| | Adrenergic Effectors
- 1-[4-(2-methoxyethyl)phenoxy]-3-propan-2-ylamino-propan-2-ol
| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-264643 | 51384-51-1 | C15H25NO3 | 2.5 g |
- 1'-Hydroxy Bufuralol-d9 (Mixture of Diastereomers)
A β-Adrenergic blocker with peripheral vasodilating activity, and a metabolite of Bufuralol.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-213561 | n.n. | C16H14D9NO3 | 500 µg |
- 2-MPMDQ
Potent and selective α1-adrenoceptor antagonist; hypotensive.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-203770 | n.n. | C23H27N5O2 | 10 mg/50 mg |
- 2-PMDQ
A potent and selective α1-adrenoceptor antagonist and antihypertensive.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-203771 | n.n. | C21H23N5O | 10 mg/50 mg |
- 3-MPPI
| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-361078 | n.n. | C23H25N5O3 | 10 mg/50 mg |
- [[4-[2-(Cyclopropylmethoxy)ethyl]phenoxy]methyl]oxirane
| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-362012 | 63659-17-6 | C15H20O3 | 25 mg |
- A 61603 HYDROBROMIDE
Potent α-adrenoceptor agonist, at least 35-fold more potent at α1A than at α1B or α1D sites. | Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-203789 | 107756-30-9 | C14H19N3O3S ·HBr | 10 mg/50 mg |
- A 80426 mesylate
| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-361095 | 152148-63-5 | C23H27NO2.CH3SO3H | 10 mg/50 mg |
- A-61603 hydrate
This is an α1A agonist, which is used in radioligand binding assays.
| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-300145 | n.n. | C14H19N3O3S··HBr•xH2O | 10 mg |
- AH 11110 hydrochloride
Subtype-selective ligand for the α1B-adrenoceptor. | Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-203502 | 179388-65-9 | C21H26N2O2•HCl | 10 mg/50 mg |
- Alfuzosin hydrochloride
An uro-selective α 1 adrenoceptor antagonist that does not distinguish between α 1 subtypes. Also Alfuzosin hydrochloride has been seen to inhibit the increase of intraurethral pressure caused by phenylephrine.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-203812 | 81403-68-1 | C19H27N5O4•HCl | 10 mg/50 mg |
- Alprenolol hydrochloride
β-adrenoceptor (β2 > β1 > β3) and a 5-HT1A receptor antagonist.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-203503 | 13707-88-5 | C15H23NO2.HCl | 50 mg |
- ARC 239 dihydrochloride hydrate
A selective α2B adrenoceptor antagonist with a pKD value of 8.8.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-203518 | 67339-62-2 | C24H29N3O3•2HCl•xH2O | 5 mg |
- Atipamezole hydrochloride
| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-291914 | 104075-48-1 | C14H16N2•HCl | 10 mg/50 mg |
- Betaxolol hydrochloride
Selective β1-adrenoceptor antagonist.
| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-203527 | 63659-19-8 | C18H29NO3.HCl | 10 mg/50 mg |
- (±)-Bisoprolol hemifumarate
Selective β1-adrenergic antagonist. Has β1/β2 selectivity of approximately 100-fold and a Kd of 2-3 nM at the β1 receptor.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-203531 | 104344-23-2 | C18H31NO4 ·½C4H4O4 | 10 mg/50 mg |
- BMY 7378 dihydrochloride
Putative 5-HT1A antagonist, selective a1D antagonist.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-203849 | 21102-95-4 | C22H31N3O3 ·2HCl | 10 mg/50 mg |
- Bopindolol malonate
A β1-adrenoceptor antagonist which slowly dissociates into active metabolites. Stabilizes membranes against H2O2-induced lipid peroxidation. Demonstrates antioxidant radical scavenging activity.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-200144 | 62658-64-4 | C23H28N2O3•C3H4O4 | 100 mg/500 mg |
- BRL 44408 MALEATE
Selective a2A antagonist| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-217791 | 118343-19-4 | C13H17N3 ·C4H4O4 | 10 mg |
- BRL-37344
Potent selective agonist of the β3-adrenergic receptor. Stimulates lipolysis in white adipocytes and lipolysis/thermogenesis in brown adipocytes.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-200154 | 127299-93-8 | C19H21ClNO4··Na | 5 mg |
- BU 226 hydrochloride
A high affinity ligand for I2 imidazoline sites (Ki = 2.7 nM) with very high selectivity (> 2000-fold) over α2 -adrenoceptors (Ki = 6700 nM).| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-203858 | n.n. | C12H11N3 ·HCl | 10 mg/50 mg |
- Bucindolol
Non-selective β-adrenoceptor antagonist with additional α1-adrenoceptor blocking activity. | Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-203860 | 71119-11-4 | C22H25N3O2 | 10 mg/50 mg |
- Carvedilol
A α1 and β-adrenergic receptor agonist with antioxidant properties. Shown to block the oscillatory intracellular calcium changes induced by α1D-AR and α1B-AR.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-200157 | 72956-09-3 | C24H26N2O4 | 100 mg |
- CGP 12177 hydrochloride
b3 partial agonist. b1/b2 antagonist| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-203878 | 81047-99-6 | C14H22ClN3O3 | 10 mg/50 mg |
- CGP 20712 Dihydrochloride
Highly potent and selective b1 antagonist| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-203879 | 105737-62-0 | C23H25F3N4O5 ·2HCl ·xH2O | 10 mg/50 mg |
- Cimaterol
β-Adrenergic agonist.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-203549 | 54239-37-1 | C12H17N3O | 10 mg/50 mg |
- Cirazoline hydrochloride
Selective a1 agonist| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-203550 | 40600-13-3 | C13H16N2O.HCl | 10 mg |
- CL 316243 disodium salt
Highly selective beta 3-adrenoceptor agonist; anti-obesity agent.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-203895 | 151126-84-0 | C20H18ClNNa2O7•xH2O | 10 mg/50 mg |
- Clonidine hydrochloride
Prototypical I1 imidazoline receptor ligand. α2-adrenergic receptor agonist. Antihypertensive.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-203002 | 4205-91-8 | C9H9CI2N3.HCl | 1 g |
- Clonidine-d4 Hydrochloride
α2-Adrenergic agonist. Antihypertensive
analgesic for neuropathic pain.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-217935 | 67151-02-4 | C9H6D4Cl3N3 | 1 mg |
- Corynanthine
| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-363622 | 483-10-3 | C21H26N2O3 | 100 mg |
- Desipramine HCl
A selective inhibitor of noradrenaline transporters SLC6A2 (norepinephrine transporter; NET), ST (SERT; serotonin transporter), and DAT (dopamine transporter).| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-200158 | 58-28-6 | C18H22N2 ·HCl | 100 mg/1 g |
- Dexmedetomidine hydrochloride
Medetomide’s active isomer which is a potent, highly selective α2-adrenoceptor agonist.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-205290 | 145108-58-3 | C13H16N2 ·HCl | 10 mg/50 mg |
- Dihydroergotamine mesylate
Partial α-adrenergic agonist. Partial D2 dopaminergic receptor agonist. Competitive 5-HT antagonist.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-203565 | 6190-39-2 | C33H37N5O5 ·CH4O3S | 100 mg |
- Dobutamine Hydrochloride
Dobutamine is a derivative of dopamine and is used as a β1-adrenergic agonist.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-203031 | 49745-95-1 | C18H23NO3.HCl | 10 mg/50 mg |
- Dopamine-d4 Hydrochloride
Endogenous catecholamine with α and β-adrenergic activity. Cardiotonic
antihypotensive.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-218267 | 203633-19-6 | C8H8D4ClNO2 | 1 mg |
- DSP-4 hydrochloride
Adrenergic neuron blocking agent with long-lasting inhibitory effect on the uptake of noradrenaline (norepinephrine) in brain slices.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-202145 | 40616-75-9 | C11H15BrClN ·HCl | 5 mg |
- Efaroxan hydrochloride
| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-203573 | 89197-00-2 | C13H16N2O•HCl | 10 mg/50 mg |
- ent-Levobunolol, Hydrochloride
A non-selective β-adrenoceptor antagonist and the enantiomer of levobunolol.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-211411 | 27867-05-6 | C17H26ClNO3 | 100 mg |
- Esmolol Hydrochloride
An anti-arrhythmic, cardioselective, β-adrenergic blocker.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-211424 | 81161-17-3 | C16H25NO4 ·HCl | 10 mg |
- Formoterol Fumarate
Shown to be a potent agonist of β-adrenoceptor with a fast onset of effect on the isolated human bronchus model. More selective for β2 than β1 receptors.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-203050 | 43229-80-7 | (C19H24N2O4)2•C4H4O4•2H2O | 10 mg/50 mg |
- Guanabenz acetate
| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-203590 | 23256-50-0 | C8H8Cl2N.CH3CO2H | 100 mg |
- Guanfacine hydrochloride
A centrally acting anti-hypertensive agent that has been shown to be a specific α2A-adrenoceptor agonist. Activation of these receptors is reported to cause a decrease in blood pressure.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-203988 | 29110-48-3 | C9H9Cl2N3O ·HCl | 10 mg/50 mg |
- HEAT hydrochloride
Very selective α1-adrenoceptor antagonist, precursor of the 3-[125I]-derivative.
| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-203996 | 30007-39-7 | C19H22ClNO2 | 10 mg/50 mg |
- ICI 89406
| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-361212 | 53671-71-9 | C19H22N4O3 | 10 mg/50 mg |
- ICI 118,551 hydrochloride
| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-361206 | 72795-01-8 | C17H27NO2.HCl | 10 mg |
- ICI 215,001 hydrochloride
| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-361210 | 141269-99-0 | C19H23NO6.HCl | 10 mg/50 mg |
- Idazoxan hydrochloride
| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-204006 | 79944-56-2 | C11H12N2O2•HCl | 10 mg/50 mg |
- Imiloxan Hydrochloride
Highly selective a2B antagonist| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-224023 | 81167-16-0 | C14H16N2O2.HCl | 5 mg/25 mg |
- Isoproterenol Hydrochloride
Phenethylamine derivative. Selective β-adrenergic agonist that increases cytosolic cAMP. Promotes glycogen breakdown and causes bronchodilation.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-202188 | 51-30-9 | C11H17NO3 ·HCl | 100 mg/500 mg |
- JP 1302 dihydrochloride
Potent and selective a2C antagonist. Strongly antagonizes adrenaline-stimulated 35GTPγS binding in vitro. Produces antidepressant and antipsychotic-like effects in vivo.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-204026 | 80259-18-3 | C24H24N4•2HCl•xH2O | 10 mg/50 mg |
- L-(-)-Epinephrine-(+)-bitartrate
An α,β-adrenergic receptor agonist. | Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-204032 | 51-42-3 | C9H13NO3 ·C4H6O6 | 100 mg |
- L-(–)-Norepinephrine-(+)-bitartrate
A bitartrate preparation of the α,β-adrenoceptor agonist norepinephrine. Used as a source of norepinephrine in studies of vascular contractility.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-203093 | 69815-49-2 | C8H11NO3 ·C4H6O6 | 100 mg |
- L-748,337
| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-204044 | 244192-94-7 | C26H31N3O5S•xH2O | 10 mg/50 mg |
- L-755,507
Verypotent and selective β3-adrenergic receptor partial agonist, selective over both β1- and β2-adrenoceptor binding. | Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-204045 | 159182-43-1 | C30H40N4O6S | 10 mg/50 mg |
- L-765,314 hydrate
This product is a potent and selective α1B-adrenoceptor antagonist.
| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-300866 | n.n. | C27H34N6O5•xH2O | 5 mg |
- L-α-Methyl-DOPA · sesquihydrate
L-Aromatic amino acid decarboxylase inhibitor. Adrenergic inhibiting agent used for antihypertensive treatment.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-204788 | 41372-08-1 | C10H13NO4 ·1.5 ·H2O | 1 g |
- Levobunolol, Hydrochloride
A non-selective β-adrenoceptor antagonist.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-211734 | 47141-42-4 | C17H26ClNO3 | 250 mg |
- Lofexidine Hydrochloride
An adrenoceptor agonist that is structurally related to Clonidine and used in the treatment of opioid withdrawal symptoms as well as an anihypertensive.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-205733 | 21498-08-8 | C11H12Cl2N2O•HCl | 1 g/5 g |
- Maprotiline HCl
Maprotiline is an inhibitor of norepinephrine reuptake and has been used clinically as an antidepressant.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-200156 | 10347-81-6 | C20H23N ·HCl | 1 g |
- Medetomidine hydrochloride
A potent α2-adrenoceptor agonist. Shows greater selectivity over α1-adrenoceptors than clonidine and UK 14,304.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-204073 | 106807-72-1 | C13H16N2.HCl | 10 mg/50 mg |
- Metoprolol Tartrate
A β1-adrenoceptor antagonist.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-205751 | 56392-17-7 | C34H56N2O12 | 5 g/25 g |
- Naftopidil hydrochloride
An α1-adrenoceptor antagonist with weak antagonism at post-junctional α2 receptors. Antihypertensive and vasodilating.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-203151 | 57149-07-2 | C24H28N2O3 ·HCl | 10 mg/50 mg |
- Naphazoline Hydrochloride
This compound produces inotropic effects via a-adrenoceptor stimulation.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-205764 | 550-99-2 | C14H14N2 ·• HCl | 25 g/100 g |
- Naphazoline Nitrate
Produces inotropic effects via a-adrenoceptor stimulation.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-205765 | 5144-52-5 | C14H14N2.HNO3 | 10 g/25 g |
- (-)-Nebivolol
A β1-Adrenergic blocker. Used as an antihypertensive.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-212366 | 118457-16-2 | C22H25F2NO4 | 1 mg |
- (+)-Nebivolol
A β-Adrenergic blocker. Used as an antihypertensive.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-212367 | 118457-15-1 | C22H25F2NO4 | 1 mg |
- Nebivolol hydrochloride
A highly selective antagonist of the β1-adrenoceptor. Produces vasodilation through induction of NO production mediated by β3-adrenoceptor agonism.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-204122 | 152520-56-4 | C22H25F2NO4•HCl | 10 mg/50 mg |
- Nicergoline
α-adrenergic, vasodilator. Cognitive enhancer.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-203643 | 27848-84-6 | C24H26BrN3O3 | 100 mg |
- Nisoxetine hydrochloride
Selective and potent inhibitor of noradrenalin uptake with little or no affinity for a range of other neurotransmitter receptors.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-203646 | 57754-86-6 | C17H21NO2 ·HCl | 10 mg/50 mg |
- NPEC-caged-noradrenalin
| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-361279 | n.n. | C17H18N2O7 | 10 mg/50 mg |
- Octopamine Hydrochloride
An adrenoceptor agonist which stimulates lipolysis in mammalian adipocytes via activation of β3 receptors.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-203168 | 770-05-8 | C8H11NO2 ·HCl | 1 g/1 g |
- Oxprenolol hydrochloride
A non-selective β-adrenergic inhibitor that also displays intrinsic sympathomimetic activity. Shown to also stabilize cellular membranes.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-204152 | 6452-73-9 | C15H23NO3 ·HCl | 100 mg |
- Oxymetazoline Hydrochloride
Partial α2A adrenoceptor agonist and α1A agonist. Agonist/antagonist activity at 5-HT receptors.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-203172 | 2315-02-8 | C16H24N2O ·HCl | 5 g/25 g |
- p-Aminoclonidine
Adrenergic receptor (alpha 2) agonist| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-296001 | 73217-88-6 | C9H10Cl2N4•HCl | 1 mg/5 mg |
- Phentolamine Hydrochloride
An a-Adrenergic blocker.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-205802 | 73-05-2 | C17H19N3O ·HCl | 50 mg/100 mg |
- Phentolamine mesylate
α-Adrenergic blocker.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-205803 | 65-28-1 | C17H19N3O ·CH3SO3H | 50 mg/100 mg |
- Pindolol
Serotonin 5-HT1A/1B receptor antagonist, with roughly equal affinity for each subtype. Partial agonist at mouse and human β3-adrenoceptors. | Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-204847 | 13523-86-9 | C14H20N2O2 | 100 mg |
- Prazosin hydrochloride
An adrenergic α, α2B-adrenoceptor and a potent melatonin MT3 receptor antagonist.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-204858 | 19237-84-4 | C19H21N5O4 ·HCl | 100 mg |
- Procaterol hydrochloride
Specific and very potent β2 agonist.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-203667 | 62929-91-3 | C16H22N2O3•HCl | 10 mg/50 mg |
- Propranolol glycol
Metabolite of propranolol.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-204214 | 36112-95-5 | C13H14O3 | 100 mg |
- (R)-(-)-Niguldipine hydrochloride
Less active enantiomer of (S)-(+)-Niguldipine hydrochloride| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-203676 | 113145-70-3 | C36H39N3O6.HCl | 10 mg/50 mg |
- (R)-(-)-Phenylephrine hydrochloride
Phenylephrine (PE) is an α1-adrenoceptor agonist that promotes hypertrophic growth in the ventricular myocytes, and activates several MAPK signaling pathways.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-203677 | 61-76-7 | C9H13NO2 ·HCl | 100 mg |
- (R)-(+)-m-Nitrobiphenyline oxalate
α2C-adrenoceptor agonist that potently inhibits cAMP accumulation in CHO cells (EC50 = 38 nM). | Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-204226 | n.n. | C17H17N3O3 ·C2H2O4 | 10 mg/50 mg |
- (R)-(+)-Propranolol hydrochloride
Less active enantiomer.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-203678 | 5051-22-9 | C16H21NO2 ·HCl | 100 mg/1 g |
- (R)-Bufuralol Hydrochloride
R-Enantiomer of Bufuralol which is a Beta-Adrenergic blocker with peripheral vasodilating activity. Categorized as an antianginal, as well as antihypertensive.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-212681 | 57704-11-7 | C16H24ClNO2 | 1 mg |
- Ractopamine hydrochloride
An adrenergic beta-agonist which increases muscle mass and decreases body fat in lifestock and rodents.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-205832 | 90274-24-1 | C18H23NO3•HCl | 1 g/5 g |
- Rauwolscine • HCl
α2-Adrenergic receptor antagonist.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-200151 | 6211-32-1 | C21H26N2O3 ·HCl | 100 mg |
- Reboxetine mesylate
An effective noradrenalin uptake inhibitor.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-204232 | 71620-89-8 | C19H23NO3 ·CH3SO3H | 10 mg/50 mg |
- Rec 15/2615 dihydrochloride
Selective α1B-adrenoceptor antagonist (Ki values are 0.3, 1.9 and 2.6 nM at human α1B, α1A and α1D receptors respectively).| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-204233 | 173059-17-1 | C26H33N5O5 ·2HCl | 10 mg/50 mg |
- Reserpine
An inhibitor of biogenic amine transport into synaptic vesicles and adrenal chromaffin granules. More specifically shown to interfere with dopamine transporter activity.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-203370 | 50-55-5 | C33H40N2O9 | 1 g |
- Rilmenidine hemifumarate
| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-203680 | 207572-68-7 | C10H16N2O ·½C4H4O4 | 10 mg/50 mg |
- Ritodrine
β2-adrenoceptor agonist; relaxes uterine muscle contraction. Used to stop premature labor.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-204882 | 23239-51-2 | C17H21NO3.HCl | 250 mg/1 g |
- RS 17053 hydrochloride
| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-361312 | 169505-93-5 | C24H29N2O2Cl.HCl | 10 mg/50 mg |
- RS 79948 hydrochloride
| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-361318 | 186002-54-0 | C19H28N2O3S.HCl | 10 mg/50 mg |
- RS 100329 hydrochloride
| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-361309 | 232953-52-5 | C20H25F3N4O3.HCl | 10 mg/50 mg |
- (RS)-Atenolol
Cardioselective β-adrenergic blocker. Antihypertensive, antianginal, antiarrhythmic.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-204895 | 29122-68-7 | C14H22N2O3 | 1 g |
- RX 821002 hydrochloride
Selective α2-adrenoceptor antagonist with low affinity for imidazoline sites. Selective for the α2D over the α2A subtypes. | Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-203686 | 102575-24-6 | C12H14N2O3 ·HCl | 10 mg/50 mg |
- S-(-)-Atenolol
Active enantiomer of atenolol.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-203687 | 93379-54-5 | C14H22N2O3 | 10 mg/50 mg |
- S-(+)-Niguldipine hydrochloride
Extremely potent (picomolar range) inhibitor of α1A-adrenergic receptors and L-type Ca2+ channels.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-203248 | 113165-32-5 | C36H39N3O6.HCl | 5 mg |
- S(-)-Propranolol • HCl
A β-Adrenergic receptor antagonist and the active isomer of (±)-Propranolol preparations.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-200153 | 4199-10-4 | C16H21NO2 ·HCl | 100 mg |
- (S)-(-)-Pindolol
More active enantiomer of pindolol.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-203688 | 26328-11-0 | C14H20N2O2 | 10 mg/50 mg |
- (S)-Bufuralol Hydrochloride
R-Enantiomer of Bufuralol which is a Beta-Adrenergic blocker with peripheral vasodilating activity. | Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-212877 | 57704-10-6 | C16H24ClNO2 | 1 mg |
- Salbutamol hemisulfate
Non-selective β-adrenergic agonist, more potent at β2 than β1 receptors.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-203373 | 51022-70-9 | (C13H21NO3)2.H2SO4 | 250 mg |
- Salmeterol
Potent and selective β2-adrenoceptor agonist (EC50 = 5.3 nM); bronchodilator. | Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-224277 | 89365-50-4 | C25H37NO4 | 10 mg/50 mg |
- SDZ 21009
b-adrenoceptor antagonist. Also 5-HT1A/1Bantagonist| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-203695 | 39731-05-0 | C19H28N2O4 | 10 mg/50 mg |
- SNAP 5089
| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-204290 | 157066-76-7 | C36H40N4O5•HCl•xH2O | 10 mg/50 mg |
- Sotalol hydrochloride
A compound with a mechanism of action that prolongs the action potential and refraction of cardiac tissue through non-selective yet potent β-adronergic blocking activity.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-203699 | 959-24-0 | C12H20N2O3S ·HCl | 10 mg/50 mg |
- SR 58611A
| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-361365 | 121524-09-2 | C22H26ClNO4.HCl | 10 mg/50 mg |
- SR 59230A hydrochloride
Potent and selective β3 antagonist adrenoceptor (IC50 values are 40, 408 and 648 nM for β3, β1 and β2 receptors respectively). Orally active in vivo.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-204302 | 174689-39-5 | C21H27NO2•HCl | 10 mg/50 mg |
- ST 91
α2-adrenoceptor agonist that does not cross the blood brain barrier. | Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-203703 | 4749-61-5 | C13H19N3 ·HCl | 10 mg/50 mg |
- Terazosin hydrochloride
| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-204337 | 63074-08-8 | C19H25N5O4•HCl | 50 mg |
- Terbutaline
A beta-adrenoceptor agonist used to treat asthma and premature labor. | Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-204911 | 23031-25-6 | C12H19NO3 | 1 g/5 g |
- Terbutaline Hemisulfate Salt
A B-Adrenergic receptor agonist and a Bronchodilator.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-213000 | 23031-32-5 | C12H19NO3•1/2H2SO4 | 2 g |
- Timolol Maleate
A β-Adrenergic receptor selective antagonist used as an antiglaucoma agent.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-203297 | 26921-17-5 | C13H24N4O3S.C4H4O4 | 100 mg/250 mg |
- Tizanidine • HCl
α2-Adrenergic receptor agonist. Displays affinity for the I1-imidazoline receptor. Spasmolytic activity.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-200148 | 64461-82-1 | C9H8ClN5S ·HCl | 100 mg/500 mg |
- Tomoxetine hydrochloride
A competitive and specific inhibitor of norepinephrine reuptake while demonstrating weak serotonin and dopamine inhibition.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-204349 | 82248-59-7 | C17H21NO ·HCl | 10 mg/50 mg |
- Tulobuterol
A β-adrenergic receptor agonist that is related structurally to Terbutaline.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-213131 | 41570-61-0 | C12H18ClNO | 100 mg |
- UK 14,304
Full α2 adrenergic agonist. Centrally active following systemic administration in vivo.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-204373 | 59803-98-4 | C11H10BrN5 | 10 mg/50 mg |
- UK 14,304 tartrate
Water-soluble form UK 14,304. Centrally active following systemic administration in vivo. Full α2 adrenergic agonist.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-204374 | 59803-99-5 | C11H10BrN5 ·C4H6O6 | 10 mg/50 mg |
- Urapidil HCl
Adrenergic α1 receptor antagonist. Serotonin 5-HT1A receptor agonist. Clinically useful antihypertensive agent.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-200155 | 64887-14-5 | C20H29N5O3··HCl | 100 mg |
- WB 4101 hydrochloride
α1A-adrenergic selective antagonist.| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-204394 | 613-67-2 | C19H23NO5.HCl | 25 mg |
- Xamoterol hemifumarate
| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-361406 | 73210-73-8 | C16H25N3O5 ·0.5C4H4O4 | 10 mg/50 mg |
- Yohimbine hydrochloride
α2-adrenoceptor antagonist (pKi values are 8.52, 8.00 and 9.17 for human a2A, a2B and a2C receptors respectively).| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-204412 | 65-19-0 | C21H26N2O3•HCl | 1 g |
- ZD 2079
| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-361416 | 178600-17-4 | C18H21NO4.HCl | 10 mg/50 mg |
- ZD 7114 hydrochloride
| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-361417 | 129689-30-1 | C22H30N2O6.HCl | 10 mg/50 mg |
- Zinterol hydrochloride
| Katalog # | CAS Nummer | Summenformel | Menge |
|---|
| sc-204418 | 37000-20-7 | C19H26N2O4S ·HCl | 10 mg/50 mg |
|