Dopaminergics

2-Chloro-11-(4-methylpiperazino)dibenz[b,f]oxepin maleate
A high affinity dopamine D4 receptor ligand that is almost 40 times more potent than clozapine.
Katalog # CAS Nummer Summenformel Menge
sc-205920 n.n. C₁₉H₁₉N₂OCl ·C₄H₄O₄ 5 mg
3-(3,4-Dimethylphenyl)-1-propyl-piperidine hydrochloride
Highly selective ligand for the D4 dopamine receptor.
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sc-202411 219704-16-2 C₁₆H₂₅N•HCl 1 mg/5 mg
3-CPMT
Cocaine analog that binds with high affinity to the dopamine transporter (Ki = 30 nM) and blocks re-uptake of dopamine. However, it is a weak psychomotor stimulant and does not substitute for cocaine in addicted rats.
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sc-203777 14008-79-8 C₂₁H₂₄CINO•HCl 10 mg/50 mg
3-Hydroxytyramine, Hydrochloride
Dopaminergic neurotransmitter. Precursor of adrenaline and noradrenaline.
Katalog # CAS Nummer Summenformel Menge
sc-202417 62-31-7 C₈H₁₂ClNO₂ 25 g
3-Mercaptotyramine, Hydrochloride
A 3-Mercaptotyramine and the mercapto analog of dopamine which irreversibly inhibits the enzyme, catechol-O-methyltransferase by the formation of an SS bridge to a reactive mercapto group in the reactive site.
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sc-206656 37736-93-9 C₈H₁₁NOS•HCl 10 mg
3'-Fluorobenzylspiperone maleate
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sc-361079 n.n. C₃₀H₃₁F₂N₃O₂.C₄H₄O₄ 10 mg/50 mg
3α-Bis-(4-fluorophenyl) methoxytropane hydrochloride
A potent inhibitor of dopamine uptake and transport (Ki = 11.8 nM).
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sc-203778 n.n. C₂₁H₂₃F₂NO ·HCl 10 mg/50 mg
4-Phenyl-1,2,3,4-tetrahydroisoquinoline hydrochloride
Inhibitor of release of dopamine induced by methamphetamine.
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sc-203476 75626-12-9 C₁₅H₁₅N ·HCl 10 mg/50 mg
6-Hydroxydopamine hydrochloride
Selective catecholaminergic neurotoxin. Depletes brain catecholamine levels via uptake and accumulation by a transport mechanism specific to these neurons. Causes almost complete destruction of nigral dopaminergic neurons and their striatal terminals when injected into the substantia nigra of rats, producing an animal model of Parkinson's disease.
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sc-203482 28094-15-7 C₈H₁₁NO₃ ·HCl 100 mg
6,7-ADTN·HBr
6,7-ADTN is a potent dopamine agonist that displays some alpha adrenergic activity as well.
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sc-200393 73304-33-3 C₁₀H₁₃NO₂ ·HBr 25 mg
7-Hydroxy-DPAT·HBr
A selective D-3 dopamine receptor agonist that is primarily found in neurons of the brain.
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sc-200400 74938-11-7 C₁₆H₂₅NO ·HBr 10 mg/50 mg
7-Hydroxy-PIPAT maleate
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sc-361088 159559-71-4 C₁₆H₂₂INO.C₄H₄O₄ 5 mg/50 mg
A 68930 hydrochloride
Potent and selective D1-like dopamine receptor agonist (EC₅₀ values are 2.1 and 3910 nM for D1-like and D2-like receptors respectively). Centrally active following systemic administration in vivo.
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sc-203485 130465-39-3 C₁₆H₁₇NO₃ ·HCl 10 mg/50 mg
A 77636 hydrochloride
A selective and potent dopamine D1-like agonist stimulating the release of adenylate cyclase. It has been reported that upon binding to dopamine D1 receptors, A 77636 hydrochloride displays 85% of the intrinsic activity that dopamine provides.
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sc-203486 145307-34-2 C₂₀H₂₇NO₃.HCl 10 mg/50 mg
A-77636 hydrochloride hydrate
This is a potent, orally active D1 dopamine receptor agonist.
Katalog # CAS Nummer Summenformel Menge
sc-239151 145307-34-2 (anhydrous) C₂₀H₂₇NO₃•HCl•xH₂O 10 mg
ABT 724 trihydrochloride
A selective dopamine D₄ receptor partial agonist with an EC₅₀=12.4nM.
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sc-203489 70006-24-5 C₁₇H₁₉N₅ ·3HCl 10 mg/50 mg
ABT-418 hydrochloride
Neuronal nicotinic acetylcholine receptor agonist with anxiolytic and cognition enhancing activities.
Katalog # CAS Nummer Summenformel Menge
sc-239177 147388-83-8 C₉H₁₄N₂O•HCl 5 mg
AJ-76 HCL
A selective antagonist of dopamine autoreceptors, which displays a reduction in ventral firing rates of dopaminergic neurons.
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sc-200394 85379-09-5 C₁₅H₂₄ClNO 10 mg
AMI-193
Selective 5-HT antagonist that binds to 5-HT₂ sites as potently as spiperone but has lower affinity for 5-HT_2C receptors.
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sc-203509 510-74-7 C₂₂H₂₆FN₃O₂ 10 mg/50 mg
Amisulpride
Selective, potent dopamine D2 and D3 receptor antagonist. (Ki values are 2.8 and 3.2 nM respectively for human D2 and D3 and > 1000 nM for human D1, D4 and D5 receptors.)
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sc-203510 71675-85-9 C₁₇H₂₇N₃O₄S 50 mg
B-HT 920
Dopamine D₂ receptor agonist, 5-HT₃ receptor antagonist and α2-adrenoceptor agonist. Also displays antiparkinsonian activity.
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sc-203523 36085-73-1 C₁₀H₁₅N₃S.2HCl 10 mg/50 mg
bis-(4-Methyl-1-homopiperazinylthiocarbonyl)disulfide
A dopamine β-hydroxylase inhibitor.
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sc-202502 26087-98-9 C₁₄H₂₆N₄S₄ 10 mg
Bromocriptine mesylate
An agonist of the D₂ and D₃ dopamine receptors. Demonstrates ten-fold higher affinity at D₂ over D₃ in recombinant dopamine receptors.
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sc-200395 22260-51-1 C₃₂H₄₀BrN₅O₅ ·CH₃SO₃H 100 mg/500 mg
Cabergoline
A D2-like agonist, shown to have a high affinity for serotonin receptors.
Katalog # CAS Nummer Summenformel Menge
sc-203864 81409-90-7 C₂₆H₃₇N₅O₂ 10 mg/50 mg
Carmoxirole hydrochloride
Selective,peripherally acting D2-like agonist
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sc-203539 98323-83-2 C₂₄H₂₆N₂O₂•HCl•xH₂O 10 mg/50 mg
cis-8-Hydroxy-3-(n-propyl)-1,2,3a,4,5,9b-hexahydro-1H-benz[e]indole hydrobromide
D3 dopamine receptor agonist.
Katalog # CAS Nummer Summenformel Menge
sc-300375 n.n. C₁₅H₂₁NO•HBr 5 mg
Clothiapine
Structurally analogous to quetiapine (sc-219681), clothiapine is an atypical antipsychotic of the dibenzothiazepine chemical class.
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sc-200404 2058-52-8 C₁₈H₁₈ClN₃S 20 mg/100 mg
Clozapine
Selective antagonist for D4- and D2-dopamine receptors with activity at several serotonin receptors.
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sc-200402 5786-21-0 C₁₈H₁₉ClN₄ 50 mg/500 mg
CY 208-243
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sc-361163 100999-26-6 C₁₉H₁₈N₂ 10 mg/50 mg
Diclofensine
A stimulant. Inhibits reuptake of dopamine and noradrenaline, is an effective antidepressant. Compound exhibits significant addictive properties.
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sc-207563 67165-56-4 C₁₇H₁₇Cl₂NO 10 mg
Dihydrexidine hydrochloride
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sc-361168 123039-93-0 C₁₇H₁₇NO₂.HCl 5 mg/25 mg
Domperidone
An antagonist of the peripheral dopamine D₂-like receptors.
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sc-203032 57808-66-9 C₂₂H₂₄ClN₅O₂ 50 mg/250 mg
Eticlopride hydrochloride
Selective dopamine D₂/D₃ receptor antagonist (K_i values are 0.50 and 0.16 nM respectively). Antipsychotic.
Katalog # CAS Nummer Summenformel Menge
sc-203576 97612-24-3 C₁₇H₂₅ClN₂O₃•HCl 10 mg/50 mg
FAUC 73
Selective, nonaromatic, potent D3 dopamine receptor agonist.
Katalog # CAS Nummer Summenformel Menge
sc-300690 n.n. C₁₄H₂₃N 5 mg
Fenoldopam hydrochloride
Selective D1-like dopamine receptor partial agonist. Vasodilator in vivo and does not readily cross the blood-brain barrier. Also α2-adrenoceptor antagonist in vitro.
Katalog # CAS Nummer Summenformel Menge
sc-279160 67227-56-9 C₁₆H₁₆ClNO₃.HCl 10 mg
Fenoldopam monohydrobromide
A selective dopamine agonist that is being considered for the parenteral treatment of systemic hypertension. In both an oral and parenteral form, this compound causes peripheral vasodilation by stimulating dopamine-1 adrenergic receptors. Intravenous fenoldopam may provide advantages over sodium nitroprusside because it can induce both a diuresis and natriuresis. It is not light sensitive, nor is it associated with cyanide toxicity. There is no evidence for rebound hypertension after discontinuation of fenoldopam infusion.
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sc-215032 67287-54-1 C₁₆H₁₆ClNO₃ ·HBr 5 mg/20 mg
GBR 12783 dihydrochloride
A very potent and selective inhibitor of dopamine uptake (IC₅₀ for inhibition of [3H]-dopamine uptake in rat striatal synaptosomes is 1.8 nM).
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sc-203587 67469-57-2 C₂₈H₃₂N₂O ·2HCl 10 mg/50 mg
GBR 12935 dihydrochloride
Selective dopamine uptake inhibitor
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sc-203965 76778-22-8 C₂₈H₃₄N₂O ·2HCl 10 mg/50 mg
GBR 12935 dihydrochloride
An inhibitor of the dopamine and norepinephrine transporters with Ki s of 21.5 nM and 225 nM, respectively and it does not inhibit the serotonin transporter (Ki = 6.5 µM). Binds to a nondopaminergic piperazine site in blood platelets and brain that has been identified as cytochrome P450.
Katalog # CAS Nummer Summenformel Menge
sc-215069 67469-81-2 C₂₈H₃₄N₂O ·2HCl 25 mg/100 mg
GBR 13069 dihydrochloride
Potent dopamine uptake inhibitor. Systemically active post-administration in vivo.
Katalog # CAS Nummer Summenformel Menge
sc-203966 77862-93-2 C₂₈H₃₀F₂N₂O•2HCl 10 mg/50 mg
GR 103691
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sc-361188 162408-66-4 C₃₀H₃₅N₃O₃ 10 mg/50 mg
Haloperidol hydrochloride
Dopamine antagonist partly selectivity for D2-like receptors (Ki values are 1.2, ~ 7, 2.3, ~ 80 and ~ 100 nM for D2, D3, D4, D1 and D5 receptors respectively). Subtype selective NMDA antagonist.
Katalog # CAS Nummer Summenformel Menge
sc-203593 52-86-8 C₂₁H₂₃ClFNO₂ ·HCl 100 mg
Imipramine Hydrochloride
A tricyclic antidepressant. Inhibits the serotonin and norepinephrine transporters but has little effect on the dopamine transporter.
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sc-207753 113-52-0 C₁₉H₂₅ClN₂ 100 mg
L-3,4-Dihydroxyphenylalanine methyl ester hydrochloride
A precursor to L-DOPA which crosses the blood-brain barrier; antiparkinsonian agent.
Katalog # CAS Nummer Summenformel Menge
sc-250211 1421-65-4 C₁₀H₁₃NO₄··HCl 500 mg/1 g
L-741,742 hydrochloride
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sc-361227 156337-32-5 C₂₃H₂₅N₂ClO.HCl 10 mg/50 mg
L-745,870 hydrochloride
This product is a selective D4 dopamine receptor antagonist.
Katalog # CAS Nummer Summenformel Menge
sc-300864 n.n. C₁₈H₁₉ClN₄•HCl 5 mg
L-750,667 trihydrochloride
This product is a selective D4 dopamine receptor antagonist.
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sc-300865 n.n. C₁₈H₁₉IN₄•3HCl 5 mg
LE 300
Potent and selective dopamine D1 receptor antagonist (Ki values are 0.08-1.9 nM and 6-45 nM for D1 and D2 receptors respectively). Also displays moderate affinity for the 5-HT2A receptor (Ki = 20 nM). Active in vivo.
Katalog # CAS Nummer Summenformel Menge
sc-203622 274694-98-3 C₂₀H₂₂N₂•xH₂O 10 mg/50 mg
Levodopa
Natural form of DOPA used in the treatment of Parkinson's disease. Immediate precursor of dopamine and product of tyrosine hydroxylase.
Katalog # CAS Nummer Summenformel Menge
sc-205372 59-92-7 C₉H₁₁NO₄ 5 g/25 g
Lisuride maleate
Katalog # CAS Nummer Summenformel Menge
sc-361233 19875-60-6 C₂₀H₂₆N₄O.C₄H₄O₄ 10 mg/50 mg
Loxapine, Succinate
A D2/D4-Dopamine receptor and serotonergic receptor antagonist. Also a dibenzoxazepine anti-psychotic agent.
Katalog # CAS Nummer Summenformel Menge
sc-211754 27833-64-3 C₂₂H₂₄ClN₃O₅ 500 mg
Mesoridazine besylate
Mesoridazine besylate is a phenothiazine dopamine receptor antagonist. Demonstrates high-affinity for a cloned rat dopamine D4 receptor.
Katalog # CAS Nummer Summenformel Menge
sc-201133 32672-69-8 C₂₁H₂₆N₂OS₂ ·C₆H₆O₃S 1 g
N-[2-(4-(4-Chlorophenyl)piperazin-1-yl)ethyl]-3-methoxybenzamide
A selective and potent ligand for the D4 dopamine receptor.
Katalog # CAS Nummer Summenformel Menge
sc-301260 n.n. n.n. 25 mg
N-Allyl-(±)-SKF-38393 hydrobromide
Selective dopamine D1-like receptor partial agonist. Centrally active following systemic administration in vivo.
Katalog # CAS Nummer Summenformel Menge
sc-224127 300561-58-4 C₁₉H₂₂BrNO₂ 25 mg/100 mg
N-Methyl-(R)-salsolinol hydrobromide
On dopaminergic neurons N-Methyl-(R)-salsolinol hydrobromide acts as an endogenous nerotoxin.
Katalog # CAS Nummer Summenformel Menge
sc-301368 n.n. C₁₁H₁₅NO₂•HBr 1 mg
Nafadotride
Katalog # CAS Nummer Summenformel Menge
sc-361269 149649-22-9 C₂₂H₂₇N₃O₂ 10 mg/50 mg
Nemonapride
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sc-204123 75272-39-8 C₂₁H₂₆ClN₃O₂ 10 mg/50 mg
NGB 2904
Highly-selective dopamine D3 receptor antagonist. Attenuates cocaine's rewarding effects and inhibits relapse to drug-seeking behavior.
Katalog # CAS Nummer Summenformel Menge
sc-204127 189060-98-8 C₂₈H₂₉Cl₂N₃O ·HCl 10 mg/50 mg
NGD 94-1
High affinity D4 receptor ligand and is selective over D1, D2, D3 and D5 receptors.
Katalog # CAS Nummer Summenformel Menge
sc-358837 179333-18-7 C₁₈H₂₀N₆ 10 mg/50 mg
NPEC-caged-dopamine
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sc-359018 n.n. C₁₇H₁₈N₂O₆ 10 mg/50 mg
OSU 6162 hydrochloride
Dopamine stabilizer that lacks high in vitro affinity for various neuroreceptors. In vivo, shows high D2 receptor occupancy and is highly active on dopamine synthesis and turnover. Induces stabilizing effects on psychomotor function in behavioral tests without inducing hypolocomotion or catalepsy.
Katalog # CAS Nummer Summenformel Menge
sc-204825 156907-84-5 C₁₅H₂₃NO₂S ·HCl 10 mg/50 mg
Paliperidone
Serotonin (5-HT2) and dopamine (D2) combined receptor antagonist. Indicated in the treatment of schizophrenia, depression, and manic and mixed episodes occurring in tandem with Bipolar I Disorder.
Katalog # CAS Nummer Summenformel Menge
sc-204828 144598-75-4 C₂₃H₂₇FN₄O₃ 25 mg/100 mg
Palmatine Chloride Hydrate
A protoberberine alkaloid that is isolated from medicinal herbs like Coptis chinensis Franch. Sedative effect of palmatine is related to its ability to inhibit dopamine generation. It also acts as a selective topoisomerase I and II position and as vasodilator that effectively reduces Ca²⁺ concentration.
Katalog # CAS Nummer Summenformel Menge
sc-205788 171869-95-7 C₂₁H₂₂NO₄•Cl•xH₂O 1 g/5 g
(+)-PD 128907 HYDROCHLORIDE
Potent D3 dopamine receptor agonist (Ki = 2.3 nM). Displays 18-200-fold selectivity over other dopamine receptor subtypes.
Katalog # CAS Nummer Summenformel Menge
sc-204162 300576-59-4 C₁₄H₂₀ClNO₃ 10 mg/50 mg
PD 168077 maleate
D4 dopamine agonist. >400-fold selectivity over D2 with >300-fold selectivity v.s. D3 subtypes. Generates synaptic translocation of CaMK II to postsynaptic sites in cultured prefrontal cortical neurons. Shown to be centrally active in vivo.
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sc-204165 190383-31-4 C₂₀H₂₂N₄O ·C₄H₄O₄ 10 mg/50 mg
PD 168568 dihydrochloride
Selective D4 antagonist. Reverses amphetamine-stimulated movement in vivo and is orally active.
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sc-204167 210688-56-5 C₂₂H₂₇N₃O ·2HCl ·xH₂O 10 mg
Pergolide Mesylate
An antiparkinsonian agent. A dopaminergic agonist that also decrease plasma prolactin concentrations.
Katalog # CAS Nummer Summenformel Menge
sc-212538 66104-23-2 C₂₀H₃₀N₂O₃S₂ 2.5 mg
Pimozide
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sc-203662 2062-78-4 C₂₈H₂₉F₂N₃O 100 mg
Piribedil dihydrochloride
A dopamine agonist reported to have selectivity for D3 subtype receptors with moderate to non-significant affinity for D2 and D1 receptors.
Katalog # CAS Nummer Summenformel Menge
sc-204198 78213-63-5 C₁₆H₁₈N₄O₂•2HCl 10 mg/50 mg
Piribedil maleate salt
A dopamine agonist reported to have selectivity for D3 subtype receptors with moderate to non-significant affinity for D2 and D1 receptors.
Katalog # CAS Nummer Summenformel Menge
sc-301552 n.n. C₂₀H₂₂N₄O₆ 10 mg
PNU 177864 hydrochloride
Highly selective dopamine D3 receptor antagonist. Exhibits antischizophrenic activity and induces phospholipidosisin vivo.
Katalog # CAS Nummer Summenformel Menge
sc-204205 250266-51-4 C₁₈H₂₁F₃N₂O₃S ·HCl 10 mg/50 mg
PNU 96415E
Displays highest affinity for dopamine D4 and serotonergic 5-HT2A receptors and relatively weak affinity at D2 receptors.
Katalog # CAS Nummer Summenformel Menge
sc-204852 170856-41-4 C₂₁H₂₅FN₂O•2HCl 10 mg/50 mg
Prochlorperazine dimaleate
Antagonist to D2 receptor. Also interacts with 5-HT3 and nAChR. Displays antispasmodic, antipsychotic, antiemetic and antinociceptive activity in vivo.
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sc-204213 84-02-6 C₂₀H₂₄ClN₃S ·2C₄H₄O₄ 100 mg
Quetiapine Fumarate
Used as an antipsychotic. Benzothiazepine with mixed serotonin and dopamine receptor antagonistic properties.
Katalog # CAS Nummer Summenformel Menge
sc-219681 111974-72-2 2(C₂₁H₂₅N₃O₂S)•C₄H₄O₄ 1 g
Quinelorane dihydrochloride
D2 dopamine receptor agonist; 2-aminopyridine analog of quinpirole.
Katalog # CAS Nummer Summenformel Menge
sc-255455 97548-97-5 C₁₄H₂₂N₄•2HCl 5 mg/25 mg
(-)-Quinpirole·HCl
An agonist of D₂-like dopamine receptors. Stimulation of D₂ receptors demonstrates a neuroprotective effect against glutamate excitotoxicity and oxidative damage.
Katalog # CAS Nummer Summenformel Menge
sc-200406 85760-74-3 C₁₃H₂₁N₃ ·HCl 5 mg/25 mg
R (+)-Eticloride hydrochloride
The inactive enantiomer of the dopamine D2 antagonist S(-)-Eticlopride
Katalog # CAS Nummer Summenformel Menge
sc-296183 84226-12-0 C₁₇H₂₅ClN₂O₃•HCl 5 mg/10 mg
R(+)-6-Bromo-APB hydrobromide
This product is the more potent D1 Dopamine receptor agonist enantiomer.
Katalog # CAS Nummer Summenformel Menge
sc-301656 139689-19-3 C₁₉H₂₁Br₂NO₂ 25 mg
(R)-(-)-Apomorphine hydrochloride
Prototypical dopamine agonist (pK_i values are 6.43, 7.08, 7.59, 8.36, and 7.83 for human recombinant D₁, D_2L, D₃, D₄ and D₅ receptors respectively).
Katalog # CAS Nummer Summenformel Menge
sc-203675 314-19-2 C₁₇H₁₇NO₂ ·HCl 50 mg
Raclopride
Potent,selective D2/D3 antagonist. Centrally active post systemic administration in vivo.
Katalog # CAS Nummer Summenformel Menge
sc-204229 84225-95-6 C₁₅H₂₀Cl₂N₂O₃ 10 mg/50 mg
RBI 257 maleate salt
A high affinity D4 dopamine receptor ligand.
Katalog # CAS Nummer Summenformel Menge
sc-311521 n.n. C₂₁H₂₈IN₃O ··· ·C₄H₄O₄ 10 mg
Remoxipride Hydrochloride
Remoxipride, a substituted benzamide, is an atypical antipsychotic agent and a selective and potent dopamine D2 agonist, binding to dopamine D2 receptors.
Katalog # CAS Nummer Summenformel Menge
sc-200410 73220-03-8 C₁₆H₂₃BrN₂O₃··HCl 10 mg/50 mg
Ro 10-5824 dihydrochloride
Selective dopamine D4 receptor partial agonist that binds with high affinity (K_i = 5.2 nM). Displays 250-fold selectivity over D3 receptors and > 1000-fold selectivity over D2, D1 and D5 receptors.
Katalog # CAS Nummer Summenformel Menge
sc-204886 189744-46-5 C₁₇H₂₀N₄.2HCl 10 mg/50 mg
Roxindole hydrochloride
Selective and potent presynaptic D-2 dopamine autoreceptor agonist. Inhibits serotonin (5-HT) uptake.
Katalog # CAS Nummer Summenformel Menge
sc-203685 112192-04-8 C₂₃H₂₆N₂O.HCl 10 mg/50 mg
(RS)-(±)-Sulpiride
Selective antagonist at postsynaptic D2-receptors. Also found to upregulate GHB receptors in rats.
Katalog # CAS Nummer Summenformel Menge
sc-205494 15676-16-1 C₁₅H₂₃N₃O₄S 100 mg
S(-)-DS 121 hydrochloride
Dopamine autoreceptor antagonist with selectivity for the D3 dopamine receptor.
Katalog # CAS Nummer Summenformel Menge
sc-311528 n.n. C₁₅H₂₀N₂•HCl•0.5HCO₃ 5 mg
(S)-(-)-Sulpiride
D2 dopamine receptor antagonist; antipsychotic.
Katalog # CAS Nummer Summenformel Menge
sc-258111 23672-07-3 C₁₅H₂₃N₃O₄S 5 g
SCH 23390
A selective and highly effective dopamine D1 and D5 receptor antagonist. In vitro studies reveal its ability to bind to the serotonin receptors 5-HT2 and 5-HT1C.
Katalog # CAS Nummer Summenformel Menge
sc-200408 125941-87-9 C₁₇H₁₈ClNO•HCl 5 mg/25 mg
SCH 39166 hydrobromide
High affinity dopamine D1/D5 receptor antagonist; displays Ki values of 1.2, 2, 980, 5520, 80 and 731 nM for binding to D1, D5, D2, D4, 5-HT and α2a receptors, respectively.
Katalog # CAS Nummer Summenformel Menge
sc-204270 n.n. C₁₉H₂₀ClNO.HBr 10 mg/50 mg
SKF 38393 HCl
A selective dopamine D₁ receptor agonist that seems to be correlated to induced desynchronization of electroencephalographic activity in rats.
Katalog # CAS Nummer Summenformel Menge
sc-203264 81633-77-4 C₁₆H₁₇NO₂ ·HCl 25 mg
SKF 81297 hydrobromide
Dopamine D1-like receptor agonist. Centrally active following systemic administration in vivo.
Katalog # CAS Nummer Summenformel Menge
sc-204283 71636-61-8 C₁₆H₁₆ClNO₂ ·HBr 10 mg/50 mg
SKF 83566 hydrobromide
Katalog # CAS Nummer Summenformel Menge
sc-361360 108179-91-5 C₁₇H₁₈BrNO ·HBr 10 mg/50 mg
SKF 83822 hydrobromide
High affinity, selective dopamine D1-like receptor agonist. K_i values are 3.2, 3.1, 186, 66, 335, 1167, 1251 and 1385 nM at recombinant D1, D5, D2, D3, D4, 5-HT2A, α1A and α1B receptors respectively. Stimulates adenylyl cyclase (EC₅₀ = 65 nM) but not phosphoinositide hydrolysis. Induces extreme arousal and hyperlocomotion following subcutaneous administration in monkeys.
Katalog # CAS Nummer Summenformel Menge
sc-204284 74115-08-5 C₂₀H₂₂ClNO₂ ·HBr 10 mg/50 mg
SKF 83959
D1-like partial agonist. May act as an antagonist in vivo, exhibiting antiparkinsonian effects and antagonizing the behavioral effects of cocaine.
Katalog # CAS Nummer Summenformel Menge
sc-204285 80751-85-5 C₁₈H₂₀ClNO₂ ·HBr 10 mg/50 mg
SKF-75670 hydrobromide
Atypical D1 dopamine receptor agonist. Displays antagonist activity in vitro and agonist activity in vivo.
Katalog # CAS Nummer Summenformel Menge
sc-301809 62717-63-9 C₁₇H₁₉NO₂•HBr 5 mg
SKF-89145 hydrobromide
D1 dopamine receptor agonist.
Katalog # CAS Nummer Summenformel Menge
sc-301811 n.n. C₁₄H₁₅NO₂S•HBr 5 mg
SKF-89626 hydrobromide
D1 dopamine receptor agonist.
Katalog # CAS Nummer Summenformel Menge
sc-301812 n.n. C₁₃H₁₄BrNO₂S 25 mg
ST-148
ST-148 is a D2 dopamine receptor antagonist. Compared to haloperidol and (S)-nafodotride, ST-148 exhibits improved selectivity for hD2L receptors. ST-148 has a pKi = 7.85 at hD2L receptors.
Katalog # CAS Nummer Summenformel Menge
sc-301838 n.n. C₃₁H₄₀N₄O₇S 5 mg
Tetrabenazine
Potent inhibitor of vesicular monoamine uptake; depletes stores of serotonin, dopamine and noradrenalin.
Katalog # CAS Nummer Summenformel Menge
sc-204338 58-46-8 C₁₉H₂₇NO₃ 10 mg/50 mg
Thioridazine·HCl
Dopamine D4 receptor antagonist. High affinity for the cloned rat dopamine D4 receptor (K_i<20 nM).
Katalog # CAS Nummer Summenformel Menge
sc-201149 130-61-0 C₂₁H₂₆N₂S₂ ·HCl 5 g/5 mg
U 99194 maleate
Potent,selective D3 antagonist
Katalog # CAS Nummer Summenformel Menge
sc-204365 83598-46-3 C₂₁H₃₁NO₆ 10 mg/50 mg
U-101958 Maleate
Selective D4 dopamine receptor antagonist.
Katalog # CAS Nummer Summenformel Menge
sc-222396 n.n. C₂₁H₂₉N₃O··C₄H₄O₄ 5 mg
U-99194A maleate
D3 dopamine receptor agonist.
Katalog # CAS Nummer Summenformel Menge
sc-202373 153570-58-2 C₁₇H₂₇NO₂ ·C₄H₄O₄ 10 mg/50 mg
(+)-UH 232 maleate
D2-likeautoreceptor antagonist and D3 partial agonist.
Katalog # CAS Nummer Summenformel Menge
sc-203717 95999-12-5 C₁₈H₂₉NO ·C₄H₄O₄ 10 mg/50 mg
Zotepine
Katalog # CAS Nummer Summenformel Menge
sc-360895 26615-21-4 C₁₈H₁₈ClNOS 10 mg/50 mg