Drug Analogues

• 1-(1-Naphthyl)-2-chloroethane
  An analogue and derivative of Tamoxifen.

  Katalog #	CAS Nummer	Summenformel	Menge
  sc-216108	41332-02-9	C12H11Cl	5 mg

• 1-(Benzylideneamino)parabanic Acid
  An analog of Nitrofurantoin.

  Katalog #	CAS Nummer	Summenformel	Menge
  sc-208553	42839-64-5	C10H7N3O3	2 g

• (1R,4S)-N-Desmethyl Sertraline Hydrochloride
  Used for treatment of CNS disorders. A metabolite of Sertraline.

  Katalog #	CAS Nummer	Summenformel	Menge
  sc-206300	675126-08-6	C16H16Cl3N	1 mg

• (1S,4R)-N-Desmethyl Sertraline Hydrochloride
  Used for treatment of CNS disorders. A metabolite of Sertraline.

  Katalog #	CAS Nummer	Summenformel	Menge
  sc-206308	675126-07-5	C16H16Cl3N	1 mg

• (1S,4S)-N-Desmethyl Sertraline Hydrochloride
  A metabolite of Sertraline. A significantly less active compared to the methylated compound, Sertraline.

  Katalog #	CAS Nummer	Summenformel	Menge
  sc-206309	675126-10-0	C16H16Cl3N	1 mg

• 2-(4'-Acetoxy-2-fluoro-biphenyl-4-yl)-propionic Acid Methyl Ester

  Katalog #	CAS Nummer	Summenformel	Menge
  sc-206325	215175-84-1	C18H17FO4	10 mg

• 2-Amino-4-ethylpyridine
  An analogue of pirlimycin which is an antibiotic.

  Katalog #	CAS Nummer	Summenformel	Menge
  sc-209039	33252-32-3	C7H10N2	1 g

• 2'-O-Benzyloxy-2-O-desmethylcarvedilol
  Carvedilol analog with multiple-action, neurohormonal antagonism used in the treatment of hypertension.

  Katalog #	CAS Nummer	Summenformel	Menge
  sc-214075	72955-92-1	C30H30N2O4	5 mg

• 2R,S-Hydroxy-4[[(2R)-2-hydroxy-2-(3-hydroxyphenyl)ethyl]methylamino]-4-oxo-butanoic Acid
  A phenylephrine derivative.

  Katalog #	CAS Nummer	Summenformel	Menge
  sc-223486	1217525-08-0	C13H17NO6	5 mg

• 3-Cyano-7-methoxycoumarin
  A fluorescent CYP1A1 &1A2 substrate

  Katalog #	CAS Nummer	Summenformel	Menge
  sc-252000	13229-92-0	C11H7NO3	5 mg

• 3,5-Diiodothyroacetic Acid
  The acetic acid analog of Thyroxine and a potent

  Katalog #	CAS Nummer	Summenformel	Menge
  sc-209717	1155-40-4	C14H10I2O4	1 mg

• 4-(3-Nitrophenyl)-2-dimethoxymethyl-1,4-dihydropyridine-3,5-dicarboxylic Acid 5-Isopropyl Ester 3-Methyl Ester

  Katalog #	CAS Nummer	Summenformel	Menge
  sc-223595	75530-94-8	C21H26N2O8	50 mg

• 4-(3-Nitrophenyl)-2-formyl-6-methyl-1,4-dihydropyridine-3,5-dicarboxylic Acid 5-Isopropyl Ester 3-Methyl Ester
  A nilvadipene analogue.

  Katalog #	CAS Nummer	Summenformel	Menge
  sc-206756	75530-60-8	C19H20N2O7	50 mg

• 4-Acetoxy-N-isopropyl-N-methyltryptamine

  Katalog #	CAS Nummer	Summenformel	Menge
  sc-206799	1024612-25-6	C16H22N2O2	5 mg

• 4-Epianhydrochlortetracycline Hydrochloride
  A modified Tetracycline analog.

  Katalog #	CAS Nummer	Summenformel	Menge
  sc-210035	158018-53-2	C22H21ClN2O7.HCl	2.5 mg

• 4-Hydroxy-N-isopropyl-N-methyltryptamine
  A related homologue of Psilocin.

  Katalog #	CAS Nummer	Summenformel	Menge
  sc-210083	77872-43-6	C14H20N2O	5 mg

• (+/-)-4ε-Methoxymephenytoin

  Katalog #	CAS Nummer	Summenformel	Menge
  sc-299183	n.n.	C13H16N2O3	5 mg

• 5'-Benzyloxy Carvedilol
  An analogue of Carvedilol which is a multiple-action, neurohormonal antagonist that is used in treating hypertension.

  Katalog #	CAS Nummer	Summenformel	Menge
  sc-210406	887353-00-6	C31H32N2O5	5 mg

• 5[(R)-(2-Aminopropyl)]-2-methoxybenzenesulfonamide Hydrochloride
  A precursor in the synthesis of Tamsulosin and other alpha-andregenic antagonists.

  Katalog #	CAS Nummer	Summenformel	Menge
  sc-207075	112101-75-4	C10H17ClN2O3S	1 g

• 6-Cyano-3,4-dihydro-2,2-dimethyl-trans-4-(1-pyrrolidinyl)-2H-benzo-[b]-pyrano-3-ol
  Cromakalin analog, generating vasodilation via activation of potassium channels.

  Katalog #	CAS Nummer	Summenformel	Menge
  sc-214370	75611-78-8	C16H20N2O2	25 mg

• 6α-Naloxol Hydrochloride
  A metabolite of Naloxone. Naltrexone analogs and Naloxone analogs are neutral µ- opioid antagonists and are used in the treatment of drug abuse and pain.

  Katalog #	CAS Nummer	Summenformel	Menge
  sc-210579	34520-00-8	C19H24ClNO4	1 mg

• 7-Bromo Epinastine
  Epinastine analogue.

  Katalog #	CAS Nummer	Summenformel	Menge
  sc-217423	n.n.	C16H14BrN3	10 mg

• 7-Chloro Epinastine Hydrochloride
  An Epinastine analog.

  Katalog #	CAS Nummer	Summenformel	Menge
  sc-214397	80012-45-9	C16H15Cl2N3	5 mg

• 7-Hydroxycoumarin glucuronide sodium salt
  Phase II (UDP-GT) metabolite of 7-hydroxycoumarin.

  Katalog #	CAS Nummer	Summenformel	Menge
  sc-252309	66695-14-5 (non-salt)	C15H13NaO9	5 mg

• 9-Didemethyl Minocycline
  A Tetracycline analog used in antibiotic pharmaceutical compositions.

  Katalog #	CAS Nummer	Summenformel	Menge
  sc-207219	5874-95-3	C21H23N3O7	1 mg

• 11-Azaartemisinin
  A nontoxic analog of Artemisinin

  Katalog #	CAS Nummer	Summenformel	Menge
  sc-208842	162791-23-3	C15H23NO4	1 mg

• 14-Bromo Daunorubicin Formate Salt
  Adriamycin analogue. Used as anticancer agent.

  Katalog #	CAS Nummer	Summenformel	Menge
  sc-208862	n.n.	C27H28BrNO10	1 mg

• 14-Chloro Daunorubicin
  An Adriamycin analogue that is used as an anticancer agent.

  Katalog #	CAS Nummer	Summenformel	Menge
  sc-206279	121250-06-4	C27H28ClNO10	1 mg

• 15-Hydroxy Lubiprostone
  A halogenated, bioactive lipid

  Katalog #	CAS Nummer	Summenformel	Menge
  sc-213612	475992-30-4	C20H34F2O5	1 mg/500 µg

• 15(R)-Pinane Thromboxane A2
  A stable analog of thromboxane A2 (TXA2); a thromboxane (TP) receptor antagonist and an inhibitor of thromboxane synthase.

  Katalog #	CAS Nummer	Summenformel	Menge
  sc-220628	n.n.	C24H40O3	500 µg/1 mg

• 17-Ethoxycarbonyl-3-methoxymorphinan
  A derivative of Dextrorphan.

  Katalog #	CAS Nummer	Summenformel	Menge
  sc-208872	524713-55-1	C20H27NO3	25 mg

• 17-Keto Vecuronium Bromide
  An analog of Vecuronium bromide

  Katalog #	CAS Nummer	Summenformel	Menge
  sc-208873	50587-93-4	C32H53BrN2O3	1 mg

• Amino Tadalafil
  A drug analog of Tadalafil.

  Katalog #	CAS Nummer	Summenformel	Menge
  sc-210797	385769-84-6	C21H18N4O4	2.5 mg

• Anhydrotetracycline Hydrochloride
  A Tetracycline derivative exhibiting no antibiotic activity, but is a useful effector of tetracycline-dependent gene expression in bacterial expression systems.

  Katalog #	CAS Nummer	Summenformel	Menge
  sc-210820	13803-65-1	C22H23ClN2O7	2.5 mg

• Anthrax Lethal Factor Protease Inhibitor III
  A cell-permeable, rhodanine-acetic acid analog that chelates the active site Zn2+ and acts as a potent inhibitor of anthrax lethal factor (LF) metalloproteinase.

  Katalog #	CAS Nummer	Summenformel	Menge
  sc-221254	n.n.	C17H9ClF3NO4S2	5 mg

• Aspirin-L-argininie

  Katalog #	CAS Nummer	Summenformel	Menge
  sc-337539	37466-21-0	n.n.	500 mg

• Atorvastatin Impurity F (sodium salt)

  Katalog #	CAS Nummer	Summenformel	Menge
  sc-362044	n.n.	C40H47FN3NaO8	10 mg

• Atorvastatin N-(3,5-Dihydroxy-7-heptanoic Acid)amide (Ca+ Salt)

  Katalog #	CAS Nummer	Summenformel	Menge
  sc-362045	1105067-87-5	C40H48FN3O8•0.5Ca	5 mg

• BD 1008 Dihydrobromide
  An α receptor antagonist which attenuates the biochemical effects of cocaine. This compounds ability to prevent neuropathic pain following chemotherapy was also studied.

  Katalog #	CAS Nummer	Summenformel	Menge
  sc-207316	138356-09-9	C15H22Cl2N2 ·2HBr	10 mg

• Benzo[a]pyrene

  Katalog #	CAS Nummer	Summenformel	Menge
  sc-257130	50-32-8	C20H12	1 g

• Benzydamine N-oxide hydrogen maleate
  CYP2C9 substrate.

  Katalog #	CAS Nummer	Summenformel	Menge
  sc-252419	72962-60-8	C19H23N3O2··C4H4O4	5 mg

• BH3I-1'
  A cell-permeable fluorescent thiozolidineacetic acid analog which acts as a BH3 mimetic. Binds to the hydrophobic cleft on the surface of Bcl-x and specifically prevents BH3 domain-mediated protein-protein interaction between pro-apoptotic and anti-apoptotic members of the Bcl-2 family. Induces apoptosis independent of Bcl-x pore formation.

  Katalog #	CAS Nummer	Summenformel	Menge
  sc-221353	n.n.	C15H15NO3S2	5 mg

• β-Hydroxy Tamoxifen
  A hydroxylated analogue of tamoxifen with anti-estrogenic properties.

  Katalog #	CAS Nummer	Summenformel	Menge
  sc-280801	97151-03-6	C26H29NO2	5 mg

• β-Secretase Inhibitor IV
  A cell-permeable isophthalamide compound containing a hydroxyethylamine motif which binds to BACE-1 active site and potently blocks its proteolytic activity. Displays greater selectivity over other aspartyl proteases.

  Katalog #	CAS Nummer	Summenformel	Menge
  sc-222304	797035-11-1	C31H38N4O5S	1 mg

• Carboxyethyl- -aminobutyric acid
  Cell growth promoter

  Katalog #	CAS Nummer	Summenformel	Menge
  sc-252548	4386-03-2	C7H13NO4	15 mg

• cis-α-Hydroxy Tamoxifen
  A hydroxylated analogue of tamoxifen; has anti-estrogenic properties.

  Katalog #	CAS Nummer	Summenformel	Menge
  sc-211112	97170-41-7	C26H29NO2	5 mg

• cis-β-Hydroxy Tamoxifen
  A hydroxylated analogue of tamoxifen containing anti-estrogenic properties.

  Katalog #	CAS Nummer	Summenformel	Menge
  sc-217908	97151-04-7	C26H29NO2	5 mg

• Clencyclohexerol
  An analog of Clenbuterol which is a β-agonist which can be used as a growth promoter in farm animals.

  Katalog #	CAS Nummer	Summenformel	Menge
  sc-211114	157877-79-7	C14H20Cl2N2O2	10 mg

• CRAC Channel Inhibitor, BTP2
  A cell-permeable analog of 3,5-bis(trifluoromethyl)pyrazole (BTP) which specifically inhibits CRAC-mediated calcium influx in T-cells with an IC₅₀about 10 nM and displays ~31-fold greater selectivity over VOC. This blocks the calcium-induced activation and translocation of nuclear factor of activated T-cells (NFAT). It does not affect the activation of NF-κB and AP-1. It potently inhibits cytokine production (IC₅₀= 1.7 µM for IL-2) and PBMC proliferation (IC₅₀ = 190 nM).

  Katalog #	CAS Nummer	Summenformel	Menge
  sc-221441	223499-30-7	C15H9F6N5OS	5 mg

• Cytochrome P450 1B1 Inhibitor, TMS
  A cell-permeable trans-stilbene analog that acts as a potent, selective, and competitive inhibitor of cytochrome P450 1B1. Reversibly binds to the heme region of P450 1B1 and blocks the activity of P450 1A1 and 1A2 at much higher concentrations. Shown to effectively block the metabolic hydroxylation of 17-β-estradiol by cytochrome P450 1B1 in bicistronic membranes.

  Katalog #	CAS Nummer	Summenformel	Menge
  sc-221453	n.n.	C18H20O4	1 mg

• D-threo-1-(4-Aminophenyl)-2-dichloroacetylamino-1,3-propanediol Hydrochloride
  An analog of Chloramphenicol with an aniline group in place of the aryl nitro group.

  Katalog #	CAS Nummer	Summenformel	Menge
  sc-207482	57704-36-6	C11H15Cl3N2O3	100 mg

• D-threo-1-(4-Chlorosulfonylphenyl)-2-dichloroacetylamino-1,3-propanediol
  A Chloramphenicol analogue.

  Katalog #	CAS Nummer	Summenformel	Menge
  sc-218037	n.n.	C11H12Cl3NO5S	25 mg

• D-threo-1-(4-Sulfonylphenyl)-2-dichloroacetylamino-1,3-propanediol Sodium Salt
  A Chloramphenicol analogue.

  Katalog #	CAS Nummer	Summenformel	Menge
  sc-218038	903508-30-5	C11H12Cl2NNaO6S	50 mg

• Deoxy Artemisinin
  An analog of Artemisinin, an antimalarial agent.

  Katalog #	CAS Nummer	Summenformel	Menge
  sc-207521	72826-63-2	C15H22O4	10 mg

• Desmethoxy Gatifloxacin Trifluoroacetate
  A Gatifloxacin derivative and a new anti-mycobacterial.

  Katalog #	CAS Nummer	Summenformel	Menge
  sc-211261	93107-32-5	C20H21F4N3O5	10 mg

• Desmethyl-4'-chlorodiazepam
  Precursor to radiolabeled 4'-chlorodiazepam.

  Katalog #	CAS Nummer	Summenformel	Menge
  sc-300422	n.n.	C15H10Cl2N2O	5 mg

• (E,Z)-1-Bromo-2-[4-[2-(dimethylamino)ethoxy]phenyl]-1,2-diphenylethene
  An analogue of tamoxifen with anti-estrogenic properties.

  Katalog #	CAS Nummer	Summenformel	Menge
  sc-211396	19076-79-0	C24H24BrNO	25 mg

• (E)-1-(4-Hydroxyphenyl)-1-[4-(trimethylacetoxy)phenyl]-2-phenylbut-1-ene
  A analogue of tamoxifen with anti-estrogenic properties.

  Katalog #	CAS Nummer	Summenformel	Menge
  sc-218285	177748-17-3	C27H28O3	10 mg

• (E)-1-[4-[2-(N,N-Dimethylamino)ethoxy]phenyl]-1-[4-(trimethylacetoxy)phenyl]-2-phenylbut-1-ene
  A analogue of tamoxifen with anti-estrogenic properties.

  Katalog #	CAS Nummer	Summenformel	Menge
  sc-223956	177748-19-5	C31H37NO3	10 mg

• (E/Z)-4,4'-Dihydroxy Tamoxifen
  A Tamoxifen analog. A triphenylalkene derivative.

  Katalog #	CAS Nummer	Summenformel	Menge
  sc-218291	n.n.	C26H29NO3	10 mg

• (E/Z)-4,4'-Dihydroxy-N-desmethyl Tamoxifen
  A Tamoxifen analog.

  Katalog #	CAS Nummer	Summenformel	Menge
  sc-218292	n.n.	C25H27NO3	10 mg

• Fluoxetine-d5 solution

  Katalog #	CAS Nummer	Summenformel	Menge
  sc-300722	n.n.	C17D5H13F3NO	1 ml

• Gendenafil
  A Sildenafil analog found in dietary supplements.

  Katalog #	CAS Nummer	Summenformel	Menge
  sc-211558	147676-66-2	C19H22N4O3	5 mg

• Homo Sildenafil
  An analog of Sildenafil.

  Katalog #	CAS Nummer	Summenformel	Menge
  sc-211595	642928-07-2	C23H32N6O4S	2.5 mg

• Hydroxy Acetildenafil
  A Sildenafil analog found in herbal dietary supplements which is known to enhance male sexual function.

  Katalog #	CAS Nummer	Summenformel	Menge
  sc-211602	147676-56-0	C25H34N6O4	10 mg

• Hydroxyhomo Sildenafil
  An analog of Sildenafil and a potential PDE5 inhibitor.

  Katalog #	CAS Nummer	Summenformel	Menge
  sc-211615	139755-85-4	C23H32N6O5S	5 mg

• Hydroxythio Acetildenafil
  A Sildenafil (S435000) analog, is said to enhance male sexual function

  Katalog #	CAS Nummer	Summenformel	Menge
  sc-280805	n.n.	C25H34N6O3S	5 mg

• Hydroxythiohomo Sildenafil
  A thio analog of Sildenafil with reported PDE5 inhibiting properties.

  Katalog #	CAS Nummer	Summenformel	Menge
  sc-207746	479073-82-0	C23H32N6O4S2	1 mg

• Inhoffen Lythgoe Diol Monotosylate
  A vitamin D analog

  Katalog #	CAS Nummer	Summenformel	Menge
  sc-211645	66774-80-9	C20H30O4S	250 mg

• Isofolic Acid
  The 7-Isomer of Folic acid which is used as a potential PET radiopharmaceutical.

  Katalog #	CAS Nummer	Summenformel	Menge
  sc-211669	47707-78-8	C19H19N7O6	10 mg

• Lamivudine
  A potent nucleoside analog reverse transcriptase inhibitor (nRTI). An analog of cytidine that can inhibit both types (1 and 2) of HIV reverse transcriptase as well as the reverse transcriptase of hepatitis B. Needs to be phosphorylated to its triphosphate form before it is active.

  Katalog #	CAS Nummer	Summenformel	Menge
  sc-221830	134678-17-4	C8H11N3O3S	10 mg/50 mg

• LXRα/β Agonist
  A cell-permeable maleimide analog which acts as a potent and specific liver X receptor (LXR) dual agonist.

  Katalog #	CAS Nummer	Summenformel	Menge
  sc-221864	n.n.	C24H20N2O3	10 mg

• Mafosfamide Sodium Salt
  A Cyclophosphamide analog. Acts as an antitumor agent

  Katalog #	CAS Nummer	Summenformel	Menge
  sc-211761	84211-05-2	C9H18Cl2N2NaO5PS2	5 mg

• Methyl-4,4-dimethoxy-2-(3-nitrobenzylidene)-acetoacetate
  A precursor for the synthesis of a complex pyridine.

  Katalog #	CAS Nummer	Summenformel	Menge
  sc-218830	67448-15-1	C14H15NO7	100 mg

• Monensin Methyl Ester
  A neutral analog of monensin. Used in the preparation of ion-selective membranes for ion-selective electrodes.

  Katalog #	CAS Nummer	Summenformel	Menge
  sc-221957	28636-21-7	C37H64O11	100 mg

• Montelukast Gem-dimethylmethylene Analogue
  An analog of Montelukast that is used for preparation of MK-0476

  Katalog #	CAS Nummer	Summenformel	Menge
  sc-211924	162489-70-5	C35H38ClNO3S	5 mg

• N-(2-Hydroxyethyl)-11-azaartemisinin
  An 11-Azaartemisinin derivative. Exhibits activity against multidrug-resistant malaria upon oral consumption.

  Katalog #	CAS Nummer	Summenformel	Menge
  sc-211955	255731-00-1	C17H27NO5	1 mg

• N-Acetylneuraminic Acid Dimer, Disodium Salt, E. coli
  Prepared by the hydrolysis of colominic acid and then highly purified by ion exchange chromatography. Suitable for use as a standard marker or as a starting material to prepare complex carbohydrates.

  Katalog #	CAS Nummer	Summenformel	Menge
  sc-221985	n.n.	C22H34N2O17•2Na	10 mg

• N-Acetylneuraminic Acid, 2,3-Dehydro-2-deoxy-, Sodium Salt

  Katalog #	CAS Nummer	Summenformel	Menge
  sc-221987	24967-27-9	C11H16NNaO8	10 mg

• N-Amino-11-azaartemisinin
  11-Azaartemisinin derivative which displays a high order of activity against multidrug-resistant malaria by oral route.

  Katalog #	CAS Nummer	Summenformel	Menge
  sc-212117	1086409-78-0	C15H24N2O4	1 mg

• N-Deformyl-N-benzyloxycarbonyl Orlistat
  Orlistat analogue.

  Katalog #	CAS Nummer	Summenformel	Menge
  sc-212174	108051-94-1	C36H59NO6	1 mg

• N-Deformyl-N-pivaloyl Orlistat
  An Orlistat analogue.

  Katalog #	CAS Nummer	Summenformel	Menge
  sc-219100	n.n.	C33H61NO5	1 mg

• N-Desmethyl N-Ethoxycarbonyl Dextrorphan
  A dextrorphan derivative.

  Katalog #	CAS Nummer	Summenformel	Menge
  sc-212190	1079043-47-2	C19H25NO3	2.5 mg

• N-Desmethyl Sildenafil
  A metabolite of Sildenafil and a potential selective type 5 cGMP phosphodiesterase inhibitor.

  Katalog #	CAS Nummer	Summenformel	Menge
  sc-208029	139755-82-1	C21H28N6O4S	5 mg

• N-Hydroxy-11-azaartemisinin
  11-Azaartemisinin derivative which displayed a high order of activity against multidrug-resistant malaria by oral route.

  Katalog #	CAS Nummer	Summenformel	Menge
  sc-212218	1086409-82-6	C15H23NO5	1 mg

• N-Methyl-N-(2-hydroxyethyl)tamoxifen
  An analogue and derivative of Tamoxifen.

  Katalog #	CAS Nummer	Summenformel	Menge
  sc-212235	77214-91-6	C27H31NO2	5 mg

• NAADP Receptor Modulator
  A cell-permeable nicotinic acid analog that acts as a selective antagonist of NAADP-induced Ca²⁺ release, while at higher concentrations, also exhibits weak agonistic property towards NAADPR (nicotinic acid adenine dinucleotide phosphate receptor).

  Katalog #	CAS Nummer	Summenformel	Menge
  sc-222036	n.n.	C8H9IN2O3	25 mg

• NF023
  A suramin analog that acts as a selective and direct G-protein antagonist for α-subunits of the Go/Gi group (EC₅₀ ~ 300 nM). Suppresses GTPγS binding to recombinant G-protein α-subunits. Acts by inhibiting the formation of the agonist-specific ternary complex (agonist/receptor/G-protein). NF023 does not interfere with the interaction between α-subunits and βγ-dimer but competes with the effector binding site. Also a P2X receptor antagonist (IC₅₀ = 240 nM for P2X1; 8.5 µM for P2X3 receptor in rat muscle). Causes a concentration dependent inhibition of excitatory junction potentials (IC₅₀ = 4.8 pM).

  Katalog #	CAS Nummer	Summenformel	Menge
  sc-222065	n.n.	C35H20N4O21S6•6Na	10 mg

• Norneo Sildenafil
  An analog of Sildenafil and a potential PDE5 inhibitor.

  Katalog #	CAS Nummer	Summenformel	Menge
  sc-212414	371959-09-0	C22H29N5O4S	5 mg

• Paclitaxel C
  A Paclitaxel related compound C. Paclitaxel analogs have been tested for tubulin assembly and cytotoxicity, and have shown to retain potency similar to Paclitaxel.

  Katalog #	CAS Nummer	Summenformel	Menge
  sc-212517	153415-45-3	C46H57NO14	1 mg

• PDM 11
  Structurally very similar to several resveratrol analogs which act as a potent and selective AhR antagonists and agonists.2 One of these compounds, which contains fluorine in place of the 4'-chlorine of PDM11, acts as a AhR antagonist with a Ki of approximately 3 nM.2 This fluorine-containing compound is inactive as a ligand for the estrogen receptor even at 100 µM. As AhR knockout mice are insensitive to the carcinogenic effects of classical AhR ligands, antagonists of AhR could potentially serve as therapeutic agents for the treatment for dioxin and other aryl hydrocarbon poisonings.

  Katalog #	CAS Nummer	Summenformel	Menge
  sc-222145	n.n.	C16H15ClO2	10 mg/25 mg

• Pepstatin A Methyl Ester
  A cell-permeable methyl ester derivative of Pepstatin A that acts as a potent, non-competitive, transition-state analog inhibitor of γ-secretase.

  Katalog #	CAS Nummer	Summenformel	Menge
  sc-222147	n.n.	C35H65N5O9	1 mg

• Phenyl-d5-7-hydroxywarfarin
  7-Hydroxywarfarin internal standard. Labeled metabolite of warfarin.

  Katalog #	CAS Nummer	Summenformel	Menge
  sc-255417	94820-65-2	C19H11D5O5	5 mg

• PPACK, Dihydrochloride, Biotinylated
  Biotin-X-analog of PPACK, Dihydrochloride. Specific probe for active serine proteases. Potent inhibitor of thrombin and tissue plasminogen activator (tPA). Useful for Western blot analyses of Factor VIIa, Factor XIa, thrombin, and tPA.

  Katalog #	CAS Nummer	Summenformel	Menge
  sc-222186	n.n.	C43H70N10O7SCl•2HCl	1 mg

• Pristane
  A hydrocarbon oil adjuvant widely used to induce tumorgenesis in mice and arthritis and lupus nephritis in rats.

  Katalog #	CAS Nummer	Summenformel	Menge
  sc-281684	1921-70-6	C19H40	100 ml/250 ml

• Prochlorperazine, dimaleate
  Antipsychotic agent; used in the treatment of spastic gastrointestinal disorders.

  Katalog #	CAS Nummer	Summenformel	Menge
  sc-296136	84-02-6	C20H24N3SCl•2C4H4O4	1 g/5 g

• Progesterone 11α-glucuronide
  Phase II metabolite of progesterone

  Katalog #	CAS Nummer	Summenformel	Menge
  sc-301611	n.n.	C27H38O9	5 mg

• Proteasome Inhibitor IX, AM114
  A cell-permeable boronate chalcone compound with ~ 30-fold higher potency than MG-132 in inhibiting 20S proteasome chymotrypsin-like activity. Blockage of proteasome degradation of cellular ubiquitinated p53 by AM114 has been attributed to its preferential apoptotic effect against p53-expressing cancer cells.

  Katalog #	CAS Nummer	Summenformel	Menge
  sc-222199	n.n.	C20H21B2NO5	10 mg

• Proteasome Inhibitor VII, Antiprotealide
  A cell-permeable, Omuralide-Salinosporamide hybrid that irreversibly inactivates the β5-subunit of the human 20S proteasome. Shown to be ~2.5-fold more potent than Omuralide and is expected to exhibit comparable whole cell potency to Salinosporamide A.

  Katalog #	CAS Nummer	Summenformel	Menge
  sc-222200	n.n.	C12H18ClNO4	50 µg

• Proteasome Inhibitor VIII, β-Lactam 3
  A β-lactam analog of Proteasome Inhibitor VII, Antiprotealide which acts as a selective and irreversible inhibitor of the 20S proteasome. While the rate of proteasome inhibition is slower than Omuralide, β-lactam 3 displays prolonged aqueous stability and therefore may be better suited for biological evaluation.

  Katalog #	CAS Nummer	Summenformel	Menge
  sc-222201	n.n.	C11H17ClN2O3	100 µg

• Pseudo Vardenafil
  A Vardenafil

  Katalog #	CAS Nummer	Summenformel	Menge
  sc-212602	224788-34-5	C22H29N5O4S	5 mg

• Pyrazole N-Demethyl Sildenafil
  A pyrazolopyrimidine derivative of Sildenafil.

  Katalog #	CAS Nummer	Summenformel	Menge
  sc-212604	139755-95-6	C21H28N6O4S	1 mg

• (R)-(+)-2'-O-Benzyloxy-2-O-desmethylcarvedilol
  An analogue of Carvedilol that has multiple-action and is a neurohormonal antagonist that is used in the treatment of hypertension.

  Katalog #	CAS Nummer	Summenformel	Menge
  sc-219724	n.n.	C30H30N2O4	1 mg

• (R)-(+)-5'-Benzyloxy Carvedilol
  An analogue of Carvedilol that has multiple-action and is a neurohormonal antagonist that is used in the treatment of hypertension.

  Katalog #	CAS Nummer	Summenformel	Menge
  sc-219727	n.n.	C31H32N2O5	1 mg

• (R)-(+)-Warfarin
  CYP1A2/3A4 substrate. Anticoagulant.

  Katalog #	CAS Nummer	Summenformel	Menge
  sc-255498	5543-58-8	C19H16O4	5 mg

• rac 4-Amino Deprenyl
  Deprenyl structural analog.

  Katalog #	CAS Nummer	Summenformel	Menge
  sc-212707	217808-43-0	C13H18N2	2.5 mg

• rac 4-Azido Deprenyl
  Photoaffinity analogue of Deprenyl.

  Katalog #	CAS Nummer	Summenformel	Menge
  sc-219782	n.n.	C13H16N4	5 mg

• rac-cis-N-Desmethyl Sertraline Hydrochloride
  A racemate of a metabolite of Sertraline. N-Desmethyl sertraline is significantly less active analogue compared to Sertraline.

  Katalog #	CAS Nummer	Summenformel	Menge
  sc-208291	91797-57-8	C16H16Cl3N	5 mg

• rac-trans-N-Desmethyl Sertraline Hydrochloride
  This is a metabolite of Sertraline. It is used for treatment of CNS disorders.

  Katalog #	CAS Nummer	Summenformel	Menge
  sc-219920	1310676-34-6	C16H16Cl3N	10 mg

• Reversan
  A selective inhibitor of multidrug resistance-associated protein 1 (MRP1) and P-glycoprotein (P-gp). Increases the sensitivity of MRP1-overexpressing tumor cells (MCF7/VP) to doxorubicin, vincristine and etoposide by 3.8-, 14.6- and 11.6-fold respectively. Increases the efficacy of vincristine and etoposide in murine models of neuroblastoma in vivo. Has been shown to display activity on MRP2, MRP3, MRP5 and MRP5 transporters.

  Katalog #	CAS Nummer	Summenformel	Menge
  sc-296262	313397-13-6	C26H27N5O2	10 mg/50 mg

• Ro106-9920, Control
  A cell-permeable tetrazolopyridazine-phenylsulfide analog which serves as an inactive control.

  Katalog #	CAS Nummer	Summenformel	Menge
  sc-222260	n.n.	C10H7N5S	1 mg

• (S)-(-)-5'-Benzyloxyphenyl Carvedilol
  An optically active metabolite of Carvedilol which is a multiple-action, neurohormonal antagonist that is used in the treatment of hypertension.

  Katalog #	CAS Nummer	Summenformel	Menge
  sc-220034	887353-00-6	C31H32N2O5	1 mg

• (S)-(-)-Warfarin
  CYP2C9 substrate; anticoagulant.

  Katalog #	CAS Nummer	Summenformel	Menge
  sc-253488	5543-57-7	C19H16O4	5 mg

• Salicyl sulfate disodium salt
  Phase II metabolite of aspirin; analgesic; anti-inflammatory.

  Katalog #	CAS Nummer	Summenformel	Menge
  sc-253528	56343-01-2	C7H4Na2O6S	5 mg

• Sildenafil
  A type 5 cGMP phosphodiesterase (PDE5) inhibitor and a potential mild vasodilator.

  Katalog #	CAS Nummer	Summenformel	Menge
  sc-338584	139755-83-2	C22H30N6O4S	1 g

• SMC Proliferation Inhibitor-2w
  A diaryl amide analog that exhibits about 15 fold greater selectivity in inhibiting the proliferation of human coronary artery smooth muscle cells over the endothelial cells.

  Katalog #	CAS Nummer	Summenformel	Menge
  sc-222319	n.n.	C21H25NO8	5 mg

• Steviol
  An inhibitor of hOAT1 and hOAT3 organic anion transporters. Human organic anion transporter hOAT1 belongs to a superfamily of organic anion transporters, which play critical roles in the body disposition of clinically important drugs including anti-HIV therapeutics, anti-tumor drugs, antibiotics, anti-hypertensives, and anti-inflammatories. Also a useful tool for studying renal drug clearance.

  Katalog #	CAS Nummer	Summenformel	Menge
  sc-253605	471-80-7 (anhydrous)	C20H30O3 ·xH2O	50 mg

• Sulfadiazine sodium salt

  Katalog #	CAS Nummer	Summenformel	Menge
  sc-251082	547-32-0	C10H9N4NaO2S	25 g

• Tetraiodothyroformic Acid
  Thyroxine impurity and a potent thyroid hormone analog.

  Katalog #	CAS Nummer	Summenformel	Menge
  sc-213024	2055-97-2	C13H6I4O4	2.5 mg

• Thiohomo Sildenafil
  An analog of the cGMP-specific phosphodiesterase type 5 inhibitor Sildenafil.

  Katalog #	CAS Nummer	Summenformel	Menge
  sc-213034	479073-80-8	C23H32N6O3S2	5 mg

• trans-(E)-1-Bromo-2-[4-[2-(dimethylamino)ethoxy]phenyl]-1,2-diphenylethene
  An analogue of tamoxifen with anti-estrogenic properties.

  Katalog #	CAS Nummer	Summenformel	Menge
  sc-213076	19118-19-5	C24H24BrNO	10 mg

• Trityl Olmesartan Medoxomil
  An Olmesartan medoxomil intermediate.

  Katalog #	CAS Nummer	Summenformel	Menge
  sc-213128	144690-92-6	C48H44N6O6	10 mg

• Trospectomycin Dihydrochloride
  A Spectinomycin analog

  Katalog #	CAS Nummer	Summenformel	Menge
  sc-216025	85951-37-7	C17H30N2O7	50 mg

• γ-Secretase Inhibitor XI
  A cell-permeable, active site directed, irreversible serine protease inhibitor that belongs to the class of isocoumarin analogs. Acts as a potent and selective inhibitor of γ-secretase and blocks the production of both amyloid-β40 and Aβ42 in HEK293 cells expressing wild-type and Swedish-mutant β-amyloid precursor protein (APP).

  Katalog #	CAS Nummer	Summenformel	Menge
  sc-222305	n.n.	C10H8ClNO3	5 mg

• γ-Secretase Inhibitor XVI
  A cell-permeable γ-secretase inhibitor with anti-aggregation properties. Prevents early Aβ oligomerization by selectively blocking the Aβ dimer and Aβ trimer formation.

  Katalog #	CAS Nummer	Summenformel	Menge
  sc-222306	208255-51-0	C20H20F2N2O4	5 mg

• γ-Secretase Inhibitor XX
  A γ-secretase inhibitor which has also been shown to inhibit Notch processing.

  Katalog #	CAS Nummer	Summenformel	Menge
  sc-222307	209984-56-5	C26H23F2N3O3	500 µg