 | C28H35FO7 | 1 g |
- Amodiaquin dihydrochloride dihydrate
| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-233870 | 6398-98-7 | C20H22ClN3O•2HCl•2H2O | 5 g |
- Antazoline phosphate salt
An imidazoline agonist that is more potent than efaroxan in inducing insulin release from β cells; H1 histamine receptor antagonist.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-239251 | 154-68-7 | C17H22N3O4P | 1 g |
- Ara-G hydrate
An inducer of apoptosis inhibitor of DNA synthesis antimetabolite and antineoplastic. Ara-G is converted by cellular kinases to the active 5'-triphosphate, Ara-GTP. Incorporation of Ara-GTP into DNA leads to inhibition of DNA synthesis and apoptosis. The cellular accumulation of Ara-GTP is indicative of the clinical response to treatment with nelarabine, the prodrug. The differential accumulation and consequent selective cytotoxicity of Ara-G in T cells has been postulated to be due to the higher accumulation and slower elimination of ara-GTP in these cells. Nelarabine was developed because of poor water solubility of Ara-G, but Ara-G is DMSO-soluble. Nelarabine is approved in the United States for the treatment of T-cell acute lymphoblastic leukemia (T-ALL) and T-cell lymphoblastic lymphoma (T-LBL). | Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-214548 | 38819-10-2 (anhydrous) | C10H13N5O5 ·xH2O | 5 mg/25 mg |
- Arecaidine hydrochloride
| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-233889 | 6018-28-6 | C7H11NO2 ·HCl | 100 mg |
- Arecaidine propargyl ester hydrobromide
A potent muscarinic acetylcholine receptor agonist exhibiting slight selectivity for M2 receptors; inactive at nicotinic receptors.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-257091 | 116511-28-5 | C10H13NO2•HBr | 25 mg |
- Atropine
Competitive nonselective antagonist at central and peripheral muscarinic acetylcholine receptors.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-252392 | 51-55-8 | C17H23NO3 | 5 g |
- AZ11645373
A selective and potent human P2X7 purinoceptor antagonist. | Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-252394 | 227088-94-0 | C24H21N3O5S | 5 mg |
- β, γ-Methyleneadenosine 5'-triphosphate disodium salt
Selective P2X purinoceptor agonist which is more potent than ATP and less potent than α, β-methylene-L-adenosine 5'-triphosphate.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-253042 | 7414-56-4 | C11H16N5O12P3 ·2Na | 5 mg/10 mg |
- B-HT 933 dihydrochloride
A selective α2-adrenoceptor agonist.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-254951 | 36067-72-8 | C9H15N3O•2HCl | 5 mg |
- Bamethane hemisulfate salt
| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-233908 | 5716-20-1 | HOC6H4CH(OH)CH2NH(CH2)3CH3•1/2H2SO4 | 5 g |
- Benazoline oxalate salt
I2 imidazoline receptor agonist; has high affinity and selectivity for I2 imidazoline receptors over α-adrenoceptors.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-257119 | 1021868-82-5 | C13H12N2•C2H2O4 | 5 mg |
- Bendroflumethiazide
| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-233928 | 73-48-3 | C15H14F3N3O4S2 | 1 g |
- Benfotiamine
Lipid-soluble thiamine derivative used as a treatment for diabetic neuropathy. More effective at increasing thiamin levels in blood and tissues than water-soluble salts like the previous vitamin B1.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-204639 | 22457-89-2 | C19H23N4O6PS | 250 mg/1 g |
- Benoxathian hydrochloride
Selective α1-adrenoceptor antagonist.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-254954 | 92642-97-2 | C19H23NO4S•HCl | 10 mg |
- Benzbromarone
| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-233934 | 3562-84-3 | C17H12Br2O3 | 1 g |
- Bephenium hydroxynaphthoate
| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-234012 | 3818-50-6 | C17H22NO•C11H7O3 | 10 g |
- Bicyclol
A anti-hepatitis drug, used in China for chronic hepatitis B and presumably C. The drug appears to protect against liver injury in animals. Recently was reported that bicyclol induces the expression of hepatic HSP27 and HSP70, and consequently inhibits the transcription factor NF-?B-mediated apoptosis and necrosis in liver tissue. It appears that bicyclol induces hepatic HSP27 and HSP70 expression through the activation transcription of HSPs genes.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-252435 | 118159-48-1 | C19H18O9 | 5 mg |
- Bilobalide
Bilobalide is a terpenoid extracted from ginkgo biloba with neuroprotective, antibacterial, and inhibitory effects.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-201061 | 33570-04-6 | C15H18O8 | 10 mg/50 mg |
- BRL 35135A
BRL 35135A is an agonist for the β3-adrenoceptor.
| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-300301 | n.n. | C20H25BrClNO4 | 25 mg |
- BRL 37344 sodium salt hydrate
A selective β3-adrenoceptor agonist. Studies support the hypothesis that there are peripheral β3 adrenergic receptors that can reduce food intake and that central β2 or β3 adrenergic receptors mediate the peripheral effects of the β3 agonist.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-252513 | 127299-93-8 (anhydrous) | C19H21ClNNaO4•xH2O | 5 mg |
- BU224 hydrochloride
BU224 hydrochloride is an antagonist for the I2 Imidazoline receptor.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-300306 | 187173-05-3 | C12H11N3•HCl | 5 mg |
- Bufexamac
| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-227537 | 2438-72-4 | C12H17NO3 | 10 g |
- Buflomedil hydrochloride
| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-234225 | 35543-24-9 | C17H25NO4•HCl | 1 g |
- Bupivacaine hydrochloride
Na+ channel blocker, local anesthetic.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-252524 | 18010-40-7 | C18H28N2O··HCl | 1 g/5 g |
- Butacaine
| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-234227 | 149-16-6 | C18H30N2O2 | 1 g |
- (±)-Butaclamol hydrochloride
| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-234228 | 36504-94-6 | C25H31NO•HCl | 25 mg |
- (-)-Butaclamol hydrochloride
Dopamine receptor antagonist; less active enantiomer.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-252526 | 55528-08-0 | C25H31NO•HCl | 25 mg |
- (+)-Butaclamol hydrochloride
A dopamine D2 receptor antagonist. This compound is 2 to 4 times more active than its enantiomer at inhibiting the D2 receptor.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-252525 | 55528-07-9 | C25H31NO•HCl | 5 mg |
- Butethamate citrate salt
| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-227540 | 13900-12-4 | C16H25NO2 ·C6H8O7 | 5 g |
- Butoxamine hydrochloride
| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-234233 | 5696-15-1 | C15H25NO3 ·HCl | 50 mg |
- Camylofine dihydrochloride
| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-234275 | 54-30-8 | C19H32N2O2•2HCl | 1 g |
- Carbamyl-β-methylcholine chloride
| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-234279 | 590-63-6 | C7H17N2O2Cl | 5 g |
- Carprofen
A non-steroidal anti-inflammatory drug whose mechanism of action is dependent upon inhibiting the production of cox-2 and other sources of prostaglandins| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-205621 | 53716-49-7 | C15H12ClNO2 | 1 g/5 g |
- CAY10415
Potent antidiabetic drug that, when adminstered as a food admixture at 100 mg/kg for four days, effectively lowers blood glucose levels in obese, hyperglycemic, hyperinsulinemic, and insulin-resistant KKAy mice. Also shown to enhance the rate of insulin-stimulated lipogenesis in 3T3-L1 adipocytes in a dose-dependent manner.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-205236 | 146062-49-9 | C19H18N2O4S | 1 mg/10 mg |
- Cefadroxil
| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-234291 | 50370-12-2 | C16H17N3O5S | 1 g |
- Cerivastatin Lactone
Synthesized statin used to lower cholesterol and prevent cardiovascular disease.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-204679 | 145599-86-6 | C26H32FNO4 | 5 mg/10 mg |
- CGP 35348 hydrate
A GABAB-receptor antagonist.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-252561 | 123690-79-9 (non-salt) | C8H20NO4P•xH2O | 5 mg |
- CGS-21680 hydrochloride hydrate
An adenosine receptor agonist that possesses selectivity for A2 verses A1 receptors.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-252562 | 124182-57-6 (anhydrous) | C23H29N7O6•HCl•xH2O | 5 mg/10 mg |
- Chloro-APB hydrobromide
Full D1 dopamine receptor agonist.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-252573 | 80751-65-1 | C19H20ClNO2•HBr | 5 mg/25 mg |
- Chlorocitalopram
This compound is an internal standard of Citalopram, as well as an uptake inhibitor of serotonin (5-HT).| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-207423 | 64169-57-9 | C20H21ClN2O | 1 mg |
- Chlorocitalopram, Hydrobromide
An internal standard of Citalopram which is also an uptake inhibitor of serotonin (5-HT).| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-207424 | 64169-58-0 | C20H22BrClN2O | 1 mg |
- Chloroethylclonidine dihydrochloride
An rreversible α1B-adrenoceptor alkylating agent.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-252587 | 98086-36-3 | C13H17Cl3N4•2HCl | 10 mg/25 mg |
- Chloropyramine hydrochloride
| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-234345 | 6170-42-9 | C16H20ClN3•HCl | 1 g |
- Chlorzoxazone
Muscle relaxant (skeletal).| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-211078 | 95-25-0 | C7H4ClNO2 | 10 mg |
- Choline bitartrate
Acyl group acceptor| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-252599 | 87-67-2 | C9H19NO7 | 100 g |
- CI 1020
Highly selective, orally active, non-peptide endothelin-A receptor (ETA) antagonist (IC50 values are 0.3 and 480 nM for ETA and ETB receptors respectively). Antihypertensive; blocks ET-1-induced pressor responses following oral administration. | Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-204687 | 162256-50-0 | C28H26O9 | 10 mg/50 mg |
- Cinchonine hemisulfate salt
| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-234360 | 5949-16-6 | C19H22N2O•1/2H2SO4 | 100 g |
- Ciproxifan hydrochloride
Ciproxifan belongs to a novel chemical series of histamine H3-receptor antagonists. In vitro, it behaved as a competitive antagonist at the H3 autoreceptor controlling 3H histamine release from synaptosomes and displayed similar Ki values (0.5-1.9 nM) at the H3 receptor controlling the electrically-induced contraction of guinea pig ileum or at the brain H3 receptor labeled with 125I-iodoproxyfan. This appears to be an orally bioavailable, extremely selective and potent H3-receptor antagonist whose vigilance- and attention-promoting effects are promising for therapeutic applications in aging disorders.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-257245 | 1049741-81-2 | C16H18N2O2•HCl | 5 mg |
- Ciproxifan maleate
Strong, selective H3 histamine receptor antagonist.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-252608 | 184025-19-2 | C16H18N2O2•C4H4O4 | 5 mg |
- cis-Entacapone
An antiparkinsonian (Z)-Isomer of Entacapone polymorphic form B. | Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-214739 | 145195-63-7 | C14H15N3O5 | 2.5 mg |
- Cisapride monohydrate
5-HT4 serotonin receptor agonist| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-252619 | 260779-88-2 | C23H29N3O4ClF•H2O | 10 mg |
- Clenbuterol Hydrochloride
β2-adrenoreceptor agonist with ability to potentiate hyopxemia due to increased shunt fraction in horses anesthetized via IV. Has also been shown to enhance memory in sham-lesioned male Sprague Dawley rats.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-205635 | 21898-19-1 | C12H18Cl2N2O ·HCl | 25 mg/100 mg |
- Clioquinol
A metal chelating ligand and a member of the hydroxyquinoline family, which inhibits certain enzymes related to DNA replication.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-201066 | 130-26-7 | C9H5ClINO | 1 g/5 g |
- Clofazimine
| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-234402 | 2030-63-9 | C27H22Cl2N4 | 5 g |
- Clofibric acid
A compound that reduces cholesterol levels in blood through diminishing the activity of NADPH.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-203000 | 882-09-7 | C10H11ClO3 | 10 g/50 g |
- Clofoctol
| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-234403 | 37693-01-9 | C21H26Cl2O | 1 g |
- Cloperastine hydrochloride
| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-234405 | 14984-68-0 | C20H24ClNO•HCl | 10 g |
- Clozapine N-oxide
Major metabolite of Clozapine (sc-200402). Observed to to decrease 5-HT2 serotonin receptor density in vitro.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-201111 | 34233-69-7 | C18H19ClN4O | 5 mg/25 mg |
- Condelphine
A nicotinic acetylcholine receptor antagonist.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-252625 | 7633-69-4 | C25H39NO6 | 20 mg |
- Cyclazosin hydrochloride
α1B-adrenoceptor antagonist.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-239599 | 146929-33-1 | C23H27N5O4•HCl | 5 mg |
- Cysteamine S-phosphate sodium salt
| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-234499 | 3724-89-8 | C2H7NO3PSNa | 50 mg |
- D-Tryptophan
An unnatural isomer of tryptophan.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-255066 | 153-94-6 | C11H12N2O2 | 5 g/25 g |
- DEABL
Anticonvulsant; positive modulator of GABAA receptor| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-252664 | 175698-05-2 | C8H15NO | 50 mg |
- Deacetylforskolin
| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-234516 | 64657-20-1 | C20H32O6 | 1 mg |
- Debrisoquin sulfate (Ro 5-3307)
This is an antihypertensive. It is metabolized to 4-hydroxydebrisoquin by debrisoquin 4-hydroxylase. Useful indicator for cytochrome P-450 polymorphism. | Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-200725 | 581-88-4 | C20H28N6O4S | 50 mg/500 mg |
- Delsoline
Nicotinic receptor antagonist, ganglion blocker; exhibits weak affinity at brain α-bungarotoxin-sensitive nicotinic acetylcholine receptors.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-252666 | 509-18-2 | C25H41NO7 | 20 mg |
- Desoximetasone
| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-234529 | 382-67-2 | C22H29FO4 | 1 g |
- Despropionylfentanyl
| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-221537 | 21409-26-7 | C19H24N2 | 1 mg/10 mg |
- Desvenlafaxine hydrochloride
A dual SERT/NET reuptake inhibitor and a major active metabolite of venlafaxine. A brain penetrant.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-255071 | 300827-87-6 | C16H25NO2•HCl | 10 mg |
- Diacerein
An interleukin-1 inhibitor used for treating osteoarthritis. | Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-204717 | 13739-02-1 | C19H12O8 | 50 mg/250 mg |
- Diaveridine
A coccidiostat and antiprotozoal drug. | Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-205646 | 5355-16-8 | C13H16N4O2 | 1 g/10 g |
- Diethylstilbestrol dipropionate
| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-227859 | 130-80-3 | C24H28O4 | 1 g |
- Diflorasone diacetate
| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-227861 | 33564-31-7 | C26H32F2O7 | 100 mg |
- Dihydroergotamine (+)-tartrate salt
Vasoconstrictor and vascular serotonin receptor agonist. Also exhibits alpha-adrenergic and dopamine D2 receptor partial agonist activity.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-263091 | 5989-77-5 | (C33H37N5O5)2•C4H6O6 | 50 mg |
- Dihydrotachysterol
| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-234695 | 67-96-9 | C28H46O | 50 mg |
- Dimenhydrinate
| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-234708 | 523-87-5 | C17H21NO•C7H7ClN4O2 | 10 g |
- Diminazene Aceturate
An anti-protozoal drug and anti-trypanosomal.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-205651 | 908-54-3 | C14H15N7•2C4H7NO3 | 1 g/5 g |
- Diperodon hydrochloride
| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-234775 | 537-12-2 | C22H27N3O4•HCl | 5 g |
- Dipyrone
A non-steroidal anti-inflammatory drug that, when coadministered with morphine, potentiates its antinociceptive action and delays the development of tolerance. Dipyrone is a selective inhibitor of cyclooxygenase-3 (COX-3), with lower activity against COX-1 and no activity against COX-2. This also blocks PGE2-induced hyperalgesia in several models.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-252755 | 68-89-3 | C13H16N3O4SNa | 25 g |
- Diquine
A nicotinic cholinoreceptor antagonist at the neuromuscular junction which is a curare-like ganglioblocker.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-255119 | 3563-63-1 | C34H50Cl2N2 | 2 mg |
- Dithiobiuret
Paralytic agent.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-252760 | 541-53-7 | C2H5N3S2 | 100 mg |
- DL-threo-β-(3,4-Dihydroxyphenyl)serine
An amino acid precursor of noradrenaline (NA); elevates the concentration of NA in the brain.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-252764 | 3916-18-5 | C9H11NO5 | 1 g |
- Dothiepin hydrochloride
Dothiepin hydrochloride is a tricyclic antidepressant.
| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-300503 | 897-15-4 | C19H21NS ·HCl | 5 mg |
- Doxazosin Mesylate
An alpha-blocker drug. It reduces progression of benign prostatic hyperplasia.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-205656 | 77883-43-3 | C24H29N5O8S | 50 mg/250 mg |
- Drofenine hydrochloride
| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-234845 | 548-66-3 | C20H31NO2•HCl | 10 g |
- (±)-Dropropizine
| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-234846 | 17692-31-8 | C13H20N2O2 | 5 g |
- DS1
Potently (low nM) enhances GABA-evoked currents mediated by α4β3δ receptors. It has little effect on GABA responses mediated by α4β3 2 receptors. At similar concentrations, DS1 directly activates this receptor and is the most potent known agonist of α4β3δ receptors. This compound has an opportunity to be become an agonist golden stardard for δ-GABAA receptors.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-252769 | 372497-52-4 | C18H10Br2ClN3OS | 5 mg |
- Dyclonine, Hydrochloride
Used as a local anesthetic.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-211385 | 536-43-6 | C18H28ClNO2 | 25 g |
- Eletriptan Free Base
Used in the treatment of migraine headaches.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-204736 | 143322-58-1 | C22H26N2O2S | 1 mg/5 mg |
- (-)-Epinephrine
A predominent neurotransmitter. Found to be effective beta2-agonist bronchodilator.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-205674 | 51-43-4 | C9H13NO3 | 1 g/5 g |
- (±)-Epinephrine
| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-252779 | 329-65-7 | C9H13NO3 | 5 g/25 g |
- (±)-Epinephrine hydrochloride
Adrenergic receptor agonist.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-252780 | 329-63-5 | C9H13NO3 ·HCl | 5 g |
- Etbicythionat
A potent non-competitive GABA antagonist in mammals. Causes epileptiform seizures.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-252786 | 224790-71-0 | C6H11O3PS | 100 µg |
- Ethylhydrocupreine
| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-235094 | 522-60-1 | C21H28N2O2 | 5 g |
- Ethylhydrocupreine hydrochloride
Sensitive and specific reagent for the identification of Streptococcus pneumoniae. | Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-255166 | 3413-58-9 | n.n. | 100 mg/1 g |
- Famprofazone
| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-235122 | 22881-35-2 | C24H31N3O | 10 g |
- FAUC 213
A highly selective D4 dopamine receptor full antagonist.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-252820 | 337972-47-1 | C18H19ClN4 | 5 mg |
- Fenoprofen calcium salt hydrate
| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-239989 | 53746-45-5 | C30H26O6Ca. ·xH2O | 5 g |
- Fenoterol hydrobromide
A β2-adrenoceptor agonist. Bronchodilator.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-252822 | 1944-12-3 | C17H21NO4•HBr | 1 g |
- Fiduxosin hydrochloride
Has been shown to be an α1-Adrenoceptor antagonist.
| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-300692 | 208992-74-9 | C30H29N5O4S•HCl | 5 mg |
- Fipexide HCl
Fipexide has been shown to be a nootropic agent and possible mild dopamine agonist.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-201065 | 34161-23-4 | C20H21ClN2O4 ·HCl | 1 g |
- Fipexide hydrochloride
| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-235136 | 34161-24-5 | C20H21ClN2O4•HCl | 5 g |
- Flucybene
A potent non-competitive GABA antagonist in mammals, molluscs and insects; convulsant.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-252825 | 3289-22-3 | C11H8F6N2 | 1 mg |
- Fluorocurarine chloride
A short-acting selective sympathetic ganglioblocker with weak antagonist activity on the nicotinic receptor at the neuromuscular junction. Hypotensive.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-252829 | 22273-09-2 | C20H23ClN2O | 20 mg |
- Fluspirilene
Dopamine receptor antagonist; calcium channel blocker; antipsychotic.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-252832 | 1841-19-6 | C29H31F2N3O | 10 mg |
- FSCPX
Irreversible A1 adenosine receptor antagonist.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-252841 | 156547-56-7 | C23H27FN4O6S | 25 mg |
- gamma-oryzanol
| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-295006 | 11042-64-1 | C40H58O4 | 25 g/250 g |
- Gefitinib
An epidermal growth factor receptor (EGFR)-tyrosine kinase inhibitor that has been shown to increase phosphorylation of c-Jun NH2 -terminal kinase (JNK) and p38 mitogen-activated protein kinase (MAPK) in HaCaT cells.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-202166 | 184475-35-2 | C22H24ClFN4O3 | 100 mg/250 mg |
- Glycine hydrochloride
Spinal cord inhibitory neurotransmitter. Also allosterically regulates NMDA receptors. | Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-263346 | 6000-43-7 | C2H5NO2 ·HCl | 100 g/500 g |
- Guaifenesin
An expectorant reported to have muscle relaxant and sedative activity, where it is often used as anesthetic during animal surgery.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-205710 | 93-14-1 | C10H14O4 | 25 g/100 g |
- Guvacine hydrochloride
Inhibits GABA uptake.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-263347 | 6027-91-4 | C6H9NO2•HCl | 25 mg |
- Hemicholinium-3
A potent and selective choline uptake blocker.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-252873 | 312-45-8 | C24H34Br2N2O4 | 100 mg |
- Hesperetin
A dietary flavanone with a chemopreventive effect.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-252878 | 69097-99-0 | C16H14O6 | 1 g |
- Hexamethonium chloride
A preferential nicotinic receptor blocker at the level of autonomic ganglia. Has been shown to cross the blood-brain barrier only in high doses. | Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-263383 | 60-25-3 | (CH3)3N(Cl)(CH2)6N(Cl)(CH3)3 | 5 g |
- Hexestrol dipropionate
| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-250111 | 4825-53-0 | C24H30O4 | 5 g |
- Hydrastinine hydrochloride
| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-250124 | 4884-68-8 | C11H13NO3•HCl | 100 mg |
- Hydrocortisone 17-valerate
| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-235332 | 57524-89-7 | C26H38O6 | 500 mg |
- Hydrocortisone 21-hemisuccinate
| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-228319 | 2203-97-6 | C25H34O8 | 1 g |
- Hydroxocobalamin hydrochloride
| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-235336 | 58288-50-9 | C62H89CoN13O15P•HCl | 100 mg |
- Hydroxyzine pamoate salt
| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-228327 | 10246-75-0 | C44H43ClN2O8 | 10 g |
- I-AB-MECA
A reference standard used for radioiodinated I-AB-MECA. This is a widely used, high affinity radioligand for the A3 adenosine receptor.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-250141 | 152918-27-9 | C18H20IN7O4 | 1 mg |
- Imidazole-4-acetic acid sodium salt
Competitive antagonist at GABAC receptors.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-252900 | 56368-58-2 | C5H5N2NaO2 | 500 mg/1 g |
- Imipramine N-oxide
The tertiary amine-oxidized metabolite of Imipramine. A useful standard for investigating FMO-mediated oxidation activity with Imipramine as a substrate. | Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-200973 | 6829-98-7 | C19H24N2O | 5 mg/25 mg |
- Indapamide
An antihypertensive agent that reduces intracellular calcium levels. Maintains magnesium ion but reduces phosphate ions involved in arterial rigidity and many other functions.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-204777 | 26807-65-8 | C6H16ClN3O3S | 250 mg/1 g |
- Indoramin hydrochloride
α1-adrenoceptor antagonist.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-252906 | 38821-52-2 | C22H26ClN3O | 10 mg |
- Ipratropium bromide monohydrate
N-isopropyl quaternary salt of atropine. A nonselective muscarinic acetylcholine receptor antagonist; bronchodilator.
| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-252911 | 66985-17-9 | C20H31BrNO3 | 250 mg |
- Isoetharine mesylate salt
β-Adrenergic receptor agonist, bronchodilator.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-252918 | 7279-75-6 | C13H21NO3 ·CH4O3S | 1 g |
- (-)-Isoproterenol (+)-bitartrate salt
β-Adrenoceptor agonist. increases cytosolic cAMP.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-252926 | 54750-10-6 | C11H17NO3 ·C4H6O6 | 100 mg/500 mg |
- Isosilybin
Useful in the treatment of liver disease.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-215199 | 72581-71-6 | C25H22O10 | 1 mg |
- JNJ7777120
A potent, selective non-imidazole H4 histamine receptor antagonist.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-252930 | 459168-41-3 | C14H16N3OCl | 5 mg |
- Kisspeptin-234 trifluoroacetate salt
| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-300857 | n.n. | C63H76N17O14•xC2HF3O2 | 1 mg |
- L-741,626
A selective antagonist of the dopamine D2 receptor.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-252936 | 81226-60-0 | C20H21ClN2O | 10 mg |
- L-Allylglycine
A Glutamic acid decarboxylase inhibitor.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-255236 | 16338-48-0 | C5H9NO2 | 500 mg |
- L-Cysteinesulfinic acid monohydrate
A putative excitatory amino acid neurotransmitter.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-215212 | 207121-48-0 | C3H7NO4S•H2O | 100 mg/250 mg |
- L-Glutamic acid monosodium salt hydrate
An excitatory amino acid neurotransmitter which is an agonist at kainate, quisqualate and NMDA receptors.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-215218 | 142-47-2 (anhydrous) | C5H8NNaO4•xH2O | 100 g/500 g |
- L-Histidine monohydrochloride monohydrate
Histamine precursor via histidine decarboxylase.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-263442 | 5934-29-2 | C6H9N3O2•HCl•H2O | 5 g/25 g |
- L-Tyrosine disodium salt hydrate
This is an amino acid precursor of dopamine and other catecholamines.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-252940 | 69847-45-6 | C9H9NNa2O3•xH2O | 25 g/100 g |
- Labetalol hydrochloride
Competitive β-adrenoceptor antagonist.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-252942 | 32780-64-6 | C19H24N2O3 ·HCl | 5 g |
- Lapatinib Ditosylate
A selective and effective inhibitor of ErbB-2 and EGFR dual tyrosine kinases. Research studies have reported that the compound can inhibit breast cancer cell proliferation. | Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-202205 | 388082-78-8 | C29H26ClFN4O4S ·2C7H8O3S | 10 mg/25 mg |
- Lofepramine hydrochloride
An antidepressant and a serotonin and norepinephrine re-uptake inhibitor (SNRI).| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-255256 | 26786-32-3 | C26H28Cl2N2O | 5 mg |
- Lupinine
An alkaloid isolate from Anabisis aphylla. Able to reduce the effect of ethanol anesthesia. | Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-205737 | 486-70-4 | C10H19NO | 25 mg/100 mg |
- LY-165,163
Selective 5-HT1A and 5-HT1D serotonin receptor antagonists.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-252977 | 1814-64-8 | C19H22F3N3 | 25 mg |
- m-Tyramine hydrochloride
| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-255257 | 3458-98-8 | C8H11NO··HCl | 100 mg |
- MADAM dihydrochloride
High affinity ligand for the serotonin transporter SERT| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-252980 | 411208-45-2 | C16H22Cl2N2S | 5 mg |
- Magnesium L-aspartate salt
| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-295263 | 18962-61-3 | n.n. | 25 g |
- Mebeverine hydrochloride
| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-235579 | 2753-45-9 | C25H35NO5•HCl | 10 g |
- Mebhydroline 1,5-naphthalenedisulfonate salt
Antagonist to H1 Histamine receptors.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-263459 | 6153-33-9 | C19H20N2 ·1/2C10H8O6S2 | 1 g |
- Melphalan
Cytotoxic drug used to treat multiple myeloma. Phenylamine derivative of mechorethamine.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-204799 | 148-82-3 | C13H18Cl2N2O2 | 100 mg/250 mg |
- Mepirizole
| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-235589 | 18694-40-1 | C11H14N4O2 | 10 g |
- Metaproterenol hemisulfate salt
This compound is a β2-adrenoceptor agonist.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-257701 | 5874-97-5 | C22H36N2O10S | 1 g |
- Metaraminol (+)-bitartrate salt
An α-adrenoceptor agonist.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-253004 | 33402-03-8 | C9H13NO2•C4H6O6 | 1 g |
- Methazolamide
| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-235615 | 554-57-4 | C5H8N4O3S2 | 1 g |
- Methiothepin mesylate salt
Methiothepin mesylate salt is a 5-HT1, 5-HT6, 5-HT7 serotonin receptor antagonist that blocks serotonin auto receptors.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-253005 | 74611-28-2 | C20H24N2S2•CH3SO3H | 100 mg |
- Methoctramine hydrate
This is a selective M2 muscarinic receptor antagonist at nM concentrations. At mM concentrations, methoctramine directly inhibits the high affinity GTPase activity of G proteins. The increase in calcium and arachidonic acid release were attenuated by the M2 receptor antagonist methoctramine, this is not only by the M3 receptor antagonist p-fluoro-hexahydro siladifenidol.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-257709 | 104807-46-7 (anhydrous) | C36H62N4O2•4HCl•xH2O | 10 mg/25 mg |
- Methoxamine hydrochloride
Agonist to alpha-1-adrenoceptors. | Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-263468 | 61-16-5 | C11H17NO3•HCl | 500 mg |
- Methyl 6-Methoxy-2-naphthylacetate
A potential prodrug.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-211871 | 23981-48-8 | C14H14O3 | 25 mg |
- Methyllycaconitine citrate hydrate
A potent and specific nicotinic receptor antagonist that binds to neuronal α-bungarotoxin sites.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-253043 | 21019-30-7 (non-salt) | C43H58N2O17 | 5 mg |
- Metoclopramide hydrochloride
This is a D2 antagonist and a 5-HT3 antagonist. Antipsychotic. Anti-emetic.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-253046 | 7232-21-5 | C14H22ClN3O2•HCl | 10 g/25 g |
- Metrazoline
A potent and selective imidazoline binding site ligand.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-253047 | 221225-04-3 | C14H16N2O4 | 5 mg |
- Minaprine dihydrochloride
Antidepressant| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-253049 | 25905-77-5 | C17H22N4O•2HCl | 1 g |
- MK-912 hydrate
A selective α2-adrenoceptor antagonist.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-253050 | 119942-70-0 (anhydrous) | C20H25N3O2•HCl•xH2O | 5 mg |
- Moguisteine
An anti-tussive with similar properties to codeine.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-204810 | 119637-67-1 | C16H21NO5S | 100 mg/250 mg |
- Montelukast Sodium
A potent, selective CysLT1 receptor antagonist (IC50 < 5nM), competitive with respect to LTD4, with no appreciable affect on the CysLT2 receptor.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-202231 | 151767-02-1 | C35H35ClNO3S•Na | 10 mg/25 mg |
- Mosapride citrate dihydrate
Antagonist to both 5-HT4 and 5-HT3 receptors.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-263722 | 636582-62-2 | C21H25ClFN3O3 ·C6H8O7 ·2H2O | 10 mg |
- Moxisylyte hydrochloride
α1-adrenoceptor antagonist; peripheral vasodilator.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-255308 | 964-52-3 | C16H25NO3•HCl | 1 g/5 g |
- MPP+ iodide
MPP+ iodide is an active metabolite of dopaminergic neurotoxin MPTP.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-255309 | 36913-39-0 | C12H12IN | 100 mg |
- MRS 1191
A selective A3 adenosine receptor antagonist. Selective for both human and rat.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-253056 | 185222-90-6 | C31H27NO4 | 2 mg |
- MRS 1523
A selective A3 adenosine receptor antagonist in the rat.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-253057 | 212329-37-8 | C23H29NO3S | 5 mg |
- MRS 2179 ammonium salt hydrate
Competitive to P2Y1 puinoreceptor antagonist.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-253058 | 101204-49-3 (non-salt) | C11H17N5O9P2•xNH3•yH2O | 5 mg |
- MRS 2395
An antagonist for the P2Y12 purinoceptor, which causes platelet aggregation in rats via ADP induction.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-253059 | 491611-55-3 | C20H30ClN5O4 | 5 mg |
- MSX-3 hydrate
A selective A2A adenosine receptor antagonist prodrug.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-255310 | 261717-23-1 (anhydrous) | C21H21N4O7PNa2•xH2O | 5 mg |
- (+)-Muscarine chloride
Active enantiomer; prototype muscarinic acetylcholine receptor agonist.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-253060 | 2303-35-7 | C9H20ClNO2 | 5 mg |
- (±)-Muscarine chloride hydrate
A muscarinic acetylcholine receptor agonist which was originally isolated from Amanita muscaria.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-255311 | 2936-25-6 (anhydrous) | C9H20ClNO2•xH2O | 5 mg |
- (+)-Muscarine iodide
| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-362769 | 24570-49-8 | C9H20INO2 | 10 mg |
- N -Methyl-5-hydroxy trypt amine oxalate salt
A serotonin receptor ligand.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-253061 | 1975-81-1 | C13H16N2O5 | 500 mg |
- N-Acetyl-N-acetoxy-4-chlorobenzenesulfonamide
A pro-drug of the potent vasorelaxant nitroxyl, H-N=O, which it slowly releases in neutral solution. HNO eventually dimerizes and dehydrates to N2O, without producing NO. | Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-203441 | 142867-52-5 | C10H10CINO5S | 10 mg/50 mg |
- N-Desmethylclozapine
A major metabolite of clozapine (sc-200402), found to act as a potent antagonist of the 5-HT1C serotonin receptor, and a moderate agonist of M(1) mAChR.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-201113 | 6104-71-8 | C17H17ClN4 | 5 mg/25 mg |
- N-Methyl dopamine hydrochloride
Used as an internal standard for catecholamine analyses.
Dopamine receptor agonist, α-adrenoceptor agonist.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-358430 | 62-32-8 | C9H13NO2•HCl | 25 mg/50 mg |
- N-Methylhistaprodifen dioxalate salt
More potent than a histamine by a factor of 3.5 on guinea pig ileum and more potent than histamine by a factor of 4.3 on guinea pig arterial H1-receptor-mediated vasoconstriction. The most potent H1-receptor agonist on the guinea pig ileum out of 17 agonists tested. Does not stimulate H2 and H3 histamine receptors and has potential use in the study of H1-receptor-mediated physiological and pathophysiological functions.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-255360 | 270079-48-6 | C21H25N3•2 ·C2H2O4 | 5 mg |
- (-)-N-Methylphysostigmine
| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-236078 | 103877-07-2 | C16H23N3O2 | 5 mg |
- N-Methylspiperone hydrochloride
A D2 dopamine receptor antagonist.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-253121 | 87539-19-3 | C24H28FN3O2•HCl | 5 mg |
- N,N-Dipropyl-5-carboxamidotryptamine maleate salt
A selective and potent 5-HT1A serotonin receptor agonist.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-253151 | 74885-25-9 | C17H25N3O ·C4H4O4 | 5 mg |
- Nα-Methylhistamine dihydrochloride
Production of N-alpha-methyl-histamine, which is a histamine 3 receptor (H3R) agonist, is promoted in Helicobacter pylori infected human gastric mucosa. NAMH acts directly on H2Rs in animals to stimulate acid secretion and to be a H2R agonist. NAMH dose dependently stimulated cAMP productions in CHO-H2R cells. This production was inhibited by famotidine but not by thioperamide. Control CHO cells were unresponsive to either histamine or NAMH. In addition, the effect of NAMH, in terms of cAMP production in CHO-H2R cells, was more potent than that of histamine-that is, with a lower EC50 concentration and higher maximal cAMP production. Both NAMH and histamine, but not R-alpha-methyl-histamine, effectively inhibited [(3)H] tiotidine binding to CHO-H2R cells. These results confirm that NAMH, which is produced in the gastric mucosa by H pylori, is a potent H2R agonist as well as a H3R agonist.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-253174 | 16503-22-3 | C6H11N3•2HCl | 10 mg |
- N6-(2-Phenylethyl)adenosine
Selective A1 adenosine receptor agonist.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-253168 | 20125-39-7 | C18H21N5O4 | 10 mg |
- (-)-N6-(2-Phenylisopropyl)adenosine
A1 adenosine receptor agonist. Its affinity for adenosine receptor is approximately 100x that of the (+)-isomer.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-253169 | 38594-96-6 | C19H23N5O4 | 25 mg |
- N6-2-(4-Aminophenyl)ethyladenosine
A potent, non-selective A3 adenosine receptor agonist.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-253170 | 89705-21-5 | C18H22N6O4 | 25 mg |
- N6-Cyclohexyladenosine
Selective A1 adenosine receptor agonist.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-255385 | 36396-99-3 | C16H23N5O4 | 50 mg |
- N8-Acetylspermidine dihydrochloride
| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-236151 | 34450-15-2 | C9H21N3O•2HCl | 100 mg |
- Nadolol
A polar and hydrophilic, non-selective β blocker, which displays activity against β-1 and β-2 receptors. It is known that Nadolol inhibits the release of catecholamines from the adrenal glands.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-253175 | 42200-33-9 | C17H27NO4 | 1 g |
- Nafronyl oxalate salt
Exhibits properties of a vasodilator.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-253176 | 3200-06-4 | C24H33NO3•C2H2O4 | 5 g |
- Naftopidil hydrochloride hydrate
Antihypertensive and antagonist to α1-adrenoceptor.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-263941 | 57149-07-2 (non-salt) | C24H28N2O3•xHCl•yH2O | 25 mg |
- NCS-356 sodium salt hydrate
γ-Hydroxybutyrate (GHB) receptor agonist.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-253182 | 430440-66-7 | C10H8ClO3Na•xH2O | 50 mg |
- Nefiracetam
A nootropic drug of the racetam family. Used to treat Alzheimer’s disease and other diseases related to learning and memory deficits. | Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-205766 | 77191-36-7 | C14H18N2O2 | 100 mg/250 mg |
- Nifekalant Hydrochloride
A class III antiarrhythmic drug that has shown to be effective against ventricular tachyarrhythmias by inhibiting HERG channels in a voltage-dependent and frequency-dependent manner.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-204819 | 130656-51-8 | C19H27N5O5 ·HCl | 10 mg/25 mg |
- Nifenazone
| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-236175 | 2139-47-1 | C17H16N4O2 | 5 g |
- (±)-Norepinephrine (+)-bitartrate salt
An adrenergic neurotransmitter.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-255396 | 3414-63-9 | C8H11NO3•C4H6O6 | 1 g |
- (+)-Norfenfluramine hydrochloride
(+)-Norfenfluramine is the major hepatic metabolite of (+)-fenfluramine and is primarily responsible for the anorexic effect, as well as side effects; (+)-norfenfluramine causes vasoconstriction and a blood pressure increase in rats with normal blood; more potent than fenfluramine at inducing dopamine release; acts primarily on the cytoplasmic pool of serotonin.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-253200 | 37936-89-3 | C10H12F3N ·HCl | 10 mg |
- Norfentanyl
Major urinary metabolite of a narcotic analgesic fentanyl.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-222077 | 1609-66-1 | C14H20N2O | 1 mg/10 mg |
- Nylidrin hydrochloride
| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-358467 | 849-55-8 | C19H25NO2•HCl | 200 mg/5 g |
- Octoclothepin maleate salt
5-HT2 serotonin receptor antagonist; D2 dopamine receptor antagonist.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-253215 | 4789-68-8 | C23H25ClN2O4S | 25 mg |
- Opiorphin
A natural analgesic that is secreted into human saliva. Opiorphin demonstrates dual-inhibitory potency on the enkephalin-inactivating ectopeptidases human NEP (hNEP) and human AP-N (hAP-N). As an analgesic, Opiorphin is 6 times stronger than the opiate morphine. Opiorphin is closely related to the rat sialorphin peptide, which is an inhibitor of pain perception and acts by potentiating endogenous micro- and ∂-opioid receptor-dependent enkephalinergic pathways. In rat studies, Opiorphin suppressed pain sensation for both chemical-induced inflammation and acute physical pain. In both cases, the administered dose of 1 mg/kg provided the same painkilling power as 3-6 mg/kg of morphine.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-253217 | 864084-88-8 | C29H48N12O8 | 1 mg |
- Org 24598 lithium salt
This is a selective, potent inhibitor of glial GlyT (GlyT1, glycine transporter type 1). In rats (P12-P16) and kynurenic acid, 6-cyano-7-nitroquinoxaline-2,3-dione (CNQX) and bicuculline, ORG 24598 at a concentration of 10 µM induced a mean inward current of -10/-50 pA at -60 mV and increased significantly the decay time constants of miniature (mIPSCs), spontaneous (sIPSCs) and electrically evoked glycinergic (eIPSCs) inhibitory postsynaptic currents. Replacing extracellular sodium with N-methyl-d-glucamine or superfusing the slice with micromolar concentrations of glycine also increased the decay time constant of glycinergic IPSCs. Glycine (1-5 µM and d-serine (10 µM) increased the amplitude of eEPSCs whereas l-serine had no effect. Org 24598 increased significantly the amplitude of NMDA receptor-mediated eEPSCs without affecting the amplitude of non-NMDA receptor-mediated eEPSCs. This brings conclusion that blocking glial glycine transporter by Org 24598 increased the level of glycine in spinal cord slices, which in turn prolonged the duration of glycinergic synaptic current and potentiated the NMDA-mediated synaptic response.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-253218 | 722456-08-8 | C19H19F3LiNO3 | 5 mg |
- p-Aminoclonidine hydrochloride
This product is an α2-adrenoceptor agonist.
| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-301508 | 73218-79-8 | C9H10Cl2N4•xHCl | 1 mg |
- p-Fluorohexahydro-sila-difenidol hydrochloride
High affinity M3 muscarinic acetylcholine receptor antagonist.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-257953 | 116679-83-5 | C20H32FNOSi ·HCl | 10 mg |
- p-MPPI monohydrochloride
A selective 5-HT1A serotonin receptor antagonist that crosses the blood-brain barrier.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-253226 | 220643-77-6 | C25H27IN4O2 ·HCl | 250 mg |
- p-MPPI trihydrochloride
| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-358823 | 155204-23-2 (free base) | C25H27IN4O2 | 10 mg |
- P1,P4-Di(adenosine-5') tetraphosphate ammonium salt
A derivative of Diadenosine polyphosphate, which is stored in secretory granules of thrombocytes, chromaffin, and neuronal cells. Has been shown to function as a pancreatic cell secondary messenger, phospholipase D stimulator, change intracellular calcium levels, nitric oxide release inductor, 5’-nucleotidase activator and adenosine kinase activity inhibitor in vitro. | Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-253229 | 102783-36-8 | C20H31N11O19P4 | 10 mg |
- P7C3
| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-362776 | 301353-96-8 | C21H18Br2N2O | 10 mg/50 mg |
- Pasiniazid
| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-250652 | 2066-89-9 | C13H14N4O4 | 10 g |
- PD 116,948
PD 116,948, a xanthine derivative, is a very potent and selective adenosine A1 receptor antagonist.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-200115 | 102146-07-6 | C16H24N4O2 | 20 mg/100 mg |
- (+/-)-PD 128,907 hydrochloride
Selective D3 dopamine receptor agonist.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-257969 | 112960-16-4 | C14H19NO3•HCl | 5 mg |
- Pheniramine maleate salt
A H1 histamine receptor antagonist.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-253258 | 132-20-7 | C16H20N2•C4H4O4 | 5 g |
- Phenyltoloxamine citrate salt
| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-228940 | 1176-08-5 | C17H21NO•C6H8O7 | 50 g |
- Picrotoxinin
GABAA receptor antagonist that binds to the GABA receptor-linked Cl- channel.
Active component of picrotoxin| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-253277 | 17617-45-7 | C15H16O6 | 250 mg |
- Pimethixene maleate salt
| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-228949 | 13187-06-9 | C19H19NS•C4H4O4 | 250 mg |
- Pipamperone dihydrochloride
Antipsychotic; D2 dopamine receptor antagonist; 5-HT2 serotonin receptor antagonist.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-253278 | 2448-68-2 | C21H30N3O2F•2HCl | 100 mg |
- Piperidine-4-sulfonic acid
GABAAreceptor agonist.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-253279 | 72450-62-5 | C5H11NO3S | 25 mg |
- Pirenperone
5-HT2 serotonin receptor antagonist.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-253280 | 75444-65-4 | C23H24FN3O2 | 25 mg |
- (±)-PPHT hydrochloride
Potent D2 dopamine receptor agonist. A series of new dopamine (DA) receptor agonists, of the 2-aminotetralin group, i.e. N-0434, N-0437 and N-0734 were investigated both in vivo and in vitro pharmacological test systems. In vivo, the reversal of the gamma-butyrolactone-induced an increase in rat central DOPA biosynthesis, the rate was taken as a measure of presynaptic activity. The homovanillic acid (HVA) decrease, after intraperitoneal and after oral administration of the drugs was also taken as a measure of presynaptic activity. Postsynaptic activity was measured in two behavioural models, i.e. stereotypy induction and reserpine reversal. The effects of (±)-PPHT (N-0434) these drugs on noradrenaline and dopamine turnover (alpha-MpT method) were studied in addition. The results indicate that all three compounds N-0434 ((±)-PPHT), N-0437 and N-0734 are potent and selective DA agonists that lack significant alpha 2 activity. | Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-253313 | 71787-90-1 | C21H28ClNO | 10 mg |
- Pramoxine hydrochloride
Skin or mucous membrane topical anesthetic.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-264141 | 637-58-1 | C17H28ClNO3 | 10 g |
- Pranoprofen
A non-steroidal antiinflammatory drug. It inhibits platelet aggregation. | Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-205814 | 52549-17-4 | C15H13NO3 | 100 mg/250 mg |
- Primaquine phosphate
Antimalarial drug with genotoxicity (Ames test) and cardiotoxicity (inhibitor of cardiac Na+ current).| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-205817 | 63-45-6 | C15H21N3O.2H3PO4 | 5 g/10 g |
- Propantheline bromide
Inhibits action of acetylcholine at post-ganglionic synapses; muscarinic acetylcholine receptor antagonist; antispasmodic; reduces gastric acid secretion.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-253320 | 50-34-0 | C23H30NO3Br | 5 g |
- Proparacaine hydrochloride
Topical ophthalmic anesthetic| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-264146 | 5875-06-9 | C16H27ClN2O3 | 1 g |
- Protriptyline hydrochloride
A norepinephrine uptake blocker.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-250799 | 1225-55-4 | C19H21N•HCl | 100 mg |
- Proxymetacaine Hydrochloride
A local anesthetic that is used to numb the surface of a body part. | Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-205820 | 5875-06-9 | C16H27ClN2O3 | 100 mg/250 mg |
- PSB 1115 potassium salt hydrate
A highly selective, water-soluble, human A2B adenosine receptor antagonist.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-253323 | 409344-71-4 (anhydrous) | C14H13KN4O5S•xH2O | 10 mg |
- Pyridoxal phosphate-6-azo(benzene-2,4-disulfonic acid) tetrasodium salt hydrate
A selective P2 purinoceptor antagonist which blocks responses at both pre- and post-junctional sites.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-253332 | 192575-19-2 (anhydrous) | C14H10N3Na4O12PS2•xH2O | 10 mg/50 mg |
- (±)-Quinpirole dihydrochloride
D2-like dopamine receptor agonist which has some activity at D3 sites.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-253338 | 73625-62-4 | C13H21N3•2HCl | 50 mg |
- (-)-Quinpirole hydrochloride
The putative D2 dopamine receptor agonist quinpirole is the most widely used D2 agonist in in vivo and in vitro studies. Active enantiomer of (±)-quinpirole. Quinpirole is a dopamine agonist with high affinity for the D2 and D3 dopamine receptor subtypes. Specific [3H]quinpirole binding in rat brain was saturable, and dependent on temperature, membrane concentration, sodium concentration and guanine nucleotides. Saturation analysis revealed high affinity binding characteristics (Kd = 2.3 +/- 0.3 nM) which were confirmed by association-dissociation kinetics. The regional distribution of [3H]quinpirole binding sites roughly paralleled the distribution of [3H]spiperone binding sites, with greatest densities present in the striatum, nucleus accumbens and olfactory tubercles. A variety of drugs, most notably monoamine oxidase inhibitors (MAOls), inhibit the binding of [3H]quinpirole, but not [3H]spiperone or [3H](-)N-n-Propylnorapomorphine, in rat striatal membranes by a mechanism that does not appear to involve the enzymatic activity of MAO. Clinically antidepressant MAOIs exhibited selectivity between sites labeled by [3H]quinpirole and [3H]spiperone as did a number of structurally related propargylamines and N-acylethylenediamine derivatives and other drugs such as debrisoquin and phenylbiguanide. The MAOIs clorgyline and Ro 41-1049 were the most potent. MAOIs interact with a novel binding site,may be associated with D2-like dopamine receptors, that is labeled by [3H]quinpirole or that modulates [3H]quinpirole binding.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-253339 | 85798-08-9 | C13H21N3•HCl | 10 mg/25 mg |
- (+/-)-Quinuclidinyl benzilate
Nonselective antagonist to muscarinic ACh receptors.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-264194 | 6581-06-2 | C21H23NO3 | 5 mg/10 mg |
- Quirestine
Potent short-acting ganglioblocker. Nicotinic acetylcholine receptor antagonist.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-253340 | 41663-80-3 | C12H24IN | 2 mg |
- R-(-)-Apomorphine hydrochloride hemihydrate
A nonselective dopamine agonist that causes nausea and emesis.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-253341 | 41372-20-7 | C17H17NO2 ·HCl ·1/2H2O | 100 mg/250 mg |
- R-(-)-Desmethyldeprenyl hydrochloride
Neuroprotectant and an anti-apoptotic.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-258056 | 115586-38-4 | C12H15N•HCl | 5 mg |
- R(-)-2,10,11-Trihydroxy-N-propyl-noraporphine hydrobromide hydrate
A potent, selective D2 dopamine receptor agonist.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-253350 | 79640-85-0 (anhydrous) | C19H21NO3•HBr•xH2O | 10 mg/25 mg |
- R(-)-2,10,11-Trihydroxyaporphine hydrobromide
Dopamine receptor agonist.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-253351 | 77630-01-4 | C17H17NO3•HBr | 50 mg |
- R(-)-Denopamine
| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-360703 | 71771-90-9 | C18H23NO4 | 5 mg |
- R(-)-Propylnorapomorphine hydrochloride
Very potent and selective D2 dopamine receptor agonist.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-253354 | 18426-20-5 | C19H21NO2•HCl | 10 mg/25 mg |
- R(+)-3-(3-Hydroxyphenyl)-N-propylpiperidine hydrochloride
A D2 dopamine receptor agonist. Also functions as 1 receptor antagonist with essentially no affinity for the phencylidine site on the NMDA receptor.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-253355 | 89874-80-6 | C14H21NO•HCl | 25 mg |
- R(+)-7-Hydroxy-DPAT hydrobromide
Active enantiomer of (±)-7-hydroxy-DPAT; selective D3 dopamine receptor agonist.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-253356 | 82730-72-1 | C16H26BrNO | 5 mg |
- R(+)-SKF-81297 hydrobromide
A selective D1 dopamine receptor agonist.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-253357 | 253446-15-0 | C16H16ClNO2•HBr | 5 mg |
- R(+)-UH-301 hydrochloride
A potent and selective 5-HT1A serotonin receptor agonist.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-253358 | 127126-18-5 | C16H25ClFNO | 1 mg |
- (R)-(+)-8-Hydroxy-DPAT hydrobromide
(R)-(+)-8-Hydroxy-DPAT is a full 5-HT1A serotonin receptor agonist; active enantiomer of (±)-8-hydroxy-DPAT.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-253404 | 78095-19-9 | C16H25NO•HBr | 5 mg/25 mg |
- (R)-(+)-SKF-38393 hydrochloride
Active enantiomer of (±)-SKF-38393; D1 dopamine receptor agonist.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-253412 | 81702-42-3 | C16H17NO2··HCl | 5 mg |
- (R)-SKF-82957 hydrobromide
A selective D1 dopamine receptor agonist.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-255520 | 288262-87-3 | C17H18ClNO2•HBr | 5 mg |
- Reboxetine mesylate hydrate
A selective noradrenaline uptake inhibitor.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-253426 | 98769-84-7 (anhydrous) | C20H29NO7S | 5 mg |
- RF9 trifluoroacetate salt
A neuropeptide FF receptor antagonist. | Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-253428 | 876310-60-0 (non-salt) | C26H38N6O3•xC2HF3O2 | 1 mg |
- Ro 27-3225 trifluoroacetate salt
This is a selective melanocortin MC4 receptor agonist. EC50 = 1 nM.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-311523 | n.n. | C39H52N12O6•xC2HF3O2 | 1 mg |
- Ro 4-1284
A reversible VMAT2 inhibitor.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-255523 | 303-75-3 | C21H33NO3 | 5 mg |
- Ro4368554
A 5-HT6 receptor antagonist. Acts selectively at 5-HT6 receptors where it binds with a greater than 100-fold selectivity over other monoamine receptor subtypes.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-253435 | 478082-99-4 | C19H21N3O2S | 5 mg |
- S-(-)-SKF-38393 hydrochloride
Less active enantiomer of (±)-SKF-38393; D1 dopamine receptor agonist.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-253440 | 81702-43-4 | C16H17NO2•HCl | 100 mg |
- S-(+)-Chlorpheniramine maleate salt
Active isomer; H1 histamine receptor antagonist.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-253441 | 2438-32-6 | C20H23ClN2O4 | 1 g |
- S-(+)-O-Desmethylraclopride hydrobromide
Precursor to radiolabeled S-(+)-raclopride. | Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-258091 | 113310-88-6 | C14H18Cl2N2O3•HBr | 5 mg |
- S-(4-Nitrobenzyl)-6-thioinosine (NBTI, NBMPR)
An inhibitor of equilibrative nucleoside trasport proteins. Blocks the uptake and transport of adenosine.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-200117 | 38048-32-7 | C17H17N5O6S | 50 mg |
- S(-)-Baclofen hydrochloride
The less active enantiomer of baclofen, which happens to be the same enantiomer as S(+)-baclofen free base.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-264246 | 63701-56-4 | C10H12ClNO2•HCl | 25 mg/100 mg |
- S(-)-Cyanopindolol hemifumarate salt
A 5-HT1A/1B serotonin receptor antagonist; β3-adrenoceptor antagonist.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-253460 | 874882-72-1 | C32H42N6O4··C4H4O4 | 1 mg |
- S(-)-Raclopride (+)-tartrate salt
A selective D2 dopamine receptor antagonist.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-253461 | 98185-20-7 | C15H20Cl2N2O3··C4H6O6 | 25 mg |
- S(-)-UH-301 hydrochloride
A potent, selective 5-HT1A serotonin receptor antagonist and D2/D3 dopamine receptor agonist.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-253462 | 127126-22-1 | C16H24FNO•HCl | 1 mg/5 mg |
- S(+)-Propylnorapomorphine hydrochloride
Limbic-selective dopamine antagonist.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-253463 | 79703-31-4 | C19H21NO2•HCl | 5 mg |
- (S)-(-)-3-(3-Hydroxyphenyl)-N-propylpiperidine hydrochloride
A dopamine autoreceptor agonist and a postsynaptic dopamine receptor antagonist.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-253477 | 88768-67-6 | C14H22ClNO | 25 mg/100 mg |
- (S)-(+)-Apomorphine hydrochloride hydrate
Dopamine receptor antagonist. Is inactive as an agonist.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-253505 | 41035-30-7 (anhydrous) | C17H17NO2•HCl•xH2O | 5 mg |
- (S)-Mephenytoin
A hydantoin used in the (S)-Mephenytoin 4’-hydroxylation assay for studying CYP2C19 polymorphism.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-200975 | 70989-04-7 | C12H14N2O2 | 5 mg/25 mg |
- (S)-Nafadotride tartrate
D3 Dopamine receptor antagonist.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-253523 | 173429-65-7 | C26H33O8N3 | 1 mg |
- SB 242084 hydrochloride
An antagonist of the 5-HT2C receptor (pKi= 9.0), with at least 100-fold more selectivity over other 5-HT, dopamine or adrenergic receptors; used extensively in animal research to evaluate, for example, 5-HT2C receptor agonists and neurotransmitter receptor interactions in mice.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-351848 | 1049747-87-6 | C21H19ClN4O2•2HCl | 1 mg/5 mg |
- SB 242084 dihydrochloride hydrate
Crosses the blood-brain barrier; selective 5-HT2c serotonin receptor antagonist.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-253538 | 181632-25-7 (non-salt) | C21H19ClN4O2•2HCl•xH2O | 5 mg |
- SB-215505
Selective 5-HT2B serotonin receptor antagonist; 100-fold higher affinity at 2B compared to 2C.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-253540 | 162100-15-4 | C19H16N3OCl | 5 mg |
- SB-224289 hydrochloride
Selective 5-HT1B serotonin receptor antagonist| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-253541 | 180084-26-8 | C32H32N4O3•HCl | 5 mg |
- SB-269970 hydrochloride
A selective 5-HT7 serotonin receptor antagonist.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-255605 | 261901-57-9 | C18H28N2O3S•HCl | 5 mg |
- (-)-Scopolamine hydrochloride
Competitive nonselective muscarinic acetylcholine antagonist. Scopolamine-induced amnesia in laboratory animals is a commonly-used model of memory deficit.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-253544 | 55-16-3 | C17H21NO4•HCl | 1 g |
- (-)-Scopolamine methyl bromide
A competitive muscarinic acetylcholine receptor antagonist.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-253545 | 155-41-9 | C18H24NO4•Br | 1 g |
- (-)Scopolamine methyl nitrate
Competitive antagonist to muscarinic receptors for use in the treatment of motion sickness.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-264301 | 6106-46-3 | C17H21NO4•CH3NO3 | 1 g |
- Serotonin creatinine sulfate complex
A neurotransmitter. | Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-215845 | 971-74-4 | C14H19N5O2•H2O4S•H2O | 250 mg/500 mg |
- SKF 86002
A bicyclic imidazole that specifically inhibits p38 MAP kinase, and is also described as a cytokine-suppressant and an anti-inflammatory compound.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-203265 | 72873-74-6 | C16H12FN3S | 5 mg |
- (+/-)-SKF-38393 hydrochloride
Agonist to D1 Dopamine receptors.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-264306 | 62717-42-4 | C16H17NO2•HCl | 100 mg/500 mg |
- SKF-86466 hydrochloride
Selective and potent α2 adrenoceptor antagonist.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-253566 | 86129-54-6 | C11H15Cl2N | 10 mg |
- SKF-89976A
GABA transporter type 1 inhibitor that crosses the blood brain barrier.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-253567 | 85375-15-1 | C22H25NO2•HCl | 10 mg |
- SKF-95282 dimaleate salt
Antagonist to H2 His receptor| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-255616 | 104076-39-3 | C22H27N3OS•2C4H4O4 | 10 mg |
- Sulfadimethoxine sodium salt
| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-229344 | 1037-50-9 | C12H13N4O4SNa | 10 g |
- Suloctidil
| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-236957 | 54767-75-8 | C20H35NOS | 5 g |
- T62
Allosteric enhancer of A1 adenosine receptor.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-253618 | 40312-34-3 | C15H14ClNOS | 5 mg |
- Temechine hydrobromide
A neuronal nicotinic acetylcholine receptor antagonist and a potent ganglioblocker.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-255629 | 30015-57-7 | C11H21N•HBr | 2 mg |
- Tempoxime hydrochloride
A neuronal nicotinic AChR antagonist and potent ganglioblocker.
| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-301866 | 63467-53-8 | C9H18N2O•HCl | 2 mg |
- tert-Butyl bicyclo[2.2.2]phosphorothionate
GABAA receptor antagonist, chloride channel blocker and an extremely potent convulsant.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-253633 | 70636-86-1 | C8H15O3PS | 2 mg |
- Tiapride hydrochloride
D2 and D3 dopamine receptor antagonist; antipsychotic.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-253697 | 51012-32-9 | C15H24N2O4S ·HCl | 5 g |
- TMPH hydrochloride
A potent inhibitor of neuronal nicotinic receptors. Evaluation of nicotinic acetylcholine receptor subunits expressed in Xenopus laevis oocytes indicated that TMPH can produce a potent and long-lasting inhibition of neuronal nAChR formed by the pairwise combination of the most abundant neuronal alpha (i.e., alpha3 and alpha4) and beta subunits (beta2 and beta4), with relatively little effect, because of rapid reversibility of inhibition, on muscle-type (alpha1beta1gammadelta) or alpha7 receptors. However, the inhibition of neuronal beta subunit-containing receptors was also decreased if any of the nonessential subunits alpha5, alpha6, or beta3 were coexpressed. This decrease in inhibition is shown to be associated with a single amino acid present in the second transmembrane domain of these subunits. TMPH ability to relate the diverse central nervous system effects to specific nAChR subtypes makes it a helpful tool for studying the functional roles of nAChR. | Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-253705 | 849461-91-2 | C16H32ClNO2 | 5 mg |
- Tobramycin Sulfate
Used in the treatment of respiratory infection and cystic fibrosis.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-205865 | 79645-27-5 | C18H37N5O9 ··· ·xH2SO4 | 100 mg/500 mg |
- Todralazine hydrochloride
Antihypertensive| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-253707 | 3778-76-5 | C11H12N4O2•HCl | 1 g |
- Toloxatone
A reversible monoamine oxidase A inhibitor (MAOI) and antidepressant. Belongs to the aryloxazolidinones, a relatively new class of reversible monoamine oxidase A inhibitors (MAOI). Studies show that derivatives such as 3-aryloxazolidin-2-one (oxazolidinones), which are regularly used to treat gram positive infections, represent a new class of reversible as well as irreversible inhibitors for MAO-A and MAO-B enzymes that are able to inhibit protein synthesis and also used for neurodegenerative-type pathologies.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-255665 | 29218-27-7 | C11H13NO3 | 10 mg |
- Trifluperidol hydrochloride
| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-253757 | 2062-77-3 | C22H23F4NO2•HCl | 25 mg |
- Tropine 2-(phenylthio)butanoate oxalate salt
Strong analgesic. Results in an increased release of acetylcholine at central muscarinic synapses.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-253806 | 155059-55-5 | C20H27NO6S | 50 mg |
- U-99194 maleate
A putative D3 antagonist with a 30-fold preference for the dopamine D3 compared to D2 receptor.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-253817 | 234757-41-6 | C17H27NO2•C4H4O4 | 25 mg |
- Valacyclovir hydrochloride hydrate
A potent inhibitor of viral DNA polymerase which serves as a prodrug of acyclovir that is useful in viral, AIDS, and immune system regulation research. | Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-216047 | 124832-27-5 (anhydrous) | C13H20N6O4•HCl•xH2O | 50 mg/250 mg |
- VU0029767
VU0029767 is a selective, novel M1 positive allosteric modulator. M1 is a member of the muscarinic acetylcholine family of GPCRs (mAChRs) and is a therapeutic target for cognitive deficits in schizophrenia and Alzheimer's disease. VU0029767 increases both potency and efficacy of acetylcholine (ACh) at M1. VU0029767 also potentiates a mutant M1 receptor, as well as the effects of allosteric agonist TBPB. VU0029767 weakly increases ACh potency at M1 in phospholipase C and phospholipase D assays. This compound was discovered in conjuction with VU0090157 (different chemotype), another M1 modulator, which differs in its activities at the mutant form of M1, potentiation of TBPB, and phospholipase assays. The two modulators differentially regulate G protein signaling following M1 activation. Thus, VU0029767 and VU0090157 are valuable compounds when used together to tease out ligand-directed trafficking.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-253833 | 326001-01-8 | C21H21N3O3 | 25 mg |
- VU255035 hydrate
VU0255035 is the first highly selective antagonist at the orthosteric site of the M1 receptor (75-fold selective for M1 relative to other muscarininc subtypes and devoid of activity at other GPCRs, ion channels, transporters and kinases). There are no highly selective M1 muscarinic receptor antagonists. The existing non-selective drugs do not permit direct evaluation of the role of M1 receptors in CNS fucntions and do not premit therapeutic targeting of M1 receptors in various disease states in which M1 receptors are implicated (epilepsy, Parkinson's disease, attention and cognitive disorders, dystonia, etc).| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-258334 | 1135243-19-4 (anhydrous) | C18H20N6O3S2•xH2O | 5 mg |
- WAY-100635 maleate salt
Selective 5-HT1A Ser receptor antagonist.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-264493 | 634908-75-1 | C25H34N4O2•C4H4O4 | 5 mg/50 mg |
- Xanthine amine congener
Xanthine amine congener is a potent, nonselective adenosine receptor antagonist (A1 and A2B > A2A).| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-255717 | 96865-92-8 | C21H28N6O4 | 25 mg |
- Xli 093 hydrate
| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-264494 | 646066-59-3 (anhydrous) | C33H26N6O6•xH2O | 5 mg |
- Xylazine
α2-adrenoceptor agonist, sedative, muscle relaxant.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-253838 | 7361-61-7 | C12H16N2S | 1 g |
- Xylometazoline hydrochloride
α-adrenoceptor agonist; imidazoline binding site ligand.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-255719 | 1218-35-5 | C16H24N2 ·HCl | 5 g |
|